259
Views
9
CrossRef citations to date
0
Altmetric
Original Articles

SOLUBILITY OF ACETAMINOPHEN AND IBUPROFEN IN BINARY AND TERNARY MIXTURES OF POLYETHYLENE GLYCOLS 200 AND 400, PROPYLENE GLYCOL, AND WATER AT 25°C

&

References

  • Acree , Jr. , W. E. ( 1992 ). Mathematical representation of thermodynamic properties. Part II. Derivation of the combined nearly ideal binary solvent (NIBS)/Redlich-Kister mathematical representation from a two-body and three-body interactional mixing model , Thermochim. Acta , 198 , 71 – 79 .
  • Dearden , J. C. , and Patel , N. C. (1978). Dissolution kinetics of some alkyl derivatives of acetaminophen, Drug Dev. Ind. Pharm. , 4, 529–535.
  • Fini , A. , Laus , M. , Orienti , I. , and Zecchi , V. ( 1986 ). Dissolution and partition thermodynamic functions of some nonsteroidal anti-inflammatory drugs , J. Pharm. Sci. , 75 , 23 – 25 .
  • Ishihara , T. , Goto , M. , Kanazawa , H. , Higaki , M. , and Mizushima , Y. ( 2009 ). Efficient entrapment of poorly water-soluble pharmaceuticals in hybrid nanoparticles , J. Pharm. Sci. , 98 , 2357 – 2563 .
  • Jouyban , A. ( 2007 ). Prediction of drug solubility in water-propylene glycol mixtures using Jouyban-Acree model , Pharmazie , 62 , 365 – 367 .
  • Jouyban , A. , and Acree , Jr. , W. E. ( 2006 ). In silico prediction of drug solubility in water-ethanol mixtures using Jouyban-Acree model , J. Pharm. Pharm. Sci. , 9 , 262 – 269 .
  • Jouyban , A. , and Acree , Jr. , W. E. ( 2007 ). Prediction of drug solubility in ethanol-ethyl acetate mixtures at various temperatures using the Jouyban-Acree model , J. Drug Deliv. Sci. Technol. , 17 , 159 – 160 .
  • Jouyban , A. , and Soltanpour , Sh. ( 2010 ). Prediction of dielectric constants of binary solvents at various temperatures , J. Chem. Eng. Data , 55 , 2951 – 2963 .
  • Jouyban , A. , Chan , H. K. , Barzegar-Jalali , M. , and Acree , Jr. , W. E. ( 2002 ). Model to represent solvent effects on the chemical stability of solutes in mixed solvent systems , Int. J. Pharm. , 243 , 167 – 172 .
  • Jouyban , A. , Fathi-Azarbayjani , A. , and Acree , Jr. , W. E. ( 2004 ). Mathematical representation of the density of liquid mixtures at various temperatures using Jouyban-Acree model , Chem. Pharm. Bull. , 52 , 1219 – 1222 .
  • Jouyban , A. , Chan , H. K. , Chew , N. Y. K. , Khoubnasabjafari , M. , and Acree , Jr. , W. E. ( 2006 ). Solubility prediction of paracetamol in binary and ternary solvent mixtures using Jouyban-Acree model , Chem. Pharm. Bull. , 54 , 428 – 431 .
  • Jouyban , A. , Khoubnasabjafari , M. , Vaez-Gharamaleki , Z. , Fekari , Z. , and Acree , Jr. , W. E. ( 2005 ). Calculation of the viscosity of binary liquids at various temperatures using Jouyban-Acree model , Chem. Pharm. Bull. , 53 , 519 – 523 .
  • Jouyban , A. , Shokri , J. , Barzegar-Jalali , M. , Hassanzadeh , D. , Acree , Jr. , W. E. , Ghafourian , T. , and Nokhodchi , A. ( 2009 ). Solubility of chlordiazepoxide, diazepam, and lorazepam in ethanol +water mixtures at 303.2 K , J. Chem. Eng. Data , 54 , 2142 – 2145 .
  • Jouyban , A. , Soltanpour , Sh. , and Acree , Jr. , W. E. ( 2010 ). Improved prediction of drug solubilities in ethanol +water mixtures at various temperatures , Biomed. Int. , 1 , 19 – 24 .
  • Jouyban-Gharamaleki , A. , and Acree , Jr. , W. E. ( 1998 ). Comparison of models for describing multiple peaks in solubility profiles , Int. J. Pharm. , 182 , 177 – 182 .
  • Jouyban-Gharamaleki , A. , Valaee , L. , Barzegar-Jalali , M. , Clark , B. J. , and Acree , Jr. , W. E. ( 1999 ). Comparison of various cosolvency models for calculating solute solubility in water-cosolvent mixtures , Int. J. Pharm. , 171 , 93 – 101 .
  • Manzo , R. H. , and Ahumada , A. A. ( 1990 ). Effects of solvent medium on solubility. V: Enthalpic and entropic contributions to the free energy changes of di-substituted benzene derivatives in ethanol:water and ethanol:cyclohexane mixtures , J. Pharm. Sci. , 79 , 1109 – 1115 .
  • Pacheco , D. P. , Manrique , Y. J. , and Martinez , F. ( 2007 ). Thermodynamic study of the solubility of ibuprofen and naproxen in some ethanol +propylene glycol mixtures , Fluid Phase Equilib. , 262 , 23 – 31 .
  • Paruta , A. N. , and Irani , S. A. ( 1965 ). Dielectric solubility profiles in dioxane-water mixtures for several antipyretic drugs. Effect of substituents , J. Pharm. Sci. , 54 , 1334 – 1338 .
  • Rahbari-Sisakht , M. , Taghizadeh , M. , and Eliassi , A. ( 2003 ). Densities and viscosities of binary mixtures of poly(ethylene glycol) and poly(propylene glycol) in water and ethanol in the 293.15–338.15 K temperature range , J. Chem. Eng. Data , 48 , 1221 – 1225 .
  • Rytting , E. , Lentz , K. A. , Chen , X. Q. , Qian , F. , and Venkatesh , S. ( 2005 ). Aqueous and cosolvent solubility data for drug-like organic compounds , AAPS J. , 7 , E78 – E105 .
  • Soltanpour , Sh. , and Jouyban , A. (2010a). Solubility of acetaminophen and ibuprofen in binary and ternary mixtures of polyethylene glycol 600, ethanol and water, Chem. Pharm. Bull. , 58, 219–224.
  • Soltanpour , Sh. , and Jouyban , A. ( 2010b ). Solubility of acetaminophen and ibuprofen in polyethylene glycol 600, propylene glycol and water mixtures at 25°C , J. Mol. Liq. , 155 , 80 – 84 .
  • Soltanpour , Sh. , and Jouyban , A. ( 2011 ). Solubility of acetaminophen and ibuprofen in polyethylene glycol 600, N-methyl pyrrolidone and water mixtures , J. Solution Chem. , 40 , 2032 – 2045 .
  • Strickley , R. G. ( 2004 ). Solubilizing excipients in oral and injectable formulations , Pharm. Res. , 21 , 201 – 230 .
  • Wilson , K. C. , Reardon , C. , Theodore , A. C. , and Farber , H. W. ( 2005 ). Propylene glycol toxicity: A severe iatrogenic illness in ICU patients receiving IV benzodiazepines: A case series and prospective, observational pilot study , Chest , 128 , 1674 – 1681 .
  • Zar , T. , Graeber , C. , and Perazellat , M. A. ( 2007 ). Recognition, treatment, and prevention of propylene glycol toxicity , Semin. Dial. , 20 , 217 – 219 .
  • Zaslavsky , B. Y. ( 1995 ). Aqueous Two-Phase Partitioning: Physical Chemistry and Bioanalytical Applications , Marcel Dekker , New York .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.