References and notes
- Knapp , S. and Hale , J. J. 1993 . J. Org. Chem. , 58 : 2650
- Jurczak , J. and Golebiowski , A. 1989 . Chem. Rev. , 89 : 149
- Reetz , M. T. , Drewes , M. W. , Matthews , B. R. and Lennick , K. 1989 . J. Chem. Soc., Chem. Commun , : 1474
- Reetz , M. T. , Drewes , M. W. and Schmidtz , A. 1987 . Angew. Chem. Int. Ed. Engl. , 26 : 1141
- Umezawa , H. , Aoyagi , T. , Suda , H. , Hamada , M. and Takeuchi , T. 1976 . J. Antibiot. , 29 : 97
- Aoyagi , T. , Tobe , H. , Kojima , F. , Hamada , M. , Takeuchi , T. and Umezawa , H. 1987 . J. Antibiot. , 31 : 636
- Herranz , R. , Castro-Pichel , J. and Garcia-Lopez , T. 1989 . Synthesis , : 703
- Umezawa , H. , ed. 1981 . Small Molecular Immunomodifiers of Microbial Origin. Fundamental and Clinical Studies of Bestatin , Tokyo : Japan Scientific Societies Press . and Pergamon Press, Oxford
- Okura , A. , Ishizuka , M. and Takeuchi , T. 1988 . J. Antibiot. , 41 : 261
- Blomgren , H. and Wasserman , J. 1981 . Cancer Lett. , 11 : 303
- Perone , J. J. , Craik , C. S. and Fletterick , R. J. 1993 . Science , 261 : 620
- Singer , P. T. , Smalas , A. , Carty , R. P. , Mangel , W. F. and Sweet , R. M. 1993 . Science , 259 : 669
- Moriarty , R. M. , Liu , K. , Zhuang , H. , Lenz , D. , Brimfield , A. and Xia , C. 1995 . Synth. Commun. , 25 : 2763
- Reetz , M. T. 1984 . Angew. Chem. Int. Ed. Engl. , 23 : 556
- The e.e-values were determined by 1H NMR spectroscopy using (R)-(+)-α-methoxy-α-(trifluoromethyl)phenylacetic acid (Mosher's acid) as a chiral solvating agent.
- Reetz , M. T. , Drewes , M. W. , Lennick , K. , Schmidtz , A. and Holdgrun , X. 1990 . Tetrahedron: Asymmetry , 1 : 375
- Moriarty , R. M. , Zhuang , H. , Penmasta , R. , Liu , K. , Awasthi , A. K. , Tuladhar , S. M. , Rao , M. S. C. and Singh , V. K. 1993 . Tetrahedron Lett. , 34 : 8029
- Freedman , J. , Vaal , M. J. and Huber , E. W. 1991 . J. Org. Chem. , 56 : 670
- Audia , J. E. and Colocci , N. 1991 . Tetrahedron Lett. , 32 : 3779
- Poelert , M. A. , Hulshof , L. A. and Kellogg , R. M. 1994 . Recueil des Travaux Chimiques des Pays Bas (Journal of the Royal Netherlands Chemical Society) , 113 : 355
- α-Amino aldehydes are relatively unstable both chemically and configurationally. They are notoriously prone to racemization during storage and during chromatography on silica gel Jurczak J. Golebiowski A. Chem. Rev. 1989 89 149