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Xenobiotica
the fate of foreign compounds in biological systems
Volume 27, 1997 - Issue 10
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Research Article

Rifampin and rifabutin and their metabolism by human liver esterases

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Pages 1015-1024 | Published online: 22 Sep 2008

References

  • ACOCELLA, G., 1978, Clinical Pharmacokinetics of rifampicin. Clinical Pharmacokinetics, 3, 108–127.
  • ACOCELLA, G., BoNotto, L., MAINARDI M., MARGAROLI, P. and Nicous, F. B., 1974, Kinetic studies on rifampicin. III. Effect of phenobarbital on the half-life of the antibiotic. Tijdschr Gastroentero 17, 151–158.
  • ALDRIDGE W. N., 1953, Serum esterases: Two types of esterases (A and B) hydrolyzing para-nitrophenylacetate, propionate, and a method for their determination. Biochemical Journal, 53, 110–119.
  • BACIEWICZ, A. M., SELF, T. H. and BEKEMEYER, W. B., 1987, Update on rifampin drug interactions. Archives of Internal Medicine, 147, 565–568.
  • BROGDEN, R. N. and FITTON, A., 1994, Rifabutin. A review of its antimicrobial activity, pharmacokinetic properties and therapeutic efficacy. Drugs, 47, 983–1009.
  • COCCHIARA, G., STROLIN BENEDETTI, M., VICARIO, G. P., BALLABIO M., GIOIA, B., VIOGLIO, S. and VIGEVANI, A., 1989, Urinary metabolites of rifabutin, a new antimycobacterial agent, in human volunteers. Xenobiotica, 19, 769–780.
  • FURFSZ, S., 1970, Chemical and biological properties of rifampicin. Antibiotica et Chemotherapia, 16, 316–351.
  • FURESZ, S., Scorn R., PALLANZA, and MAPELLI, E., 1967, Rifampicin: a new rifamycin. 3. Absorption, distribution, and elimination in man. Arzneimittelforschung, 17, 534–537.
  • GRANGE, J. M., WINSTANLEY, P. A. and DAVIES, P. D., 1994, Clinically significant drug interactions with antituberculosis agents. Drug Safety, 11, 242–251.
  • IATSIMIRSKAIA, E., TULEBAEV S., STOROZHUK, E., UTKIN I., SMITH, B. A., GERBER, N. and KOUDRIAKOVA, T., 1997, Metabolism of rifabutin in human enterocyte and liver microsomes : kinetic parameters, identification of enzyme systems, and drug interactions with macrolides and antifungal agents. Clinical Pharmacology and Therapeutics, 61, 554–562.
  • JAMIS -DOW, C. A., KLECICER, R. W., KATKI, A. G. and COLLINS, J. M., 1995, Metabolism of taxol by human and rat liver in vitro: a screen for drug interactions and interspecies differences. Cancer Chemotherapy and Pharmacology, 36, 107–114.
  • LEWIS, R. C., HAIFIELD, N. Z. and NARANG, P. K., 1991, A sensitive method for quantitation of rifabutin and its desacetyl metabolite in human biological fluids by high-performance liquid chromato-graphy (HPLC). Pharmaceutical Research, 8, 1434–1440.
  • MAE, T., HOSOE, K., FUJII, K., YAMASHITA, K., YAMANE, T., HIDAKA T.and OASHI, T., 1996, In vitro metabolism of a rifamycin derivative by animal and human liver microsomes, whole blood and expressed human CYP3A isoform. Xenobiotka, 26, 793–802.
  • MAGGI, N., FURESZ, S., PALLANZA, R. and PELIZZA, G., 1969, Rifampicin desacetylation in the human organism. Arzneimittelforschung, 19, 651–654.
  • MAGGI, N., VIGEVANI, A. and PALLANZA, R., 1968, Desacetyl-rifamycins : preparation and antibacterial properties. Experientia, 24, 209–211.
  • MANDELL G. L. and PETRI, JR., W. A., 1996, Drugs used in the chemotherapy of tuberculosis, Mycobacterium avium complex disease and leprosy. In Goodman and Gilman' s The Pharmacological Basis of Therapeutics, 9th edn, edited by Joel G. Hardman, Lee E. Limbird, Perry B. Molinoff, Raymond W. Ruddon and Alfred Goodman Gilman (New York: McGraw-Hill), pp. 1155–1174.
  • The Merck Index, 12 edn, 1996, edited by S. Budavari (Rahway: Merck & Co.), pp. 1413–1414.
  • PARKINSON, A., 1996, Biotransformation of xenobiotics. In Casaret & Doull's Toxicology: The Basic Science of Poisons, 5th edn, edited by C. D. Klaassen (New York: McGraw-Hill), pp. 113–186.
  • SKINNER, M. H., HSIEH, M., TORSETH, J., PAULOIN, D., BHATIA, G., HARKONEN, S., MERIGAN, T. C. and BLASCHKE, T. F., 1989, Pharmacokinetics of rifabutin. Antimicrobial Agents and Chemotherapy, 33, 1237–1241.
  • STROLIN BENEDETTI, M. and DOSTERT, P., 1994, Induction and autoinduction properties of rifamycin derivatives: a review of animal and human studies. Environmental Health Perspectives, 102 (suppl. 9), 101–105.
  • TRAPNELL, C. B., JAmis -Dow, C., KLECKER, R. W. and COLLINS, J. M., 1997, Metabolism of rifabutin and its 25-desacetyl metabolite, LM565, by human liver microsomes and recombinant human cytochrome P450 3A4: relevance to clinical interaction with fluconazole. Antimicrobial Agents and Chemotherapy, 41, 924–926.
  • VITAL DURAND, D., HAMPDEN, C., BOOBIS, A. R., PARK, B. K. and DAVIES, D. S., 1986, Induction of mixed function oxidase in man by rifapentine (MDL 473), a long-acting rifamycin derivative. British Journal of Clinical Pharmacology, 21, 1–7.
  • WEBER, A., OPHEIM, K. E., SMITH, A. L. and WONG, K., 1983, High-pressure liquid chromatographic quantitation of rifampin and its two major metabolites in urine and serum. Review of Infectious Diseases, 5 (suppl. 3), S433–439.

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