Asymmetric Synthesis of Aziridinyl Phosphonates Using Darzens-Type Reaction of Chloromethyl Phosphonate to Chiral Sulfinimines

References

• Tanner , D. 1994 . Angew. Chem. Int. Ed. Engl. , 33 : 599
   Web of Science ®Google Scholar
• Zygmunt , J. 1985 . Tetrahedron , 41 : 4979 (b) Hanessian, S.; Bennani, Y. L.; Herve, Y. Synlett 1993, 35. (c) Kim, D. Y.; Rhie, D. Y. Tetrahedron 1997, 53, 13603.
   Web of Science ®Google Scholar
• Hilderbrand , R. L. 1983 . The Role of Phosphonates in Living Systems , Boca Raton, Fl. : CRC Press . (b) Kafarski, P.; Lejczak, B. Phosphorus Sulfur Silicon Relat. Elem. 1991, 63, 193. (c) Boutin, J. A.; Cudennec, C. A.; Hautefaye, P.; Lavielle, G.; Pierre, A.; Schaeffer, C. J. Med. Chem. 1991, 34, 1998. (d) Bartlett, P. A.; Kezer, W. B. J. Am. Chem. Soc. 1984, 106, 4282. (e)Bartlett, P. A.; Giannousis, P. P. J. Med. Chem. 1987, 30, 1603.
   Google Scholar
• Allen , M. C. , Fuhrer , W. , Tuck , B. , Wade , R. and Wood , J. M. 1989 . J. Med. Chem. , 32 : 1652 (b) Logusch, E. W.; Walker, D. M.; McDonald, J. F.; Leo, G. C.; Grang, J. E. J. Org. Chem. 1988, 53 4069. (c) Giannousis, P. P.; Bartlett, P. A. J. Med. Chem. 1987, 30, 1603.
   PubMed Web of Science ®Google Scholar
• Atherton , F. R. , Hassel , C. H. and Lambert , R. W. 1986 . J. Med. Chem. , 29 : 29 (b) Allen, J. G.; Atherton, F. R.; Hassel, C. H.; Holmes, S. W.; Lambert, R. W.; Nisbet, L. J.; Ringrose, P. S. Nature 1978, 272, 56. (c) Allen, J. G.; Atherton, F. R.; Hall, M. J.; Hassel, C. H.; Lambert, R. W.; Nisbet, L. J.; Ringrose, P. S. Antimicrob. Agents Chemother. 1979, 15, 684. (d) Atherton, F. R.; Hall, M. J.; Hassel, C. H.; Lambert, R. W.; Ringrose, P. S. Antimicrob. Agents Chemother. 1979, 15, 677. (e) Atherton, F. R.; Hall, M. J.; Hassel, C. H.; Lambert, R. W.; Lloyd, W. J.; Ringrose, P. S. Antimicrob. Agents Chemother. 1979, 15, 696.
   PubMed Web of Science ®Google Scholar
• Hirschmann , R. , Smith , A. B. III , Taylor , C. M. , Benkovic , P. A. , Taylor , S. D. , Yager , K. M. , Sprengler , P. A. and Venkovic , S. J. 1994 . Science , 265 : 234 (b) Napper, A. D.; Benkovic, S. J; Tramontano, A.; Lerner, R. A. Science 1987, 237, 1041. (c) Smith, A. B. III; Taylor, C. M.; Venkovic, S. J.; Hirschmann, R. Tetrahedron Lett. 1994, 37, 6854.
   PubMed Web of Science ®Google Scholar
• Davis , F. A. and McCoull , W. 1999 . Tetrahedron Lett. , 40 : 249
   Web of Science ®Google Scholar
• Davis , F. A. , Zhou , P. and Chen , B. C. 1998 . Chem. Soc. Rev. , 27 : 13
   Web of Science ®Google Scholar
• Khusainova , N. G. , Bredikhina , Z. A. , Ishmaeva , E. A. , Musina , A. A. and Pudovik , A. N. 1981 . J. Gen. Chem. USSR , 51 : 409
   Google Scholar
• Maury , C. , Gharbaoui , T. , Royer , J. and Hussen , H. P. 1996 . J. Org. Chem. , 61 : 3687 The [α]D of pure 7a was reported to +50.3(c=1, 1N NaOH);
   PubMed Web of Science ®Google Scholar
• Davis , F. A. , Reddy , R. E. , Szewczyk , J. M. , Reddy , V. , Portonovo , P. S. , Zjang , H. , Fabelli , D. , Reddy , R. T. , Zhou , P. and Carrol , P. J. 1997 . J. Org. Chem. , 62 : 2555
   PubMed Web of Science ®Google Scholar