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Xenobiotica
the fate of foreign compounds in biological systems
Volume 42, 2012 - Issue 5
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General Xenobiochemistry

Effect of voriconazole and other azole antifungal agents on CYP3A activity and metabolism of tacrolimus in human liver microsomes

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Pages 409-416 | Received 11 Aug 2011, Accepted 09 Oct 2011, Published online: 22 Nov 2011

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Josefine Schulz, Franziska Kluwe, Gerd Mikus, Robin Michelet & Charlotte Kloft. (2019) Novel insights into the complex pharmacokinetics of voriconazole: a review of its metabolism. Drug Metabolism Reviews 51:3, pages 247-265.
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Xingxian Luo, Taifeng Li, Ze Yu, Xuecai Xue, Haiyang Zhao, Na li, Liping Ma, Changqing Yang, Lin Huang & Wanyu Feng. (2019) The impact of azole antifungal drugs on imatinib metabolism in human liver microsomes. Xenobiotica 49:7, pages 753-761.
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Dan Lou, Xiao Cui, Su-Su Bao, Wei Sun, Wen-He Pan, Meng-Chun Chen, Yao-Yao Dong, Guo-Xin Hu, Rui-Jie Chen & Zhe Wang. (2019) Effects of ketoconazole, voriconazole, and itraconazole on the pharmacokinetics of apatinib in rats. Drug Development and Industrial Pharmacy 45:4, pages 689-693.
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Li Wang, Shuanghu Wang, Mengchun Chen, Xinxin Chen, Yuxian Lin, Xiaoxia Hu, Xiangxin Huang, Xiangyu Li & Guoxin Hu. (2015) Inhibitory effect of ketoconazole and voriconazole on the pharmacokinetics of carvedilol in rats. Drug Development and Industrial Pharmacy 41:10, pages 1661-1666.
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Gaotong Lin, Chenming Wang, Xiangjun Qiu, Zhe Wang, Anyue Han, Tao Xu, Xin Kan & Guoxin Hu. (2014) Differential effects of ketoconazole, itraconazole and voriconazole on the pharmacokinetics of imatinib and its main metabolite GCP74588 in rat. Drug Development and Industrial Pharmacy 40:12, pages 1616-1622.
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Juan Cai & Rongwei Shi. (2023) Exploration of the binding of antifungal drugs to human P450 2C9 based on docking and molecular dynamics simulation . International Journal of Quantum Chemistry 123:14.
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Tianrong Xun, Yan Rong, Bin Lv, Jinfei Tian, Qing Zhang & Xixiao Yang. (2023) Interaction and potential mechanisms between atorvastatin and voriconazole, agents used to treat dyslipidemia and fungal infections. Frontiers in Pharmacology 14.
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Ranita Kirubakaran, David W. Uster, Stefanie Hennig, Jane E. Carland, Richard O. Day, Sebastian G. Wicha & Sophie L. Stocker. (2022) Adaptation of a population pharmacokinetic model to inform tacrolimus therapy in heart transplant recipients. British Journal of Clinical Pharmacology 89:3, pages 1162-1175.
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Zhi-Ping Jin, Miao Yan, Si-Ze Li, Bao-Qing Wang, Qing Xu, Wei Wu, Xiao-Yu Li, Qian-Zhou Lv & Xiao-Qiang Xiang. (2023) Prediction of the Impact of CYP2C19 Polymorphism on Drug-Drug Interaction between Voriconazole and Tacrolimus Using Physiologically-Based Pharmacokinetic Modelling. Brazilian Journal of Pharmaceutical Sciences 59.
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Yuhao Fu, Ying Li, Yinling Ma, Xueru He, Xuejiao Xun, Yanjun Cui, Liju Fan & Zhanjun Dong. (2022) Effects of voriconazole and fluconazole on the pharmacokinetics of almonertinib in rats by UPLC–MS/MS. Biomedical Chromatography 37:1.
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Xiao Huang, Ying Zhou, Jing Zhang, Hongping Xiang, Hao Mei, Li Liu, Lu Tong, Fang Zeng, Yifei Huang, Hong Zhou & Yu Zhang. (2022) The importance of CYP2C19 genotype in tacrolimus dose optimization when concomitant with voriconazole in heart transplant recipients . British Journal of Clinical Pharmacology 88:10, pages 4515-4525.
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Xingxian Luo, Xuecai Xue, Taifeng Li, Ying Zhang, Lin Huang & Gang Cheng. (2020) Differential Impacts of Azole Antifungal Drugs on the Pharmacokinetic Profiles of Dasatinib in Rats by LC-MS-MS. Current Drug Metabolism 21:13, pages 1022-1030.
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Jiake He, Yang Yu, Chenglong Yin, Hailang Liu, Hua Zou, Jingsheng Ma, Wentao Yang, Ye Liu, Lin Zhong & Xijing Chen. (2019) Clinically significant drug‐drug interaction between tacrolimus and fluconazole in stable renal transplant recipient and literature review. Journal of Clinical Pharmacy and Therapeutics 45:2, pages 264-269.
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Ahmed M. Alkhunaizi, Ali M. Bazzi, Ali A. Rabaan & Elwaleed A. Ahmed. (2018) Fusarium Infection in a Kidney Transplant Recipient Successfully Treated with Voriconazole . Case Reports in Infectious Diseases 2018, pages 1-4.
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