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Original Research

Non-imidazole-based histamine H3 receptor antagonists with anticonvulsant activity in different seizure models in male adult rats

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Pages 3879-3898 | Published online: 25 Nov 2016

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Salim M Bastaki, Yousef M Abdulrazzaq, Mohamed Shafiullah, Małgorzata Więcek, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2018) Anticonvulsant and reproductive toxicological studies of the imidazole-based histamine H3R antagonist 2-18 in mice. Drug Design, Development and Therapy 12, pages 179-194.
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Articles from other publishers (24)

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Małgorzata Anna Marć, Enrique Domínguez-Álvarez, Gniewomir Latacz, Agata Doroz-Płonka, Carmen Sanmartín, Gabriella Spengler & Jadwiga Handzlik. (2022) Pharmaceutical and Safety Profile Evaluation of Novel Selenocompounds with Noteworthy Anticancer Activity. Pharmaceutics 14:2, pages 367.
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Lin Yang, Yi Wang & Zhong Chen. (2021) Central histaminergic signalling, neural excitability and epilepsy. British Journal of Pharmacology 179:1, pages 3-22.
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Justyna Godyń, Paula Zaręba, Dorota Łażewska, Dorota Stary, David Reiner-Link, Annika Frank, Gniewomir Latacz, Szczepan Mogilski, Maria Kaleta, Agata Doroz-Płonka, Annamaria Lubelska, Ewelina Honkisz-Orzechowska, Agnieszka Olejarz-Maciej, Jadwiga Handzlik, Holger Stark, Katarzyna Kieć-Kononowicz, Barbara Malawska & Marek Bajda. (2021) Cyanobiphenyls: Novel H3 receptor ligands with cholinesterase and MAO B inhibitory activity as multitarget compounds for potential treatment of Alzheimer’s disease. Bioorganic Chemistry 114, pages 105129.
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Nermin Eissa, Adel Sadeq, Astrid Sasse & Bassem Sadek. (2020) Role of Neuroinflammation in Autism Spectrum Disorder and the Emergence of Brain Histaminergic System. Lessons Also for BPSD?. Frontiers in Pharmacology 11.
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Alaa Alachkar, Shreesh K. Ojha, Adel Sadeq, Abdu Adem, Annika Frank, Holger Stark & Bassem Sadek. (2020) Experimental Models for the Discovery of Novel Anticonvulsant Drugs: Focus on Pentylenetetrazole-Induced Seizures and Associated Memory Deficits. Current Pharmaceutical Design 26:15, pages 1693-1711.
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Pakhuri Mehta, Przemysław Miszta, Przemysław Rzodkiewicz, Olga Michalak, Piotr Krzeczyński & Sławomir Filipek. (2020) Enigmatic Histamine Receptor H4 for Potential Treatment of Multiple Inflammatory, Autoimmune, and Related Diseases. Life 10:4, pages 50.
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Azadeh Yazdi, Mohammadmahdi Doostmohammadi, Farshid Pourhossein Majarshin & Siamak Beheshti. (2020) Betahistine, prevents kindling, ameliorates the behavioral comorbidities and neurodegeneration induced by pentylenetetrazole. Epilepsy & Behavior 105, pages 106956.
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Alaa Alachkar, Sheikh Azimullah, Mohamed Lotfy, Ernest Adeghate, Shreesh K. Ojha, Rami Beiram, Dorota Łażewska, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2020) Antagonism of Histamine H3 receptors Alleviates Pentylenetetrazole-Induced Kindling and Associated Memory Deficits by Mitigating Oxidative Stress, Central Neurotransmitters, and c-Fos Protein Expression in Rats. Molecules 25:7, pages 1575.
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Alaa Alachkar, Sheikh Azimullah, Shreesh K. Ojha, Rami Beiram, Dorota Łażewska, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2019) The Neuroprotective Effects of Histamine H3 Receptor Antagonist E177 on Pilocarpine-Induced Status Epilepticus in Rats. Molecules 24:22, pages 4106.
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Salim M. A. Bastaki, Naheed Amir, Małgorzata Więcek, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2019) Influence of the Novel Histamine H3 Receptor Antagonist/Inverse Agonist M39 on Gastroprotection and PGE2 Production Induced by (R)-Alpha-Methylhistamine in C57BL/6 Mice. Frontiers in Pharmacology 10.
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Alaa Alachkar, Dorota Łażewska, Gniewomir Latacz, Annika Frank, Agata Siwek, Annamaria Lubelska, Ewelina Honkisz-Orzechowska, Jadwiga Handzlik, Holger Stark, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2018) Studies on Anticonvulsant Effects of Novel Histamine H3R Antagonists in Electrically and Chemically Induced Seizures in Rats. International Journal of Molecular Sciences 19:11, pages 3386.
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Alaa Alachkar, Gniewomir Latacz, Agata Siwek, Annamaria Lubelska, Ewelina Honkisz, Anna Gryboś, Dorota Łażewska, Jadwiga Handzlik, Holger Stark, Katarzyna Kiec-Kononowicz & Bassem Sadek. (2018) Anticonvulsant evaluation of novel non-imidazole histamine H3R antagonists in different convulsion models in rats. Pharmacology Biochemistry and Behavior 170, pages 14-24.
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Katarzyna Szczepańska, Tadeusz Karcz, Szczepan Mogilski, Agata Siwek, Kamil J. Kuder, Gniewomir Latacz, Monika Kubacka, Stefanie Hagenow, Annamaria Lubelska, Agnieszka Olejarz, Magdalena Kotańska, Bassem Sadek, Holger Stark & Katarzyna Kieć-Kononowicz. (2018) Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H3R ligands. European Journal of Medicinal Chemistry 152, pages 223-234.
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Michał Abram, Mirosław Zagaja, Szczepan Mogilski, Marta Andres-Mach, Gniewomir Latacz, Sebastian Baś, Jarogniew J. Łuszczki, Katarzyna Kieć-Kononowicz & Krzysztof Kamiński. (2017) Multifunctional Hybrid Compounds Derived from 2-(2,5-Dioxopyrrolidin-1-yl)-3-methoxypropanamides with Anticonvulsant and Antinociceptive Properties. Journal of Medicinal Chemistry 60:20, pages 8565-8579.
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Alaa Alachkar, Dorota Łażewska, Katarzyna Kieć-Kononowicz & Bassem Sadek. (2017) The Histamine H3 Receptor Antagonist E159 Reverses Memory Deficits Induced by Dizocilpine in Passive Avoidance and Novel Object Recognition Paradigm in Rats. Frontiers in Pharmacology 8.
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Antonella Pisera‐Fuster, Sofía Otero, Alan Talevi, Luis Bruno‐Blanch & Ramón Bernabeu. (2017) Anticonvulsant effect of sodium cyclamate and propylparaben on pentylenetetrazol‐induced seizures in zebrafish. Synapse 71:4.
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