REFERENCES
- Lipinski , C.A. , Lombardo , F. , Dominyl , B.W. , and Feeney , P.J. ( 1997 ) Adv. Drug. Del. Rev. , 23 : 3 – 25 .
- Bashiri , A. and Szabo-Revesz Eros , I.P. ( 2003 ) Pharm. Tech. Eur. , 15 : 27 – 32 .
- Dannenfelser , R. , He , H. , Joshi , Y. , Bateman , S. , and Serajuddin , A.T.M. ( 2004 ) J. Pharm. Sci. , 93 : 1165 – 1175 .
- Vasconcelos , T.F. , Sarmento , B. , and Costa , P. ( 2007 ) Drug Discovery Today , 12 : 1068 – 1075 .
- Leuner , C. and Dressman , J. ( 2000 ) Eur. J. Pharm. Biopharm. , 50 : 47 – 60 .
- Gowariker , V.R. , Viswanathan , N.V. , and Sreedhar , J. ( 1986 ) Polymer Science ; New Delhi , India : New Age Publishers .
- Hancock , B.C. and Zografi , G. ( 1997 ) J. Pharm. Sci. , 86 : 1 – 12 .
- Sekiguchi , K. and Obi , N. ( 1961 ) Chem. Pharm. Bull. , 9 : 866 – 872 .
- Langer , M. , Holtje , M. , Urbanetz , N.A. , Brandt , B. , Holtje , H.D. , and Lippold , B.C. ( 2003 ) Int. J. Pharm. , 252 : 167 – 179 .
- Kapsi , S.G. and Ayres , J.W. ( 2001 ) Int. J. Pharm. , 229 : 193 – 203 .
- Damian , F. , Blaton , N. , Naesens , L. , Balzarini , J. , Kinget , R. , Augustijns , P. , and Van den Mooter , G. ( 2000 ) Eur. J. Pharm. Sci. , 10 : 311 – 322 .
- Van Drooge , D.J. , Hinrichs , W.L.J. , Visser , M.R. , and Frijlink , H.W. ( 2006 ) Int. J. Pharm. , 310 : 220 – 229 .
- Stefanescu , D.M. ( 1988 ) Solidification Processing of Eutectic Alloy ; New York : TMS .
- Pure and Applied Chemistry. ( 1994 ) Definitions of Terms Relating to Phase Transitions of the Solid State ; IUPAC Recommendations 1994, vol. 66, p. 577 .
- Vippagunta , S.R. , Wang , Z. , Hornung , S. , and Krill , S.L. ( 2007 ) J. Pharm. Sci. , 96 : 294 – 304 .
- Naima , Z. , Siro , T. , Juan-Manuel , G.D. , Chantal , C. , Rene , C.L. , and Jerome , D. ( 2001 ) Eur. J. Pharm. Sci. , 12 : 395 – 404 .
- Law , D. , Wang , W. , Schimtt , E.A. , Qiu , Y. , Krill , S.L. , and Fort , J.J. ( 2003 ) J. Pharm. Sci. , 92 : 505 – 515 .
- Lacoulonche , F. , Chauvet , A. , Masse , J. , Egea , M.A. , and Garcia , M.L. ( 1998 ) J. Pharm. Sci. , 87 : 543 – 551 .
- Gordon , M. and Taylor , J.S. ( 1952 ) J. Appl. Chem. , 2 : 493 – 500 .
- Weuts , I. , Kempen , D. , Decorte , A. , Verreck , G. , Peeters , J. , Brewster , M. , and Van den Mooter , G. ( 2005 ) Eur. J. Pharm. Sci. , 25 : 313 – 320 .
- Fiebich , K. and Mutz , M. ( 1999 ) J. Them. Anal. Cal. , 57 : 75 – 85 .
- Van den Mooter , G. , Wuyts , M. , Blaton , N. , Busson , R. , Grobet , P. , Augustijns , P. , and Kinget , R. ( 2001 ) Eur. J. Pharm. Sci. , 12 : 261 – 269 .
- Heo , M.Y. , Piao , Z.Z. , Kim , T.W. , Cao , Q.R. , Kim , A. , and Lee , B.J. ( 2005 ) Arch. Pharm. Res. , 28 : 604 – 611 .
- Damian , F. , Blaton , N. , Kinget , R. , and Van den Mooter , G. ( 2002 ) Int. J. Pharm. , 244 : 87 – 98 .
- Gupta , P. , Thilagavathi , R. , Chakraborti , A.S. , and Bansal , A.K. ( 2005 ) Mol. Pharm. , 2 : 84 – 391 .
- Drooge , D.J.V. , Hinrichs , W.L.J. , Visser , M.R. , and Frijlink , H.W. ( 2006 ) Int. J. Pharm. , 310 : 220 – 229 .
- Weuts , I. , Kempen , D. , Verreck , G. , Peeters , J. , Brewster , M. , Blaton , N. , and Van den Mooter , G. ( 2005 ) Eur. J. Pharm. Sci. , 25 : 387 – 393 .
- Shibata , Y. , Fuji , M. , Kokudai , M. , Noda , S. , Okada , H. , Kondoh , M. , and Watanabe , Y. ( 2007 ) J. Pharm. Sci. , 96 : 1537 – 1547 .
- Higuchi , W.I. , Mir , N.A. , and Desai , S.J. ( 1965 ) J. Pharm. Sci. , 54 : 1404 – 1410 .
- Craig , D.Q.M. ( 2001 ) Int. J. Pharm. , 231 : 131 – 144 .
- Serajuddin , A.T.M. ( 1999 ) J. Pharm. Sci. , 88 : 1058 – 1066 .
- Karavas , E. , Georgarakis , E. , Sigalas , M.P. , Avgoustakis , K. , and Bikiaris , D. ( 2007 ) Eur J. Pharm. Biopharm. , 66 : 334 – 347 .
- Muhrer , G. , Meier , U. , Fusaro , F. , Albano , S. , and Mazzotti , M. ( 2006 ) Int. J. Pharm. , 308 : 69 – 83 .
- Lofftsson , T. and Brewster , M.E. ( 1997 ) J. Pharm. Sci. , 85 : 1017 – 1025 .
- Henck , J.O. , Griesser , U.J. , and Burger , A. ( 1997 ) Pharm. Ind. , 59 : 165 – 169 .
- Smikalla , M.M. and Urbanetz , N.N. ( 2007 ) Eur J. Pharm. Sci. , 66 : 106 – 112 .
- Yoshioka , M. and Hancock , B.C. ( 1995 ) J. Pharm. Sci. , 84 : 983 – 986 .
- Ambike , A.A. , Mahadik , K.R. , and Paradkar , A. ( 2004 ) Int. J. Pharm. , 282 : 151 – 162 .
- Sertsou , G. , Butler , J. , Scott , A. , Hempenstall , J. , and Rades , T. ( 2002 ) Int. J. Pharm. , 245 : 99 – 108 .
- Gunawan , L. , Johari , G.P. , and Shanker , R.M. ( 2006 ) Pharm. Res. , 23 : 967 – 979 .
- Miyazaki , T. , Yoshioka , S. , Aso , Y. , and Kojima , S. ( 2004 ) J. Pharm Sci. , 93 : 2710 – 2717 .
- Karel , S. , Geert , V. , Jef , Peeters. , Brewster , M. , and Van den Mooter , G. ( 2004 ) J Pharm Sci. , 93 : 124 – 131 .
- Dhumal , R.S. , Shimpi , S.L. , Paradkar , A.R. ( 2007 ) Acta Pharm. , 57 : 287 – 300 .
- School of Pharmacy, London . ( 2006 ). Solid dispersion of hydrophobic bioactive. Pat. No. WO/2006/085089 .
- Drooge , D.J.V. , Hinrichs , W.L.J. , and Frijlink , H.W. ( 2004 ) J. Pharm. Sci. , 93 : 713 – 725 .
- Ningyun , S. , Xiuli , Wei. , Baojian , W. , Jian , C. , Yi , L. , and Wei , W. ( 2008 ) Powder Technol. , 182 : 72 – 80 .
- Newa , M. , Bhandari , K.H. , Li , D.X. , Kwon , T. , Kim , J.A. , Yoo , B.K. , Woo , J.S. , Lyoo , W.S. , Yong , C.S. , and Choi , H.G. (2007) Int. J. Pharm. , 343: 228–237.
- Yamashita , K. , Nakate , T. , Okimoto , K. , Ohike , A. , Tokunaga , Y. , Ibuki , R. , Higaki , K. , and Kimura , T. ( 2003 ) Int J. Pharm. , 267 : 79 – 91 .
- Nilüfer , Y. , Aysegül , K. , Yalçı , Ö. , Ayhan , S. , Sibel , A.Ö. , and Tamer , B. ( 2003 ) Eur. J. Pharm. Biopharm. , 56 : 453 – 45 .
- Sethia , S. and Squillante , E. ( 2004 ) J. Pharm. Sci. , 93 : 2985 – 2993 .
- Barker , S.A. , Yap , S.P. , Yuen , K.H. , McCoy , C.P. , Murphy , J.R. , and Craig , D.Q.M. ( 2003 ) J. Control. Rel. , 91 : 477 – 488 .
- Zerrouk , N. , Chemtob , C. , Arnaud , P. , Toscani , S. , and Dugue , J. ( 2001 ) Int. J. Pharm. , 225 : 49 – 62 .
- Timko , R.J. and Lordi , N.G. ( 1979 ) J. Pharm. Sci. , 68 : 601 – 605 .
- Lin , C.W. and Cham , T.M. ( 1996 ) Int. J. Pharm. , 22 : 909 – 916 .
- Allen , L.V. and Yanchick , V.A. ( 1977 ) J. Pharm. Sci. , 66 : 494 – 497 .
- Summers , M.P. and Enever , R.P. ( 1976 ) J. Pharm. Sci. , 65 : 1613 – 1618 .
- The role of plasticizers as functional excipients in pharmaceutical dosage forms prepared by hot-melt extrusion. (2004) Pharmaceutical Coatings Bulletin , 102 : 6 .
- Van Laarhoven , J.A.H. , Kruft , M.A.B. , and Vromans , H. ( 2002 ) Int. J. Pharm. , 232 : 163 – 173 .
- Nakamichi , K. , Yasuura , H. , Fukui., Oka , M. , and Izumi , S. ( 2001 ) Int. J. Pharm. , 218 : 103 – 112 .
- Munch , U. , Mika , H.J. , Eschermann , B. , Schmidt , R. , and Sczepanik , B. ( 1990 ) Orally administered solvent free pharmaceutical preparation with delayed active substance release and a method of preparing the preparation . Eur. Patent 0,552,227 .
- Grunhagen , H.H. ( 1996 ) Pharm. Tech. Eur. , 8 : 22 – 28 .
- Ozkan , Y. , Doganay , N. , Dikmen , N. , and Isimer , A. ( 2000 ) Il Farmaco , 55 : 433 – 438 .
- Huelsmanna , S. , Backensfelda , T. , Keitela , S. , and Bodmeier , R. ( 2000 ) Eur. J. Pharm. Sci. , 49 : 237 – 242 .
- Li , F. and Hu , J. ( 2004 ) Chem. Pharm. Bull. , 52 : 972 – 973 .
- Zajc , N. , Obreza , A. , Bele , M. , and Ca , S.S.C. ( 2005 ) Int. J. Pharm. , 291 : 51 – 58 .
- Finia , A. , Moyanob , J.R. , Ginesb , J.M. , Perez-Martinezb , J.I. , and Rabasco , A.M. ( 2005 ) Eur. J. Pharm. Sci. , 60 : 99 – 111 .
- Mooter , G.V.D. , Weuts , I. , Ridder , T.D. , and Blaton , N. ( 2006 ) Int. J. Pharm. , 316 : 1 – 6 .
- Bulau , H.C. , Ulrich , J. ( 1997 ) In Parameters Influencing the Properties of Drop-Formed Pastilles , edited by J. Ulrich ; Aachen , Germany : Shaker Verlag .
- Francois , D. and Jones , B.E. ( 1978 ) The hard capsule with the soft center. Paper presented at the European Capsule Technology Symposium, October 11–13.
- Serajuddin , A.T.M. , Sheen , P.C. , Mufson , D. , Bernstein , D.F. , and Augustine , M.A. ( 1988 ) J. Pharm. Sci. , 77 : 414 – 418 .
- Joshi , H.N. , Tejwani , R.W. , Davidovich , M. , Sahasrabudhe , V.P. , and Mohammed Serajuddin , A.T.M. ( 2004 ) Int. J. Pharm. , 269 : 251 – 258 .
- Law , S.L. , Lo , W.Y. , Lin , F.M. , and Chaing , C.H. ( 1992 ) Int. J. Pharm. , 84 : 161 – 166 .
- Wiley , G.J. , Ullah , I. , and Agharkar , S.N. ( 1995 ) Pharm. Tech. , 19 : 72 – 76 .
- Habib , M.J. ( 2000 ) Pharmaceutical Solid Dispersion Technology ; Washington , DC : CRC Press .
- Law , D. , Krill , S.L. , Schmitt , E.A. , Fort , J.J. , Qiu , Y. , Wang , W. , and Porter , W.R. ( 2000 ) J. Pharm. Sci. , 90 : 1015 – 1025 .
- Mooter , G.V.D. , Augustijns , P. , Blaton , N. , and Kinget , R. ( 1998 ) Int. J. Pharm. , 164 : 67 – 80 .
- Franco , M. , Trapani , G. , Latrofa , A. , Tullio , C. , Provenzano , M.R. , Serra , M. , Muggironi , M. , Biggio , G. , and Liso , G. ( 2001 ) Int. J Pharm. , 225 : 63 – 73 .
- Prabhu , S. , Brocks , D.R. , and Betageri , G.V. ( 2001 ) Drug. Dev. Ind. Pharm. , 27 : 413 – 418 .
- Babu , G.V.M. , Prasad , D.S. , and Murthy , K.V.R. ( 2002 ) Int. J. Pharm. , 234 : 1 – 17 .
- Pignatello , R. , Ferro , M. , Guidi , G.D. , Salemi , G. , Vandelli , M.A. , Guccione , S. , Geppi , M. , Forte , C. , and Puglisi , G. ( 2001 ) Int. J. Pharm. , 218 : 27 – 42 .
- Abdul-Fattah , A.M. and Bhargava , H.N. ( 2002 ) Int. J. Pharm. , 235 : 17 – 33 .
- Orientia , I. , Biguccia , F. , Luppia , B. , Cerchiaraa , T. , Zuccaria , G. , and Giunchedib , P. , and Zecchi , V. ( 2002 ) Eur. J. Pharm. Sci. , 54 : 229 – 233 .
- Sang-Chul , S. and Kim , J. ( 2003 ) Int. J. Pharm. , 251 : 79 – 84 .
- Watanabe , T. , Hasegawa , S. , Wakiyama , N. , Kusai , A. , and Senna , M. ( 2003 ) Int. J. Pharm. , 250 : 283 – 286 .
- Yamashita , K. , Nakate , T. , Okimoto , K. , Ohike , A. , Tokunaga , Y. , Ibuki , R. , Higaki , K. , and Kimura , T. ( 2003 ) Int. J. Pharm. , 267 : 79 – 86 .
- Ruan , L. , Yu , B. , Fu , G. , and Zhu , D. ( 2005 ) J. Phar. Bio. Anal. , 38 : 457 – 464 .
- Nijlen , T.V. , Brennan , K. , Mooter , D.V.G. , Blaton , N. , Kinget , R. , and Augustijns , P. ( 2003 ) Int. J. Pharm. , 254 : 173 – 185 .
- Drooge , V.J.D. , Hinrichs , W.L.J. , Wegman , K.A.M. , Visser , M.R.A. , Eissens , C. , and Frijlink , H.W. ( 2004 ) Eur. J. Pharm. Biopharm. , 21 : 511 – 518 .
- Mooter , D.V.G. , Weuts , I. , Ridder , T.D. , and Blaton , N. ( 2006 ) Int. J. Pharm. , 316 : 1 – 6 .
- Gong , K. , Viboonkiat , R. , Rehman , L.U. , Buckton , G. , and Darr , J.A. ( 2005 ) J. Pharm Sci. , 94 : 2583 – 2590 .
- Beten , D.B. , Amighi , K. , and Moes , A.J. ( 1995 ) Pharm. Res. , 12 : 1269 – 1272 .
- Ho , H.O. , Shu , H.L. , Tsai , T. , and Sheu , M.T. T. ( 1996 ) Int. J. Pharm. , 139 : 223 – 229 .
- Overhoff , K.A. , Moreno , A. , Miller , D.A. , Johnston , K.P. , and Williams , R.O. ( 2007 ) Int. J. Pharm. , 336 : 122 – 132 .
- Satio , M. , Ugajin , T. , Nozawa , Y. , Sadzuka , Y. , Miyagishima , A. , and Sonobe , T. ( 2002 ) Int. J. Pharm. , 249 : 71 – 79 .
- Fujii , M. , Okada , H. , Shibata , Y. , Teramachi , H. , Kondoh , M. , and Watanabe , Y. ( 2005 ) Int. J. Pharm. , 293 : 145 – 153 .
- Reneker , D.H. and Chun , I. (1996) Nanotechnology , 7: 216–223.
- Deitzel , J.M. , Kleinmeyer , J. , Harris , D. , and Beck , T.N.C. ( 2001 ) Polym. , 42 : 261 – 272 .
- Dennis , A.B. , Farr , S.J. , Kellaway , I.W. , Taylor , G. , and Davidson , R. ( 1990 ) Int. J. Pharm. , 65 : 85 – 100 .
- Remunan , C. , Bretal , M. , Nunez , A. , and Vila , J.L. ( 1992 ) Int. J. Pharm. , 80 : 151 – 157 .
- Vila , J.L.J. , Remunan , C. , and Martinez , R. ( 1990 ) S.T.P. Pharm. , 6 : 88 – 92 .
- Sharma , P.K. , Chaudhari , P.D. , Badagale , M.M. , Dave , K.D. , Kulkarni , P.A. , and Barhate , N.S. ( 2006 ) Current trends in solid dispersions techniques . Pharmainfo. Net , 17 May .
- Gattefosse Technical Brochure . ( 1999 ) Pharmaceutical Excipient for Oral Semisolids Formulations , pp. 12 – 15 .
- Sutananta , W. , Craig , D.Q.M. , and Newton , J.M. ( 1995 ) J. Pharm. Pharmacol. , 47 : 355 – 359 .
- Jones , M.C. and Leroux , J.C. ( 1999 ) Eur. J. Pharm. Biopharm. , 48 : 101 – 108 .
- Vippagunta , S.R. , Maul , K.A. , Tallavajhala , S. , and Grant , D.J.W. ( 2002 ) Int. J. Pharm. , 236 : 111 – 123 .
- Chen , Y. , Zhang , G.G.Z. , Neilly , J. , Marsh , K. , Mawhinney , D. , and Sanzgiri , Y.D. ( 2004 ) Int. J. Pharm. , 286 : 69 – 80 .
- Lasic , D.D. ( 1993 ) Liposomes: From Physics to Applications ; Amsterdam , the Netherlands : Elsevier .
- Zidan , A.S. , Habib , M.J. , and Khan , M.A. ( 2007 ) J. Pharm. Sci. , 97 : 3388 – 3399 .
- Biswas , M. , Akogyeram , C.O. , Scott , K.R. , Potti , G.K. , Gallelli , J.F. , and Habib , M.J. ( 1993 ) J. Controlled Rel. , 23 : 239 – 245 .
- Hamdani , J. , Moes , A.J. , and Amighi , K. ( 2003 ) Int. J. Pharm. , 260 : 47 – 57 .
- Chauhan , B. , Shimpi , S. , and Paradkar , A. ( 2005 ) AAPS Pharm. Sci. Tech. , 6 .
- Kerc , J. and Srcic , S. ( 1995 ) Thermochim. Acta 248 : 81 – 95 .
- Giron , D. ( 1990 ) Jugosl. , 40 : 95 – 157 .
- Giron , D. ( 1995 ) Thermochim. Acta 248 : 1 – 59 .
- Leng , Y. ( 2008 ) Materials Characterization: Introduction to Microscopic and Spectroscopic Methods . New York : John Wiley .
- Schafer , R.J. ( 1994 ) Dynamic Properties of Rubber: The Glass Transition Temperature . Lippincott and Peto, New York, Rubber World (Magazine/Journal).
- Plastics Differential Scanning Calorimetry (DSC) Part 2: Determination of Glass Transition Temperature (1999) ISO 11357–2:1999. Distributed through American National Standards Institute (ANSI) .
- Qi , S. , Gryczke , A. , Belton , P. , and Craig , D.Q.M. ( 2008 ) Int. J. Pharm. , 354 : 158 – 167 .
- Gupta , P. and Bansal , A.K. ( 2005 ) AAPS Pharm. Sci. Tech. , 6 : E223 – E230 .
- Chauhan , B. , Shimpi , S. , and Paradkar , A. ( 2005 ) Eur. J. Pharm. Sci. , 26 : 219 – 230 .
- Fini , A. , Cavallari , C. , and Ospitali , F. ( in press ) Eur. J Pharm Biopharm. , 70 : 409 – 420 .
- Dong , Z. , Chatterji , A. , Sandhu , H. , Choi , D.S. , Chokshi , H. , and Shah , N. ( 2008 ) Int. J. Pharm. , 355 : 141 – 149 .
- Wang , X. , Armas , H.N. , Blaton , N. , Michoel , A. , and Mooter , G.V. ( 2007 ) Int. J. Pharm. , 345 : 95 – 100 .
- Vrentas , J.S. and Vrentas , C.M. ( 1991 ) Macromolecules , 24 : 2404 – 2412 .
- Andronis , V. , Yoshioka , M. , and Zografi , G. ( 1997 ) J. Pharm. Sci. , 86 : 346 – 351 .
- Galop , M. ( 2005 ) Pharm. Res. , 22 : 293 – 302 .
- Hasegawa , S. , Hamaura , T. , Furuyama , N. , Horikawa , S. , Kusai , A. , Yonemochi , E. , and Terada , K. ( 2004 ) Int. J. Pharm. , 280 : 39 – 46 .
- Parikh , D.M. ( 1997 ) Handbook of Pharmaceutical Granulation Technology ; New York : Marcel Dekker .
- Bikiaris , D. , Papageorgiou , G.J. , Stergiou , A. , Pavlidou , E. , Karavas , E. , Kanaze , F. , and Georgarakis , M. ( 2005 ) Therm. Acta 439 : 58 – 67 .
- Karavas , E. , Ktistis , G. , Xenakis , A. , and Georgarakis , E. ( 2006 ) Eur J. Pharm. Biopharm. , 63 : 103 – 114 .
- Schachter , D.M. , Xiong , J. , and Tirol , G.C. ( 2004 ) Int. J. Pharm. , 281 : 89 – 101 .