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Çiğdem Bilen, Serap Beyaztaş, Oktay Arslan & Özen Özensoy Güler. (2013) Investigation of heavy metal effects on immobilized paraoxanase by glutaraldehyde. Journal of Enzyme Inhibition and Medicinal Chemistry 28:3, pages 440-446.
Read now
Read now
Wendy A Lea & Anton Simeonov. (2011) Fluorescence polarization assays in small molecule screening. Expert Opinion on Drug Discovery 6:1, pages 17-32.
Read now
Read now
Daisy Lin, Tatyana V. Pestova, Christopher U. T. Hellen & Henri Tiedge. (2008) Translational Control by a Small RNA: Dendritic BC1 RNA Targets the Eukaryotic Initiation Factor 4A Helicase Mechanism. Molecular and Cellular Biology 28:9, pages 3008-3019.
Read now
Read now
DJ McLoughlin, F Bertelli & C Williams. (2007) The A, B, Cs of G-protein-coupled receptor pharmacology in assay development for HTS. Expert Opinion on Drug Discovery 2:5, pages 603-619.
Read now
Read now
Sophie E. Schlumberger, Yumiko Saito, Thomas Giller, Edith Hintermann, Heidi Tanner, Verena Jäggin, Urs Zumsteg, Olivier Civelli & Alex N. Eberle. (2003) Different Structural Requirements for Melanin‐Concentrating Hormone (MCH) Interacting with Rat MCH‐R1 (SLC‐1) and Mouse B16 Cell MCH‐R. Journal of Receptors and Signal Transduction 23:1, pages 69-81.
Read now
Read now
Alex N. Eberle, Jószef Bódi, György Orosz, Helga Süli-Vargha, Verena Jäggin & Urs Zumsteg. (2001) ANTAGONIST AND AGONIST ACTIVITIES OF THE MOUSE AGOUTI PROTEIN FRAGMENT (91–131) AT THE MELANOCORTIN-1 RECEPTOR. Journal of Receptors and Signal Transduction 21:1, pages 25-45.
Read now
Read now
Krishnendu Ghosh, Emily S. Shen, Brian J. Arey & Francisco J. López. (1998) A global model to define the behavior of partial agonists (bell-shaped dose-response inducers) in pharmacological evaluation of activity in the presence of the full agonist. Journal of Biopharmaceutical Statistics 8:4, pages 645-665.
Read now
Read now
V. Pliska. (1995) Minireview: Multiple receptor populations: Binding isotherms and their numerical analysis. Journal of Receptors and Signal Transduction 15:1-4, pages 651-675.
Read now
Read now
Articles from other publishers (85)
David J. Fallon, Alex Phillipou, Christopher J. Schofield, David House, Nicholas C. O. Tomkinson & Jacob T. Bush. (2023) Photoaffinity labelling displacement assay using multiple recombinant protein domains. Biochemical Journal 480:15, pages 1183-1197.
Crossref
Crossref
Ryo C. Yanagita, Mao Otani, Satoshi Hatanaka, Hiroto Nishi, Shota Miyake, Yusuke Hanaki, Masashi Sato, Yasuhiro Kawanami & Kazuhiro Irie. (2022) Analysis of binding mode of vibsanin A with protein kinase C C1 domains: An experimental and molecular dynamics simulation study. Journal of Molecular Structure 1260, pages 132866.
Crossref
Crossref
Jeung- Ha, Xin Yu, Darren Carpizo & Stewart Loh. (2021) Urea Denaturation, Zinc Binding, and DNA Binding Assays of Mutant p53 DNA-binding Domains and Full-length Proteins. BIO-PROTOCOL 11:20.
Crossref
Crossref
Geoffrey A. Holdgate & Paul E. Hemsley. 2021. Protein-Ligand Interactions. Protein-Ligand Interactions
231
246
.
Adam R Blanden, Xin Yu, Alan J Blayney, Christopher Demas, Jeung-Hoi Ha, Yue Liu, Tracy Withers, Darren R Carpizo & Stewart N Loh. (2020) Zinc shapes the folding landscape of p53 and establishes a pathway for reactivating structurally diverse cancer mutants. eLife 9.
Crossref
Crossref
Mollie M. Jurewicz, Richard A. Willis, Vasanthi Ramachandiran, John D. Altman & Lawrence J. Stern. (2019) MHC-I peptide binding activity assessed by exchange after cleavage of peptide covalently linked to β2-microglobulin. Analytical Biochemistry 584, pages 113328.
Crossref
Crossref
David Reiner & Holger Stark. (2019) Ligand binding kinetics at histamine H3 receptors by fluorescence-polarization with real-time monitoring. European Journal of Pharmacology 848, pages 112-120.
Crossref
Crossref
Amy E. McGrath, Alexander P. Martyn, Louise R. Whittell, Fay E. Dawes, Jennifer L. Beck, Nicholas E. Dixon, Michael J. Kelso & Aaron J. Oakley. (2018) Crystal structures and biochemical characterization of DNA sliding clamps from three Gram-negative bacterial pathogens. Journal of Structural Biology 204:3, pages 396-405.
Crossref
Crossref
Linna An, Dillon P. Cogan, Claudio D. Navo, Gonzalo Jiménez-Osés, Satish K. Nair & Wilfred A. van der Donk. (2018) Substrate-assisted enzymatic formation of lysinoalanine in duramycin. Nature Chemical Biology 14:10, pages 928-933.
Crossref
Crossref
Xiaoling Puyang, Craig Furman, Guo Zhu Zheng, Zhenhua J. Wu, Deepti Banka, Kiran Aithal, Sergei Agoulnik, David M. Bolduc, Silvia Buonamici, Benjamin Caleb, Subhasree Das, Sean Eckley, Peter Fekkes, Ming-Hong Hao, Andrew Hart, René Houtman, Sean Irwin, Jaya J. Joshi, Craig Karr, Amy Kim, Namita Kumar, Pavan Kumar, Galina Kuznetsov, Weidong G. Lai, Nicholas Larsen, Crystal Mackenzie, Lesley-Ann Martin, Diana Melchers, Alyssa Moriarty, Tuong-Vi Nguyen, John Norris, Morgan O'Shea, Sunil Pancholi, Sudeep Prajapati, Sujatha Rajagopalan, Dominic J. Reynolds, Victoria Rimkunas, Nathalie Rioux, Ricardo Ribas, Amy Siu, Sasirekha Sivakumar, Vanitha Subramanian, Michael Thomas, Frédéric H. Vaillancourt, John Wang, Suzanne Wardell, Michael J. Wick, Shihua Yao, Lihua Yu, Markus Warmuth, Peter G. Smith, Ping Zhu & Manav Korpal. (2018) Discovery of Selective Estrogen Receptor Covalent Antagonists for the Treatment of ERαWT and ERαMUT Breast Cancer. Cancer Discovery 8:9, pages 1176-1193.
Crossref
Crossref
Brittany J. Carr, Koichiro Mihara, Rithwik Ramachandran, Mahmoud Saifeddine, Neil M. Nathanson, William K. Stell & Morley D. Hollenberg. (2018)
Myopia-Inhibiting Concentrations of Muscarinic Receptor Antagonists Block Activation of Alpha
2A
-Adrenoceptors In Vitro
. Investigative Opthalmology & Visual Science 59:7, pages 2778.
Crossref
Crossref
Nicola E. A. Chessum, Swee Y. Sharp, John J. Caldwell, A. Elisa Pasqua, Birgit Wilding, Giampiero Colombano, Ian Collins, Bugra Ozer, Meirion Richards, Martin Rowlands, Mark Stubbs, Rosemary Burke, P. Craig McAndrew, Paul A. Clarke, Paul Workman, Matthew D. Cheeseman & Keith Jones. (2018) Demonstrating In-Cell Target Engagement Using a Pirin Protein Degradation Probe (CCT367766). Journal of Medicinal Chemistry 61:3, pages 918-933.
Crossref
Crossref
Geoffrey A. Holdgate, Thomas D. Meek & Rachel L. Grimley. (2017) Mechanistic enzymology in drug discovery: a fresh perspective. Nature Reviews Drug Discovery 17:2, pages 115-132.
Crossref
Crossref
Angela F. Ku & Gregory D. Cuny. (2018) Discovery of 7-hydroxyaporphines as conformationally restricted ligands for beta-1 and beta-2 adrenergic receptors. MedChemComm 9:2, pages 353-356.
Crossref
Crossref
Mark Hedglin, Mahesh Aitha & Stephen J. Benkovic. (2017) Monitoring the Retention of Human Proliferating Cell Nuclear Antigen at Primer/Template Junctions by Proteins That Bind Single-Stranded DNA. Biochemistry 56:27, pages 3415-3421.
Crossref
Crossref
Mark Hedglin, Binod Pandey & Stephen J Benkovic. (2016) Characterization of human translesion DNA synthesis across a UV-induced DNA lesion. eLife 5.
Crossref
Crossref
Juan Zhen, Tamara Antonio, Joanna C. Jacob, David K. Grandy, Maarten E. A. Reith, Aloke K. Dutta & Dana E. Selley. (2015) Efficacy of Hybrid Tetrahydrobenzo[d]thiazole Based Aryl Piperazines D-264 and D-301 at D2 and D3 Receptors. Neurochemical Research 41:1-2, pages 328-339.
Crossref
Crossref
Xing Du, Yi Li, Yuan-Ling Xia, Shi-Meng Ai, Jing Liang, Peng Sang, Xing-Lai Ji & Shu-Qun Liu. (2016) Insights into Protein–Ligand Interactions: Mechanisms, Models, and Methods. International Journal of Molecular Sciences 17:2, pages 144.
Crossref
Crossref
Hamid R. Nasiri, Sandra Linge & Dirk Ullmann. (2016) Thermodynamic profiling of inhibitors of Nrf2:Keap1 interactions. Bioorganic & Medicinal Chemistry Letters 26:2, pages 526-529.
Crossref
Crossref
Hubert Rehm & Thomas LetzelHubert Rehm & Thomas Letzel. 2016. Der Experimentator: Proteinbiochemie/Proteomics. Der Experimentator: Proteinbiochemie/Proteomics
37
113
.
Eric R. Prossnitz & Jeffrey B. Arterburn. (2015) International Union of Basic and Clinical Pharmacology. XCVII. G Protein–Coupled Estrogen Receptor and Its Pharmacologic Modulators. Pharmacological Reviews 67:3, pages 505-540.
Crossref
Crossref
Juan Zhen, Tamara Antonio, Solav Ali, Kim A. Neve, Aloke K. Dutta & Maarten E.A. Reith. (2015) Use of radiolabeled antagonist assays for assessing agonism at D2 and D3 dopamine receptors: Comparison with functional GTPγS assays. Journal of Neuroscience Methods 248, pages 7-15.
Crossref
Crossref
Liu Liu, Denzil Bernard & Shaomeng Wang. 2015. Protein-Protein Interactions. Protein-Protein Interactions
567
585
.
Xiangqian Kong, Limin Chen, Lianying Jiao, Xiangrui Jiang, Fulin Lian, Junyan Lu, Kongkai Zhu, Daohai Du, Jingqiu Liu, Hong Ding, Naixia Zhang, Jingshan Shen, Mingyue Zheng, Kaixian Chen, Xin Liu, Hualiang Jiang & Cheng Luo. (2014) Astemizole Arrests the Proliferation of Cancer Cells by Disrupting the EZH2-EED Interaction of Polycomb Repressive Complex 2. Journal of Medicinal Chemistry 57:22, pages 9512-9521.
Crossref
Crossref
Liusong Yin & Lawrence J. Stern. (2014) A novel method to measure HLA-DM-susceptibility of peptides bound to MHC class II molecules based on peptide binding competition assay and differential IC50 determination. Journal of Immunological Methods 406, pages 21-33.
Crossref
Crossref
Astrid M. Kral, Nicole Ozerova, Joshua Close, Joon Jung, Melissa Chenard, Judith Fleming, Brian B. Haines, Paul Harrington, John Maclean, Thomas A. Miller, Paul Secrist, Hongmei Wang & Richard W. HeidebrechtJr.Jr.. (2014) Divergent Kinetics Differentiate the Mechanism of Action of Two HDAC Inhibitors. Biochemistry 53:4, pages 725-734.
Crossref
Crossref
Mayako Michino, Prashant Donthamsetti, Thijs Beuming, Ashwini Banala, Lihua Duan, Thomas Roux, Yang Han, Eric Trinquet, Amy Hauck Newman, Jonathan A. Javitch & Lei Shi. (2013) A Single Glycine in Extracellular Loop 1 Is the Critical Determinant for Pharmacological Specificity of Dopamine D2 and D3 Receptors. Molecular Pharmacology 84:6, pages 854-864.
Crossref
Crossref
Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar & Richard A. Houghten. (2013) Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries. Molecular Pharmacology 84:3, pages 314-324.
Crossref
Crossref
Maya Lévy-Bimbot, Geneviève Major, Delphine Courilleau, Jean-Paul Blondeau & Yves Lévi. (2012) Tetrabromobisphenol-A disrupts thyroid hormone receptor alpha function in vitro: Use of fluorescence polarization to assay corepressor and coactivator peptide binding. Chemosphere 87:7, pages 782-788.
Crossref
Crossref
Eun Jeong Cho, Shuangluo Xia, Li-Chung Ma, Jon Robertus, Robert M. Krug, Eric V. Anslyn, Gaetano T. Montelione & Andrew D. Ellington. (2012) Identification of Influenza Virus Inhibitors Targeting NS1A Utilizing Fluorescence Polarization–Based High-Throughput Assay. SLAS Discovery 17:4, pages 448-459.
Crossref
Crossref
Ziyan Yuan, Eric A. Kumar, Stephen J. Campbell, Nicholas Y. Palermo, Smitha Kizhake, J. N. Mark Glover & Amarnath Natarajan. (2011) Exploiting the P-1 Pocket of BRCT Domains Toward a Structure Guided Inhibitor Design. ACS Medicinal Chemistry Letters 2:10, pages 764-767.
Crossref
Crossref
Holger Kubas, Martin Schäfer, Ulrike Bauder-Wüst, Matthias Eder, Dörte Oltmanns, Uwe Haberkorn, Walter Mier & Michael Eisenhut. (2010) Multivalent cyclic RGD ligands: influence of linker lengths on receptor binding. Nuclear Medicine and Biology 37:8, pages 885-891.
Crossref
Crossref
Tomonori Arai, Mai Yatabe, Megumi Furui, Hiroyuki Akatsuka, Masayoshi Uehata & Tsutomu Kamiyama. (2010) A fluorescence polarization-based assay for the identification and evaluation of calmodulin antagonists. Analytical Biochemistry 405:2, pages 147-152.
Crossref
Crossref
Tetyana Dodatko, Monique Akoachere, Nadia Jimenez, Zadkiel Alvarez & Ernesto Abel-Santos. (2010) Dissecting interactions between nucleosides and germination receptors in Bacillus cereus 569 spores. Microbiology 156:4, pages 1244-1255.
Crossref
Crossref
Juan Zhen, Tamara Antonio, Aloke K. Dutta & Maarten E.A. Reith. (2010) Concentration of receptor and ligand revisited in a modified receptor binding protocol for high-affinity radioligands: [3H]Spiperone binding to D2 and D3 dopamine receptors. Journal of Neuroscience Methods 188:1, pages 32-38.
Crossref
Crossref
R. Z. Cer, U. Mudunuri, R. Stephens & F. J. Lebeda. (2009) IC50-to-Ki: a web-based tool for converting IC50 to Ki values for inhibitors of enzyme activity and ligand binding. Nucleic Acids Research 37:Web Server, pages W441-W445.
Crossref
Crossref
Peter Cornelius, Eunsun Lee, Wen Lin, Ruduan Wang, Wendy Werner, Janice A. Brown, Frank Stuhmeier, James G. Boyd & Kim McClure. (2009) Design, Synthesis, and Pharmacology of Fluorescently Labeled Analogs of Serotonin: Application to Screening of the 5-HT2C Receptor. SLAS Discovery 14:4, pages 360-370.
Crossref
Crossref
Susan M. Young, Cristian M. Bologa, Dan Fara, Bj K. Bryant, Juan Jacob Strouse, Jeffrey B. Arterburn, Richard D. Ye, Tudor I. Oprea, Eric R. Prossnitz, Larry A. Sklar & Bruce S. Edwards. (2009) Duplex high-throughput flow cytometry screen identifies two novel formylpeptide receptor family probes. Cytometry Part A 75A:3, pages 253-263.
Crossref
Crossref
A. Quamrul Hassan, Yongting Wang, Lars Plate & JoAnne Stubbe. (2008) Methodology To Probe Subunit Interactions in Ribonucleotide Reductases. Biochemistry 47:49, pages 13046-13055.
Crossref
Crossref
Ralph Mazitschek, Vishal Patel, Dyann F. Wirth & Jon Clardy. (2008) Development of a fluorescence polarization based assay for histone deacetylase ligand discovery. Bioorganic & Medicinal Chemistry Letters 18:9, pages 2809-2812.
Crossref
Crossref
Katrine L. Whiteson & Phoebe A. Rice. (2008) Binding and Catalytic Contributions to Site Recognition by Flp Recombinase. Journal of Biological Chemistry 283:17, pages 11414-11423.
Crossref
Crossref
Ulf Mathias & Manfred Jung. (2007) Determination of drug–serum protein interactions via fluorescence polarization measurements. Analytical and Bioanalytical Chemistry 388:5-6, pages 1147-1156.
Crossref
Crossref
Ernesto Abel-Santos & Tetyana Dodatko. (2007) Differential nucleoside recognition during Bacillus cereus 569 (ATCC 10876) spore germination. New Journal of Chemistry 31:5, pages 748.
Crossref
Crossref
Ting-Chao Chou. (2006) Theoretical Basis, Experimental Design, and Computerized Simulation of Synergism and Antagonism in Drug Combination Studies. Pharmacological Reviews 58:3, pages 621-681.
Crossref
Crossref
Bruce S. Edwards, Cristian Bologa, Susan M. Young, Konstantin V. Balakin, Eric R. Prossnitz, Nikolay P. Savchuck, Larry A. Sklar & Tudor I. Oprea. (2005) Integration of Virtual Screening with High-Throughput Flow Cytometry to Identify Novel Small Molecule Formylpeptide Receptor Antagonists. Molecular Pharmacology 68:5, pages 1301-1310.
Crossref
Crossref
Susan M. Young, Cristian Bologa, Eric R. Prossnitz, Tudor I. Oprea, Larry A. Sklar & Bruce S. Edwards. (2005) High-Throughput Screening with HyperCyt® Flow Cytometry to Detect Small Molecule Formylpeptide Receptor Ligands. SLAS Discovery 10:4, pages 374-382.
Crossref
Crossref
Boris I. Feldkoren & Stefan Andersson. (2005) Anabolic-androgenic steroid interaction with rat androgen receptor in vivo and in vitro: A comparative study. The Journal of Steroid Biochemistry and Molecular Biology 94:5, pages 481-487.
Crossref
Crossref
Juan Zhen, Soumen Maiti, Nianhang Chen, Aloke K. Dutta & Maarten E.A. Reith. (2004) Interaction between a hydroxypiperidine analogue of 4-(2-benzhydryloxy-ethyl)-1-(4-fluorobenzyl)piperidine and Aspartate 68 in the human dopamine transporter. European Journal of Pharmacology 506:1, pages 17-26.
Crossref
Crossref
Zaneta Nikolovska-Coleska, Renxiao Wang, Xueliang Fang, Hongguang Pan, York Tomita, Peng Li, Peter P. Roller, Krzysztof Krajewski, Naoyuki G. Saito, Jeanne A. Stuckey & Shaomeng Wang. (2004) Development and optimization of a binding assay for the XIAP BIR3 domain using fluorescence polarization. Analytical Biochemistry 332:2, pages 261-273.
Crossref
Crossref
Patrick D. Braun & Thomas J. Wandless. (2004) Quantitative Analyses of Bifunctional Molecules. Biochemistry 43:18, pages 5406-5413.
Crossref
Crossref
Gil Belofsky, April N. French, David R. Wallace & Summer L. Dodson. (2003)
New Geranyl Stilbenes from
Dalea
p
urpurea
with in Vitro Opioid Receptor Affinity
. Journal of Natural Products 67:1, pages 26-30.
Crossref
Crossref
Xinyi Huang. (2003) Equilibrium competition binding assay: inhibition mechanism from a single dose response. Journal of Theoretical Biology 225:3, pages 369-376.
Crossref
Crossref
Stacey E. Rutledge, Heather M. Volkman & Alanna Schepartz. (2003) Molecular Recognition of Protein Surfaces: High Affinity Ligands for the CBP KIX Domain. Journal of the American Chemical Society 125:47, pages 14336-14347.
Crossref
Crossref
Kenneth A. Krohn & Jeanne M. Link. (2003) Interpreting enzyme and receptor kinetics: keeping it simple, but not too simple. Nuclear Medicine and Biology 30:8, pages 819-826.
Crossref
Crossref
Dustin Deming, Qing Cheng & Vasanthi Jayaraman. (2003) Is the Isolated Ligand Binding Domain a Good Model of the Domain in the Native Receptor?. Journal of Biological Chemistry 278:20, pages 17589-17592.
Crossref
Crossref
Xinyi Huang. (2003) Fluorescence Polarization Competition Assay: The Range of Resolvable Inhibitor Potency Is Limited by the Affinity of the Fluorescent Ligand. SLAS Discovery 8:1, pages 34-38.
Crossref
Crossref
S. Bollini, J.J. Herbst, G.T. Gaughan, T.A. Verdoorn, J. Ditta, G.M. Dubowchik & A. Vinitsky. (2002) High-Throughput Fluorescence Polarization Method for Identification of FKBP12 Ligands. SLAS Discovery 7:6, pages 526-530.
Crossref
Crossref
Esther Arranz-Plaza, Alex S. Tracy, Aloysius Siriwardena, J. Michael Pierce & Geert-Jan Boons. (2002)
High-Avidity, Low-Affinity Multivalent Interactions and the Block to Polyspermy in
Xenopus
l
aevis
. Journal of the American Chemical Society 124:44, pages 13035-13046.
Crossref
Crossref
Penny A. Wright, Helen F. Boyd, Richard C. Bethell, Michael Busch, Phillip Gribbon, Joachim Kraemer, Eloisa Lopez-Calle, Thomas H. Mander, Dirk Winkler & Neil Benson. (2002) Development of a 1-μl Scale Assay for Mitogen-Activated Kinase Kinase 7 Using 2-D Fluorescence Intensity Distribution Analysis Anisotropy. SLAS Discovery 7:5, pages 419-428.
Crossref
Crossref
Daniel Assefa, Adam J Pawson, Craig A McArdle, Robert P Millar, Colleen A Flanagan, R Roeske & James S Davidson. (1999) A new photoreactive antagonist cross-links to the N-terminal domain of the gonadotropin-releasing hormone receptor. Molecular and Cellular Endocrinology 156:1-2, pages 179-188.
Crossref
Crossref
Krishnendu Ghosh, Dianne Kowal, Lee A. Dawson & Rene Tasse. (1999) Design and models for estimating antagonist potency (pA2, Kd and IC50) following the detection of antagonism observed in the presence of intrinsic activity. Neuropharmacology 38:3, pages 361-373.
Crossref
Crossref
Everardus J.J van Zoelen, Roel H Kramer, Herman T.B van Moerkerk & Jacques H Veerkamp. (1998) The use of nonhomologous Scatchard analysis in the evaluation of ligand–protein interactions. Trends in Pharmacological Sciences 19:12, pages 487-490.
Crossref
Crossref
R BolgerT E WieseK ErvinS NestichW Checovich. (1998) Rapid screening of environmental chemicals for estrogen receptor binding capacity.. Environmental Health Perspectives 106:9, pages 551-557.
Crossref
Crossref
Philip Seeman & Shitij Kapur. (1997) Clozapine occupies high levels of dopamine D2 receptors. Life Sciences 60:12, pages PL207-PL216.
Crossref
Crossref
Mei-Ping Kung, D.Andrew Stevenson, Zhi-Ping Zhuang, Janet M. Vessotskie, Sumalee Chumpradit, Xiao-Ming Sun & Hank F. Kung. (1996) Characterization of a novel iodinated ligand, IPMPP, for human dopamine D4 receptors expressed in CHO cells. Life Sciences 60:2, pages 91-100.
Crossref
Crossref
Philip Seeman & Hubert H.M. Van Tol. (1995) Deriving the therapeutic concentrations for clozapine and haloperidol: The apparent dissociation constant of a neuroleptic at the dopamine D2 or D4 receptor varies with the affinity of the competing radioligand. European Journal of Pharmacology: Molecular Pharmacology 291:2, pages 59-66.
Crossref
Crossref
R.P. Millar, J. Davidson, I. Wakefield & C. Flanagan. 1995. Receptor Molecular Biology. Receptor Molecular Biology
145
162
.
Rosemarie M. Booze & David R. Wallace. (2004)
Dopamine D
2
and D
3
receptors in the rat striatum and nucleus accumbens: Use of 7‐OH‐DPAT and [
125
I]‐Iodosulpride
. Synapse 19:1, pages 1-13.
Crossref
Crossref
J. Svaren, B.D. Wineinger & R. Chalkley. (1994) Extent of in vivo binding by an upstream activation factor and the role of multiple binding sites in synergistic transcriptional activation.. Journal of Biological Chemistry 269:32, pages 20771-20779.
Crossref
Crossref
S. Lazareno & N.J.M. Birdsall. (2012) Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng‐Prusoíf equations. British Journal of Pharmacology 109:4, pages 1110-1119.
Crossref
Crossref
Gábor Maksay. (1993) Partial and full agonists/inverse agonists affect [35S]TBPS binding at different occupancies of central benzodiazepine receptors. European Journal of Pharmacology: Molecular Pharmacology 246:3, pages 255-260.
Crossref
Crossref
Barbara A. Cox, Robert A. Henningsen, Athena Spanoyannis, Rachael L. Neve & Kim A. Neve. (2006) Contributions of Conserved Serine Residues to the Interactions of Ligands with Dopamine D2 Receptors. Journal of Neurochemistry 59:2, pages 627-635.
Crossref
Crossref
Jeffrey P. Bond, Shlomo Sasson & Angelo C. Notides. (1992) The binding of estrogen and estrogen antagonists to the estrogen receptor. Archives of Biochemistry and Biophysics 296:2, pages 583-591.
Crossref
Crossref
Mario Tiberi. 1992. Computers and Computations in the Neurosciences - Methods in Neurosciences. Computers and Computations in the Neurosciences - Methods in Neurosciences
196
216
.
Peter J. Munson & G. Enrico Rovati. 1992. Computers and Computations in the Neurosciences - Methods in Neurosciences. Computers and Computations in the Neurosciences - Methods in Neurosciences
175
195
.
Thérèse M. Keravis, Herrade Nehlig, Marie-Françoise Delacroix, Domenico Regoli, C. Robin Hiley & Jean-Claude Stoclet. (1991) High-affinity bradykinin B2 binding sites sensitive to guanine nucleotides in bovine aortic endothelial cells. European Journal of Pharmacology: Molecular Pharmacology 207:2, pages 149-155.
Crossref
Crossref
Richard Poulin, Denis Baker, Donald Poirier & Fernand Labrie. (1991) Multiple actions of synthetic ‘progestins’ on the growth of ZR-75-1 human breast cancer cells: Anin vitro model for the simultaneous assay of androgen, progestin, estrogen, and glucocorticoid agonistic and antagonistic activities of steroids. Breast Cancer Research and Treatment 17:3, pages 197-210.
Crossref
Crossref
David E. Schafer. 1992. New Trends in Pharmacokinetics. New Trends in Pharmacokinetics
103
123
.
R H Havunjian, B R De Costa, K C Rice & P Skolnick. (1990) Characterization of benzodiazepine receptors with a fluorescence-quenching ligand.. Journal of Biological Chemistry 265:36, pages 22181-22186.
Crossref
Crossref
C. Robin Hiley, C. Richard Jones, John T. Pelton & Robert C. Miller. (1990) Binding of [125I]-endothelin-1 to rat cerebellar homogenates and its interactions with some analogues. British Journal of Pharmacology 101:2, pages 319-324.
Crossref
Crossref
Jacques Simard, Claude Labrie, Yves Mérand, Jean-Marc Dufour, Charles Lévesque & Fernand Labrie. (1990) Pure Antagonistic Effect of a New Steroidal Antiestrogen in Rat Anterior Pituitary Cells in Culture and in Mouse Uterus. Annals of the New York Academy of Sciences 595:1 Steroid Forma, pages 425-427.
Crossref
Crossref
Fernand Labrie, Richard Poulin, Jacques Simard, Hui Fen Zhao, Claude Labrie, Sophie Dauvois, Martine Dumont, Anne-Catherine Hatton, Donald Poirier & Yves Mérand. (1990) Interactions between Estrogens, Androgens, Progestins, and Glucocorticoids in ZR-75-1 Human Breast Cancer Cells. Annals of the New York Academy of Sciences 595:1 Steroid Forma, pages 130-148.
Crossref
Crossref
Richard Poulin, Yves Merand, Donald Poirier, Charles Levesque, Jean-Marc Dufour & Fernand Labrie. (1989) Antiestrogenic properties of keoxifene,trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells. Breast Cancer Research and Treatment 14:1, pages 65-76.
Crossref
Crossref
Raymond M. Dawson & Michael Poretski. (1989) Inhibition constants and GABA-shifts at 2°C and 37°C for a spectrum of ligands acting on the benzodiazepine receptors of guinea pig hippocampus. General Pharmacology: The Vascular System 20:6, pages 843-848.
Crossref
Crossref
G.Enrico Rovati, David Rodbard & Peter J. Munson. (1988) DESIGN: Computerized optimization of experimental design for estimating Kd and Bmax in ligand binding experiments. Analytical Biochemistry 174:2, pages 636-649.
Crossref
Crossref