569
Views
9
CrossRef citations to date
0
Altmetric
Original Article

Antimicrobial and in vitro cytotoxicity of novel sulphanilamide condensed 1,2,3,4-tetrahydropyrimidinesFootnote

, , , &

References

  • Y.LeylaO.YusufK.Zafer AsimT.YagmurK.HulyaSynthesis and antimicrobial activity of some new hydrazone-bridged thiazole-pyrrole derivativesJ. Enzym. Inhib. Med. Chem.2820132013830835
  • N.G.SandipL.M.VijayM.K.KisanS.S.MurlidharV.M.DhananjaySynthesis and biological evaluation of novel 2,4,6-triazine derivatives as antimicrobial agentsBioorg. Med. Chem. Lett.22201250755077
  • P.BiginelliAldehyde-urea derivatives of aceto and oxaloacetic acidsGazs. Chim. Ital.231983360413
  • K.S.AtwalG.C.RovnyakJ.SchwartzS.MorelandA.HedbergJ.Z.GougoutasM.F.MalleyD.M.FloydDihydropyrimidine calcium channel blockers: 2-heterosubstituted 4-aryl-1,4-dihydro-6-methyl-5-pyrimidinecarboxylic acid esters as potent mimics of dihydropyridinesJ. Med. Chem.33199015101515
  • C.O.Kappe4-Aryldihydropyrimidines via the Biginelli condensation: aza-analogs of nifedipine-type calcium channel modulatorsMolecules3199819
  • D.J.TriggleR.A.JanisCalcium channel ligandsAnn. Rev. Pharmacol. Toxicol.271987347369
  • B.DesaiD.SurejaY.NaliaparaA.ShahA.K.SaxenaSynthesis and QSAR studies of 4-substituted phenyl-2,6-dimethyl-3,5-bis-n-(substituted phenyl) carbamoyl-1,4-dihydropyridines as potential antitubercular agentsBioorg. Med. Chem. Lett.9200119931998
  • S.KamaljitS.KawaljitW.BaojieF.ScottC.KellyFacile transformation of Biginelli pyrimidin-2(1H)-ones to pyrimidines. In vitro evaluation as inhibitors of Mycobacterium tuberculosis and modulators of cytostatic activityBioorg. Med. Chem. Lett.46201122902294
  • D.B.AtulB.V.KartikB.P.KetanS.N.KiranSynthesis of 1,2,3,4-tetrahydro pyrimidine derivatives as an antimicrobial agentJ. Chem. Pharm. Res.4201229722978
  • H.B.Md MosharefR.Md MizanurH.Md KamrulR.AbdurH.Md IsmailN.Md AbuSynthesis and antimicrobial evaluation of some new thienopyrimidine derivativesActa Pharm.562006441450
  • S.S.NitinkumarS.L.RaviA.M.K.ImtiyazSynthesis and antimicrobial activity of some novel thienopyrimidine and triazolothienopyrimidinesJ. Chem. Sci.1212009301307
  • S.PratibhaR.NileshV.K.GurramSynthesis and QSAR studies of pyrimido[4,5-d]pyrimidine-2,5-dione derivatives as potential antimicrobial agentsBioorg. Med. Chem. Lett.14200441854190
  • A.E.WaelM.A.OmarA.Z.RihanaA.M.AsemA.H.Abdul RehmanSynthesis and antimicrobial activity of new Substituted thienopyrimidines, their tetrazolyl and sugar derivativesActa Pol. Pharm.692012439447
  • J.GillespieA.C.IanE.D.ClaireAntagonists of the human adenosine A2A receptor. Part 3: design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3 d]pyrimidines and 6-arylpurinesBioorg. Med. Chem. Lett.18200829242929
  • O.AurelioM.RamonL.BeatrizO.RobertoNovel 2-(4-methylsulfonylphenyl) pyrimidine derivatives as highly potent and specific COX-2 inhibitorsBioorg. Med. Chem.16200821832199
  • P.EmersonJ.SebastiaoM.S.RajendraSynthesis and anti-inflammatory activity of 4-amino-2-aryl-5-cyano-6-{3- and 4-(N-phthalimidophenyl)} pyrimidine'sEur. J. Med. Chem.412006276282
  • G.AleemZ.YingR.SudhirA.I.MichaelC.D.BryanDesign, synthesis and evaluation of 2-amino-4-m-bromoanilino-6-arylmethyl-7 H-pyrrolo [2,3d]pyrimidine's as tyrosine kinase inhibitors and antiangiogenic AgentsBioorg. Med. Chem.18201052615273
  • P.HumairaH.FaisalS.AttarA.AmirSynthesis, characterization and biological evaluation of novel 6-ferrocenyl-4-aryl-2-substituted pyrimidine derivativesEur. J. Med. Chem.45201034973503
  • X.FuchunZ.HongbingZ.LizhiL.LiguangH.YouhongSynthesis and biological evaluation of novel 2,4,5-substituted pyrimidine derivatives for anticancer activityBioorg. Med. Chem. Lett.192009275278
  • J.T.SarithaG.AchaiahSynthesis of new pyrrolo[2,3-d]pyrimidine derivatives and evaluation of their activities against human colon cancer cell linesEur. J. Med. Chem.45201014531458
  • A.HulyaK.IremB.BarkinK.IsilS.GizemO.SinemK.TanilSynthesis and antimycobacterial activity of some phthalimide derivativesBioorg. Med. Chem.20201241494154
  • R.VasudevaY.RajendraG.GirijasankarG.PradeepsagarSynthesis, characterization and in vitro biological evaluation of some novel diarylsulfonylureas as potential cytotoxic and antimicrobial agentsBioorg. Med. Chem. Lett.22201210311035
  • B.ZhuB.A.MarinelliR.GoldschmidtSynthesis and antibacterial activity of 7-(1,2,3,4-tetrahydropyrrolo [1,2-a]-pyrazin-7-yl) quinolonesBioorg. Med. Chem. Lett.19200949334936
  • B.R.PrashanthaM.PankajE.KarthikeyanB.AnkurB.SujaP.VijayanSynthesis of novel Hantzsch dihydropyridines and Biginelli dihydropyrimidines of biological interest: a 3D-QSAR study on their cytotoxicityMed. Chem. Res.192010344363
  • L.S.RameshS.B.ManishSynthesis, screening and QSAR studies of 3-benzoyl-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidine analogues as antibacterial agentsBull. Chem. Soc. Ethiop.222008391402
  • C.O.KappeA reexamination of the mechanism of the Biginelli Dihydropyrimidine synthesis, support for an N-acyliminium ion intermediateJ. Org. Chem.62199772017204