Synthesis and in Vitro Antimicrobial Activity of 3-Aryl-4-S-benzyl-6-phenylimino-2-hepta-O-acetyl-β-D-lactosylimino-2,3-dihydro-1,3,5-thiadiazine (Hydrochloride)

REFERENCES

• Rawal , R. K. ; Tripathi , R. ; Katti , S. B. ; Pannecouque , C. ; De Clercq , E. Design and synthesis of 2-(2,6-dibromophenyl)-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents . Eur. J. Med. Chem. 2008 , 43 , 2800 – 2806 .
   PubMed Web of Science ®Google Scholar
• Kaplancikli , Z. A. ; Zitouni , G. T. ; Ozdemir , A. ; Revial , G. New triazole and triazolothiadiazine derivatives as possible antimicrobial agents . Eur. J. Med. Chem. 2008 , 43 , 155 – 159 .
   PubMed Web of Science ®Google Scholar
• Cateni , F. ; Bonivento , P. ; Procida , G. ; Zacchigna , M. ; Favretto , L. G. ; Scialino , G. ; Banfi , E. Chemoenzymatic synthesis and antimicrobial activity evaluation of monogalactosyl diglycerides . Eur. J. Med. Chem. 2008 , 43 , 210 – 221 .
   PubMed Web of Science ®Google Scholar
• Vergne , F. ; Bernardelli , P. ; Lorthiois , E. ; Pham , N. ; Proust , E. ; Oliveira , C. ; Mafroud , A.-K. ; Ducret , P. ; Wrigglesworth , R. ; Berlioz-Seux , F. ; Coleon , F. ; Chevalier , E. ; Moreau , F. ; Idrissi , M. ; Tertre , A. ; Descours , A. ; Berna , P. ; Li , M. Discovery of thiadiazoles as a novel structural class of potent and selective PDE 7 inhibitors, part 2: Metabolism-directed optimization studies towards orally bioavailable derivatives . Bioorg. Med. Chem. Lett. 2004 , 18 ( 14 ), 4615 – 4621 .
   Web of Science ®Google Scholar
• Tale , P. V. ; Deshmukh , S. P. Synthesis of 2-phenylimino-3-aryl-4-S-benzyl-6-hepta-O-acetyl-β-lactosylimini-2,3-dihydro-1,3,5-thiadiazine hydrochlorides . Indian J. Chem. 2006 , 45B , 558 – 560 .
   Google Scholar
• Agrawal , P. T. ; Deshmukh , S. P. Synthesis of 2-phenylimino-3-aryl-4-S-Benzyl-6-hepta-O-benzoyl-β-D-lactosylimino-2,3-dihydro-1,3,5-thiadiazine hydrochlorides . J. Indian Chem. Soc. 2010 , 87 , 1 – 4 .
   Google Scholar
• Thorat , S. M. ; Deshmukh , S. P. Synthesis and antimicrobial activity of N-lactosylated dithiazolidine (hydrochlorides) . Int. J. Chem. Sci. 2010 , 8 ( 2 ), 797 – 802 .
   Google Scholar
• Dyson , G. M. ; Harington , T. The action of chlorine on aryl thiocarbamides and the reactions of aryl isocyanodichlorides . J. Chem. Soc. 1940 , 191 .
   Google Scholar
• Bax , A. ; Egan , W. ; Kovac , P. Synthesis of α-D-lactosyl cluster-nucleoside conjugate . J. Carbohydr. Chem. 1984 , 3 , 593 .
   Web of Science ®Google Scholar
• Kawangh , F. Analytical Microbiology ; Academic Press : New York , 1963 .
   Google Scholar
• (a) Zhigun , D ; Qu , F. ; Wu , C. ; Li , W. A facile method for the synthesis of hepta-O-acetyl-D-lactosyl substituted benzoate . J. Chem. Res. Synop. 2001 , 106 (b) Varma , R. ; Kulkarni , S. Y. ; Jose , C. I. ; Pansare , V. S. Infrared spectral characteristics of some acetyated, anomeric glycosides . Carbohydr. Res. 1984 , 133 , 25 – 32 ; (c) Silverstein , R. M. ; Webster , F.X. ; Spectrometric Identification of Organic Compounds, 6th ed.; John Wiley and Sons: New York, 2004 .
   Google Scholar
• (a) Dyer , J. R. Applications of Absorption Spectroscopy of Organic Compounds, , 8th ed. ; Prentice Hall , 1991 ; (b) Jose , L. ; Blanco , J. ; Saitz , C. B. ; Benito , J. M. ; Mellet , C. O. ; Fuentes , J. ; Gonzalez , F. S. ; Garcia Fernandez , J. M. A practical amine-free synthesis of symmetric ureas and thioureas by self-condensation of iso(thio) cyanates. Synthesis, 1999, 11, 1907 .
   Google Scholar
• Jorgen , L. ; Sigfrid , S. Mass spectrometry in structural analysis of natural carbohydrates . Adv. Carbohydr. Chem Biochem. 1974 , 29 , 41 – 106 ; (b) Budzikiewicz , H. ; Djerassi , C. ; Williams , D. H. Structural Elucidation of Natural Products by Mass Spectrometry, Part II: 2nd ed.; Interscience: New York, 1949 .
   Google Scholar