Mesalazine solubility in the binary mixtures of ethanol and water at various temperatures

References

• Actis GC, Pellicano R, Rizzetto M, et al. Individually administered or co-prescribed thiopurines and mesalamines for inflammatory bowel disease. World J Gastroenterol. 2009;15:1420–1426.
   PubMed Web of Science ®Google Scholar
• Gonçalves E, Almeida LM, Dinis TC. Antioxidant activity of 5-aminosalicylic acid against peroxidation of phosphatidylcholine liposomes in the presence of α-tocopherol: a synergistic interaction? Free Radic Res. 1998;29:53–66.
   PubMed Web of Science ®Google Scholar
• Sandborn W, Feagan B, Lichtenstein G. Medical management of mild to moderate Crohn’s disease: evidence‐based treatment algorithms for induction and maintenance of remission. Aliment Pharmacol Ther. 2007;26:987–1003.
   PubMed Web of Science ®Google Scholar
• Palumbo G, Carlucci G, Mazzeo P, et al. Simultaneous determination of 5-aminosalicylic acid, acetyl-5-aminosalicylic acid and 2, 5-dihydroxybenzoic acid in endoscopie intestinal biopsy samples in humans by high-performance liquid chromatography with electrochemical detection. J Pharm Biomed Anal. 1995;14:175–180.
   PubMed Web of Science ®Google Scholar
• Patel A, Vaghasiya A, Gajera R, et al. Solubility of 5-amino salicylic acid in different solvents at various temperatures. J Chem Eng Data. 2010;55:1453–1455.
   Web of Science ®Google Scholar
• Stieger N, Liebenberg W, Andreeta M. Recrystallization of active pharmaceutical ingredients. In: Andreeta MRB, editor. Crystallization: science and technology. Ri‐jeka, Croatia: InTechOpen; 2012, Chap. 7, 183-185.
   Google Scholar
• Giulietti M, Bernardo A. Crystallization by antisolvent addition and cooling. In: Andreeta MRB, editor. Crystallization-science and technology. Ri-jeka, Croatia: IntechOpen; 2012, Chap. 14, 379-380.
   Google Scholar
• Di L, Fish PV, Mano T. Bridging solubility between drug discovery and development. Drug Discov Today. 2012;17:486–495.
   PubMed Web of Science ®Google Scholar
• Strickley RG. Solubilizing excipients in oral and injectable formulations. Pharm Res. 2004;21:201–230.
   PubMed Web of Science ®Google Scholar
• Alsenz J, Kansy M. High throughput solubility measurement in drug discovery and development. Adv Drug Deliv Rev. 2007;59:546–567.
   PubMed Web of Science ®Google Scholar
• Jouyban A. Handbook of solubility data for pharmaceuticals. Boca Raton: CRC Press; 2010.
   Google Scholar
• Lau E, Giddings S, Mohammed S, et al. Encapsulation of hydrocortisone and mesalazine in zein microparticles. Pharmaceutics. 2013;5:277–293.
   PubMedGoogle Scholar
• Jouyban A, Fakhree MAA. In: Acree Jr WE, editor. Experimental and computational methods pertaining to drug solubility, 192-193. Toxicity and drug testing. New York: Intech Co; 2012. Chap. 9.
   Google Scholar
• Vahdati S, Shayanfar A, Hanaee J, et al. Solubility of carvedilol in ethanol+ propylene glycol mixtures at various temperatures. Ind Eng Chem Res. 2013;52:16630–16636.
   Web of Science ®Google Scholar
• Perlovich GL, Kurkov SV, Bauer-Brandl A. Thermodynamics of solutions: II. Flurbiprofen and diflunisal as models for studying solvation of drug substances. Eur J Pharm Sci. 2003;19:423–432.
   PubMed Web of Science ®Google Scholar
• Zhou C, Shi X, Wang H, et al. Measurement and correlation of solubilities of trans-ferulic acid in solvents. J Chem Ind Eng. 2007;58:2705.
   Google Scholar
• Ochsner AB, Jr Belloto RJ, Sokoloski TD. Prediction of xanthine solubilities using statistical techniques. J Pharm Sci. 1985;74:132–135.
   PubMed Web of Science ®Google Scholar
• Yalkowsky SH, Roseman TJ. Solubilization of drugs by cosolvents. In: Yalkowsky SH, editor. Techniques of solubilization of drugs. New York: Marcel Dekker Inc; 1981. p. 91–134.
   Google Scholar
• Millard JW, Alvarez-Nunez F, Yalkowsky SH. Solubilization by cosolvents: establishing useful constants for the log–linear model. Int J Pharm. 2002;245:153–166.
   PubMed Web of Science ®Google Scholar
• Valvani S, Yalkowsky SH, Roseman T. Solubility and partitioning IV: aqueous solubility and octanol-water partition coefficients of liquid nonelectrolytes. J Pharm Sci. 1981;70:502–507.
   PubMed Web of Science ®Google Scholar
• Jouyban A, Acree WE. Mathematical derivation of the Jouyban-Acree model to represent solute solubility data in mixed solvents at various temperatures. J Mol Liq. 2018;256:541–547.
   Web of Science ®Google Scholar
• Jouyban A, Khoubnasabjafari M, Chan H-K, et al. Mathematical representation of solubility of amino acids in binary aqueous-organic solvent mixtures at various temperatures using the Jouyban-Acree model. Pharmazie. 2006;61:789–792.
   PubMed Web of Science ®Google Scholar
• Jouyban A, Fakhree MAA, Acree WE. Comment on measurement and correlation of solubilities of (z)-2-(2-aminothiazol-4-yl)-2-methoxyiminoacetic acid in different pure solvents and binary mixtures of water+(ethanol, methanol, or glycol). J Chem Eng Data. 2012;57:1344–1346.
   Web of Science ®Google Scholar
• Jouyban-Gharamaleki A. The modified Wilson model and predicting drug solubility in water-cosolvent mixtures. Chem Pharm Bull. 1998;46:1058–1061.
   Web of Science ®Google Scholar
• Gantiva M, Martínez F. Thermodynamic analysis of the solubility of ketoprofen in some propylene glycol+ water cosolvent mixtures. Fluid Phase Equilib. 2010;293:242–250.
   Web of Science ®Google Scholar
• Marcus Y. Solvent mixtures: properties and selective solvation. New York: Marcel Dekker, Inc.; 2002.
   Google Scholar
• Marcus Y. On the preferential solvation of drugs and PAHs in binary solvent mixtures. J Mol Liq. 2008;140:61–67.
   Web of Science ®Google Scholar
• Marcus Y. Preferential solvation of ibuprofen and naproxen in aqueous 1,2–propanediol. Acta Chim Sloven. 2009;56:40–44.
   Web of Science ®Google Scholar
• Jiménez DM, Cárdenas ZJ, Delgado DR, et al. Preferential solvation of methocarbamol in aqueous binary cosolvent mixtures at 298.15 K. Phys Chem Liq. 2014;52:726–737.
   Web of Science ®Google Scholar
• Mesalazine C. http://www.chemspider.com/Chemical-Structure.3933.html
   Google Scholar
• Ben-Naim A. Theory of preferential solvation of nonelectrolytes. Cell Biophys. 1988;12:255–269.
   PubMedGoogle Scholar
• Ben-Naim A. Preferential solvation in two- and in three-component systems. Pure Appl Chem. 1990;62:25–34.
   Web of Science ®Google Scholar
• Marcus Y. The properties of solvents. Chichester: John Wiley & Sons; 1998.
   Google Scholar
• Taft RW, Kamlet MJ. The solvatochromic comparison method II. The alpha-scale of solvent hydrogen-bond donor (HBD) acidities. J Am Chem Soc. 1976;98:2886–2894.
   Web of Science ®Google Scholar
• Ruckenstein E, Shulgin I. Effect of a third component on the interactions in a binary mixture determined from the fluctuation theory of solutions. Fluid Phase Equilib. 2001;180:281–297.
   Web of Science ®Google Scholar
• Delgado DR, Peña MA, Martínez F. Preferential solvation of acetaminophen in ethanol + water solvent mixtures according to the inverse Kirkwood-Buff integrals method. Rev Colomb Cienc Quím Farm. 2013;42:298–314.
   Google Scholar
• Delgado DR, Martínez F. Preferential solvation of sulfadiazine, sulfamerazine and sulfamethazine in ethanol + water solvent mixtures according to the IKBI method. J Mol Liq. 2014;193:152–159.
   Web of Science ®Google Scholar
• Delgado DR, Peña MA, Martínez F, et al. Further numerical analyses on the solubility of sulfapyridine in ethanol + water mixtures. Pharm Sci (Tabriz). 2016;22:143–152.
   Google Scholar
• Jouyban A, Martínez F. Preferential solvation of nifedipine in some aqueous co-solvent mixtures. Phys Chem Liq. 2016;54:563–573.
   Web of Science ®Google Scholar
• Jouyban A, Acree WE Jr, Martínez F. Solution thermodynamics and preferential solvation of atenolol in {ethanol (1) + water (2)} cosolvent mixtures. J Appl Sol Chem Mod. 2018;7:1–8.
   Google Scholar
• Tinjacá DA, Shayanfar A, Jouyban AF, et al. Preferential solvation of some antiepileptic drugs in {cosolvent (1) + water (2)} mixtures at 298.15 K. Phys Chem Liq. 2018;56:646–659.
   Web of Science ®Google Scholar
• Romdhani A, Martínez F, Almanza OA, et al. Solubility of sulfacetamide in (ethanol + water) mixtures: measurement, correlation, thermodynamics, preferential solvation and volumetric contribution at saturation. J Mol Liq. 2019;290:111219.
   Web of Science ®Google Scholar
• Mirzaeei S, Pirhayati FH, Mohammadi G, et al. Solubility of minoxidil in binary mixture of ethanol + water at various temperatures. Phys Chem Liq. Forthcoming. DOI:10.1080/00319104.2018.1528596.
   Web of Science ®Google Scholar
• Jouyban A. Review of the cosolvency models for predicting solubility of drugs in water-cosolvent mixtures. J Pharm Pharm Sci. 2008;11:32–58.
   PubMed Web of Science ®Google Scholar
• Jouyban A, Soltanpour S, Soltani S, et al. Solubility prediction of drugs in water-cosolvent mixtures using Abraham solvation parameters. J Pharm Pharm Sci. 2007;10:263–277.
   PubMed Web of Science ®Google Scholar
• Jouyban A, Soltanpour S, Soltani S, et al. Prediction of drug solubility in mixed solvents using computed Abraham parameters. J Mol Liq. 2009;146:82–88.
   Web of Science ®Google Scholar
• Jouyban A, Fathi-Azarbayjani A, Khoubnasabjafari M, et al. Mathematical representation of the density of liquid mixtures at various temperatures using Jouyban-Acree model. Ind J Chem. 2005;44A:1553–1560.
   Google Scholar