Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 38, 2008 - Issue 8
285
Views
8
CrossRef citations to date
0
Altmetric
Original Articles

N‐Glycosyl‐N′‐[p‐(isoamyloxy)phenyl]‐thiourea Derivatives: Potential Anti‐TB Therapeutic Agents

, &
Pages 1176-1183 | Received 30 Oct 2007, Published online: 17 Apr 2008

References

  • Rouhi , A. M. 1999 . Tuberculosis: A tough adversary . Chem. Eng. News , 77 : 52 – 69 .
  • Dolin , J. P. , Raviglione , M. D. and Kochi , A. 1994 . Global tubeculosis incident and mortality during 1990–2000 . Bull. World Health Org. , 72 : 213 – 220 .
  • Nunn , P. and Kochi , A. 1993 . A deadly duo—TB and AIDS . World Health , 46 : 7 – 8 .
  • 1970 . Discussion on isoxyl . Antibiot. Chemother. , 16 : 187 – 202 . Anonymous
  • Phetsuksiri , B. , Baulard , A. R. , Cooper , A. , Minnikin , D. E. , Douglas , J. D. , Besra , G. S. and Brennan , P. J. 1999 . Antimycobacterial activities of isoxyl and new derivatives through the inhibition of mycolic acid synthesis . Antimicrob. Agents Chemother. , 43 : 1042 – 1051 .
  • Lambelin , G. 1970 . Pharmacology and toxicology of Isoxyl . Antibiot. Chemother. , 16 : 84 – 95 .
  • Camarasa , M. J. , Fernandez‐Resa , P. , Garcia‐Lopez , M. T. , De Las Heras , F. G. , Mendez‐Castrillon , P. P. and San Felix , A. 1984 . A new procedure for the synthesis of glycosyl isothiocynates . Synthesis , : 509 – 510 .
  • Lopez , O. , Maya , I. , Fuentes , J. and Fernandez‐Bolanos , J. G. 2004 . Simple and efficient synthesis of O‐unprotected glycosyl thiourea and isourea derivatives from glycosylamines . Tetrahedron , 60 : 61 – 72 .
  • Babiano Caballero , R. , Fuentes Mota , J. and Galbis Perez , J. A. 1986 . A new method for the preparation of acylated glycosylamines and their transformations into glycosyl isothiocyanates and N,N′‐diglycosyl‐thioureas . Carbohydr. Res. , 154 : 280 – 288 .
  • Takahashi , H. , Nimura , N. and Ogura , H. 1979 . A one‐step synthesis of glycosylaminoisothiaazolo [3,4] pyrimidines and glycosylaminoisothiazoles . Chem. Pharm. Bull. , 27 : 1147 – 1152 .
  • Saitz‐Barria , C. , Torres‐Pinedo , A. and Santoyo‐Gonzales , F. 1999 . Synthesis of bridged thiourea calilx‐sugar . Synlett , 12 : 1891 – 1894 .
  • Gama , Y. , Shibuya , I. and Shimizu , M. 2002 . Novel efficient synthesis of 4‐dimethylamino‐2‐glycosylaminoquinazolines by cyclodesulfurization of glycosylthioureas with dimethylcyanamide . Chem. Pharm. Bull. , 50 : 1517 – 1519 .
  • Prata , C. , Mora , N. , Lacombe , J.‐M. , Maurizis , J.‐C. and Pucci , B. 1999 . Synthesis and surface‐active properties of glycosyl carbamates and thioureas . Carbohydr. Res. , 321 : 4 – 14 .
  • Sivanandan , K. , Sandanaraj , B. S. and Thayumanavan , S. 2004 . Sequences in dendrons and dendrimers . J. Org. Chem. , 69 : 2937 – 2944 .
  • Bellamy , F. D. and Ou , K. 1984 . Selective reduction of aromatic nitro compounds with stannous chloride in non acidic and non aqueous medium . Tetrahedron Lett. , 25 : 839 – 842 .
  • Alaouui , A. E. , Schmidt , F. , Monneret , C. and Florent , J.‐C. 2006 . Protecting groups for glucuronic acid: Application to the synthesis of new paclitaxel derivatives . J. Org. Chem. , 71 : 9628 – 9636 .
  • Gertzke , J. and Wellner , E. Preparation of symmetrically disubstituted thioureas . German (East) patent 19650712 . 1966 .
  • Vourinen , R. and Lampi , K. 4,4‐Bis(isoamyloxy)thiocarbanilide . Finnish patent 36860 19680215 . 1968 .
  • Liav , A. and Brennan , P. J. 2005 . Stereoselective synthesis of farnesylphosphoryl β‐D‐arabinofuranose . Tetrahedron Lett. , 46 : 2937 – 2939 .
  • Collins , L. A. and Franzblau , S. G. 1997 . Microplate alamar blue assay versus BACTAC 460 for high‐throughput screening of compounds against Mycobacterium tuberculosis and Mycobacterium avium . Antimicrob. Agents Chemother. , 41 : 1004 – 1009 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.