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Original Research

Comprehensive kinase profile of pacritinib, a nonmyelosuppressive Janus kinase 2 inhibitor

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Pages 11-19 | Published online: 16 Aug 2016

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Read on this site (10)

Naveen Pemmaraju, Prithviraj Bose, Raajit Rampal, Aaron T. Gerds, Angela Fleischman & Srdan Verstovsek. (2023) Ten years after ruxolitinib approval for myelofibrosis: a review of clinical efficacy. Leukemia & Lymphoma 64:6, pages 1063-1081.
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Khalil Saleh & Vincent Ribrag. (2023) An evaluation of fedratinib for adult patients with newly diagnosed and previously treated myelofibrosis. Expert Review of Hematology 16:4, pages 227-236.
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John Mascarenhas. (2022) Pacritinib for the treatment of patients with myelofibrosis and thrombocytopenia. Expert Review of Hematology 15:8, pages 671-684.
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Prithviraj Bose & Ruben A. Mesa. (2022) Novel strategies for challenging scenarios encountered in managing myelofibrosis. Leukemia & Lymphoma 63:4, pages 774-788.
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Giacomo Coltro & Alessandro M. Vannucchi. (2021) The safety of JAK kinase inhibitors for the treatment of myelofibrosis. Expert Opinion on Drug Safety 20:2, pages 139-154.
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Jan Philipp Bewersdorf, Sara Mohamed Jaszczur, Salma Afifi, Jennifer C Zhao & Amer M Zeidan. (2019) Beyond Ruxolitinib: Fedratinib and Other Emergent Treatment Options for Myelofibrosis. Cancer Management and Research 11, pages 10777-10790.
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Suliman Al-Fayoumi, Taishi Hashiguchi, Yuka Shirakata, John Mascarenhas & Jack W Singer. (2018) Pilot study of the antifibrotic effects of the multikinase inhibitor pacritinib in a mouse model of liver fibrosis. Journal of Experimental Pharmacology 10, pages 9-17.
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Douglas Tremblay & John Mascarenhas. (2018) Pacritinib to treat myelofibrosis patients with thrombocytopenia. Expert Review of Hematology 11:9, pages 707-714.
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Prithviraj Bose, Abdallah Abou Zahr & Srdan Verstovsek. (2017) Investigational Janus kinase inhibitors in development for myelofibrosis. Expert Opinion on Investigational Drugs 26:6, pages 723-734.
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Tania Jain & Ruben Mesa. (2016) The development, safety and efficacy of pacritinib for the treatment of myelofibrosis. Expert Review of Anticancer Therapy 16:11, pages 1101-1108.
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