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Cariprazine, a new, orally active dopamine D2/3 receptor partial agonist for the treatment of schizophrenia, bipolar mania and depression

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Pages 1141-1159 | Published online: 09 Jan 2014

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Rui-Xiang Yuan, Jun-Wei Xu, Lian-Hua Song, Yang-Li Qi, Hong Mou, Jian-Wei Wu, Ke-Yu Jiang & Xiao-Wen Chen. (2021) A convenient and practical synthesis of the cis isomer of the first orally active dopamine D3-Preferring D3-D2 receptor partial agonist cariprazine. Synthetic Communications 51:14, pages 2127-2134.
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Felix-Martin Werner & Rafael Coveñas. (2015) New developments in the management of schizophrenia and bipolar disorder: potential use of cariprazine. Therapeutics and Clinical Risk Management 11, pages 1657-1661.
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H. Javelot. (2016) Psychopharmacologie de l’anxiété et de la dépression : aspects historiques, traitements actuels et perspectives. Annales Pharmaceutiques Françaises 74:2, pages 93-118.
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