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Roberta Ettari, Santo Previti, Santina Maiorana, Alessandro Allegra, Tanja Schirmeister, Silvana Grasso & Maria Zappalà. (2019) Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense
. Natural Product Research 33:24, pages 3577-3581.
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Erick Tavares Marcelino Alves, Filipe Gomes Pernichelle, Lucas Adriano Nascimento, Glaucio Monteiro Ferreira & Elizabeth Igne Ferreira. (2023) Covalent Inhibitors for Neglected Diseases: An Exploration of Novel Therapeutic Options. Pharmaceuticals 16:7, pages 1028.
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Ammar Usman Danazumi, Ibtida Tabassum Ishmam, Salisu Idris, Matylda Anna Izert, Emmanuel Oluwadare Balogun & Maria Wiktoria Górna. (2023) Targeted protein degradation might present a novel therapeutic approach in the fight against African trypanosomiasis. European Journal of Pharmaceutical Sciences 186, pages 106451.
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Carla Di Chio, Santo Previti, Noemi Totaro, Fabiola De Luca, Alessandro Allegra, Tanja Schirmeister, Maria Zappalà & Roberta Ettari. (2023) Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense. International Journal of Molecular Sciences 24:10, pages 8477.
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Santo Previti, Roberta Ettari, Carla Di Chio, Jenny Legac, Marta Bogacz, Collin Zimmer, Tanja Schirmeister, Philip J. Rosenthal & Maria Zappalà. (2023) Influence of amino acid size at the P3 position of N-Cbz-tripeptide Michael acceptors targeting falcipain-2 and rhodesain for the treatment of malaria and human african trypanosomiasis. Bioorganic Chemistry, pages 106587.
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Santo Previti, Roberta Ettari, Elsa Calcaterra, Salvatore Di Maro, Stefan J. Hammerschmidt, Christin Müller, John Ziebuhr, Tanja Schirmeister, Sandro Cosconati & Maria Zappalà. (2023) Structure-based lead optimization of peptide-based vinyl methyl ketones as SARS-CoV-2 main protease inhibitors. European Journal of Medicinal Chemistry 247, pages 115021.
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Carla Di Chio, Santo Previti, Fabiola De Luca, Marta Bogacz, Collin Zimmer, Annika Wagner, Tanja Schirmeister, Maria Zappalà & Roberta Ettari. (2022) Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense. International Journal of Molecular Sciences 23:22, pages 14470.
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Santo Previti, Roberta Ettari, Elsa Calcaterra, Carla Di Chio, Rahul Ravichandran, Collin Zimmer, Stefan Hammerschmidt, Annika Wagner, Marta Bogacz, Sandro Cosconati, Tanja Schirmeister & Maria Zappalà. (2022) Development of Urea-Bond-Containing Michael Acceptors as Antitrypanosomal Agents Targeting Rhodesain. ACS Medicinal Chemistry Letters 13:7, pages 1083-1090.
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Susy Érika de Lima Barros, Henrique Barros de Lima, Leandra Karoline Alves Gonçalves, Lenir Cabral Correia, Maiara de Fátima de Brito Brito, Mariana Pegrucci Barcelos, Guilherme Martins Silva, Carlos Henrique Tomich de Paula da Silva, Rafael Garrett da Costa, Rodrigo Alves Soares Cruz, José Carlos Tavares Carvalho & Lorane Izabel da Silva Hage-Melim. (2022) Chromatographic profile, in silico and in vivo study of the pharmacokinetic and toxicological properties of major constituent present in kefir, the kefiran. Toxicology Research 11:3, pages 520-528.
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Santo Previti, Roberta Ettari, Carla Di Chio, Rahul Ravichandran, Marta Bogacz, Ute A. Hellmich, Tanja Schirmeister, Sandro Cosconati & Maria Zappalà. (2022) Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis. Molecules 27:12, pages 3765.
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Carla Di Chio, Santo Previti, Giorgio Amendola, Rahul Ravichandran, Annika Wagner, Sandro Cosconati, Ute A. Hellmich, Tanja Schirmeister, Maria Zappalà & Roberta Ettari. (2022) Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense. European Journal of Medicinal Chemistry 236, pages 114328.
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Aureliano Zana & Andrea Galbiati. (2021) Synthesis and Reactivity of 3‐Halo‐4,5‐dihydroisoxazoles: An Overview. ChemistrySelect 6:32, pages 8249-8261.
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Kemel Arafet, Florenci V. González & Vicent Moliner. (2021) Elucidating the Dual Mode of Action of Dipeptidyl Enoates in the Inhibition of Rhodesain Cysteine Proteases. Chemistry – A European Journal 27:39, pages 10142-10150.
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Roberta Ettari, Santo Previti, Carla Di Chio & Maria Zappalà. (2021) Falcipain-2 and Falcipain-3 Inhibitors as Promising Antimalarial Agents. Current Medicinal Chemistry 28:15, pages 3010-3031.
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Donald J. AbrahamConor R. Caffrey, Dietmar Steverding, Rafaela S. Ferreira, Renata B. Oliveira, Anthony J. O'Donoghue, Ludovica Monti, Carlo Ballatore, Kelly A. Bachovchin, Lori Ferrins, Michael P. Pollastri, Kimberley M. Zorn, Daniel H. Foil, Alex M. Clark, Melina Mottin, Carolina H. Andrade, Jair L. Siqueira‐Neto & Sean Ekins. 2003. Burger's Medicinal Chemistry and Drug Discovery. Burger's Medicinal Chemistry and Drug Discovery
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Santina Maiorana, Roberta Ettari, Santo Previti, Giorgio Amendola, Annika Wagner, Sandro Cosconati, Ute A. Hellmich, Tanja Schirmeister & Maria Zappalà. (2020) Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment. ChemMedChem 15:16, pages 1552-1561.
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Carla Di Chio, Santo Previti, Giorgio Amendola, Sandro Cosconati, Tanja Schirmeister, Maria Zappalà & Roberta Ettari. (2020)
Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from
Trypanosoma brucei rhodesiense
. ChemMedChem 15:11, pages 995-1001.
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Roberta Ettari, Santo Previti, Carla Di Chio, Santina Maiorana, Alessandro Allegra, Tanja Schirmeister & Maria Zappalà. (2020)
Drug Synergism: Studies of Combination of RK-52 and Curcumin against Rhodesain of
Trypanosoma brucei rhodesiense
. ACS Medicinal Chemistry Letters 11:5, pages 806-810.
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Roberta Ettari, Santo Previti, Santina Maiorana, Giorgio Amendola, Annika Wagner, Sandro Cosconati, Tanja Schirmeister, Ute A. Hellmich & Maria Zappalà. (2019) Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis. Journal of Medicinal Chemistry 62:23, pages 10617-10629.
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Débora A. Rocha, Elany B. Silva, Isadora S. Fortes, Marcela S. Lopes, Rafaela S. Ferreira & Saulo F. Andrade. (2018) Synthesis and structure-activity relationship studies of cruzain and rhodesain inhibitors. European Journal of Medicinal Chemistry 157, pages 1426-1459.
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Santiago Royo, Tanja Schirmeister, Marcel Kaiser, Sascha Jung, Santiago Rodríguez, José Manuel Bautista & Florenci V. González. (2018) Antiprotozoal and cysteine proteases inhibitory activity of dipeptidyl enoates. Bioorganic & Medicinal Chemistry 26:16, pages 4624-4634.
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Leonardo G. Ferreira & Adriano D. Andricopulo. (2017) Targeting cysteine proteases in trypanosomatid disease drug discovery. Pharmacology & Therapeutics 180, pages 49-61.
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Santo Previti, Roberta Ettari, Sandro Cosconati, Giorgio Amendola, Khawla Chouchene, Annika Wagner, Ute A. Hellmich, Kathrin Ulrich, R. Luise Krauth-Siegel, Peter R. Wich, Ira Schmid, Tanja Schirmeister, Jiri Gut, Philip J. Rosenthal, Silvana Grasso & Maria Zappalà. (2017) Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs). Journal of Medicinal Chemistry 60:16, pages 6911-6923.
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Milad Espahbodinia, Roberta Ettari, Wei Wen, Andrew Wu, Yu-Chuan Shen, Li Niu, Silvana Grasso & Maria Zappalà. (2017) Development of novel N -3-bromoisoxazolin-5-yl substituted 2,3-benzodiazepines as noncompetitive AMPAR antagonists. Bioorganic & Medicinal Chemistry 25:14, pages 3631-3637.
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Maude Giroud, Jakov Ivkovic, Mara Martignoni, Marianne Fleuti, Nils Trapp, Wolfgang Haap, Andreas Kuglstatter, Jörg Benz, Bernd Kuhn, Tanja Schirmeister & François Diederich. (2017) Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide⋅⋅⋅Heteroarene π-Stacking Interactions and Chalcogen Bonding in the S3 Pocket. ChemMedChem 12:3, pages 257-270.
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