Formulation and Development of Self-Nanoemulsifying Granules of Olmesartan Medoxomil for Bioavailability Enhancement

References

• Azeem , A. , M. Rizwan , F. J. Ahmad , Z. Iqbal , R. K. Khar , et al. . 2009 . Nanoemulsion components screening and selection: a technical note . AAPS PharmSciTech 10 : 69 – 76 .
   PubMed Web of Science ®Google Scholar
• Balakrishnan , P. , B. Lee , D. O. Hoon , J. O. Kim , M. J. Hong , et al. . 2009 . Enhanced oral bioavailability of dexibuprofen by a novel solid Self-emulsifying drug delivery system (SEDDS) . Eur. J. Pharm. Biopharm. 72 : 539 – 45 .
   PubMed Web of Science ®Google Scholar
• Bandivadeka , M. M. , S. S. Pancholi , R. Kaul-Ghanekar , A. Choudhari , and S. Koppikar . 2012 . Self-microemulsifying smaller molecular volume oil (Capmul MCM) using non-ionic surfactants: a delivery system for poorly water-soluble drug . Drug Dev. Ind. Pharm. 38 : 883 – 892 .
   PubMed Web of Science ®Google Scholar
• Bandyopadhyay , S. , O. P. Katare , and B. Singh . 2012 . Optimized self nano-emulsifying systems of ezetimibe with enhanced bioavailability potential using long chain and medium chain triglycerides . Colloids Surf. B 100 : 50 – 61 .
   PubMed Web of Science ®Google Scholar
• Bing , S. , T. Jingling , J. Hongyu , L. Hongmei , L. Yan , Z. Daling , and W. Linhua . 2010 . Enhanced oral bioavailability of wurenchun (fructus schisandrae chinensis extracts) by self-emulsifying drug delivery systems . Drug Dev. Ind. Pharm. 36 : 1356 – 1363 .
   PubMed Web of Science ®Google Scholar
• Brahmankar , D. M. , and B. S. Jaiswal . 1987 . Biopharmaceutics and pharmacokinetics: A treatise . New Delhi : Vallabh Prakashan .
   Google Scholar
• Carr , R. L. 1965 . Evaluating flow properties of solids. Evaluating flow properties of solids . Chem. Eng. 72 : 163 – 168 .
   Google Scholar
• Chakraborty , S. , D. Shukla , B. Mishra , and S. Singh . 2009 . Lipid—An emerging platform for oral delivery of drugs with poor bioavailability . Eur. J. Pharm. Biopharm. 73 : 1 – 15 .
   PubMed Web of Science ®Google Scholar
• Chen , M. 2008 . Lipid excipients and delivery systems for pharmaceutical development: A regulatory perspective. Adv . Drug Del. Rev. 60 : 768 – 777 .
   PubMed Web of Science ®Google Scholar
• Costa , P. , and J. M. S. Lobo . 2001 . Modeling and comparison of dissolution profiles . Eur. J. Pharm. 13 : 123 – 33 .
   Web of Science ®Google Scholar
• Desai , P. P. , A. A. Date , and V. B. Patravale . 2012 . Overcoming poor oral bioavailability using nanoparticle formulations—Opportunities and limitations . Drug Discovery Today 9 : 87 – 95 .
   Google Scholar
• Devane , J. 1998 . Oral drug delivery technology: Addressing the solubility/permeability paradigm . Pharm. Technol. 22 : 68 – 74 .
   Google Scholar
• Dixit , R. P. , and M. S. Nagarsenker . 2008 . Self-nanoemulsifying granules of ezetimibe: Design, optimization and evaluation . Eur. J. Pharm. 35 : 183 – 192 .
   Web of Science ®Google Scholar
• Emad , B. B. , S. Nevine , and M. B. Shaimaa . 2010 . SNEDDS containing bioenhancers for improvement of dissolution and oral absorption of lacidipine. I: Development and optimization . Int. J. Pharm. 391 : 203 – 211 .
   PubMed Web of Science ®Google Scholar
• Ghosh , M. N. 2008 . Fundamentals of experimental pharmacology . Calcutta : SK Ghosh & Others .
   Google Scholar
• Gupta , S. , S. Chavhan , and K. K. Sawant . 2011 . Self nanoemulsifying drug delivery system for adefovir dipivoxil: Design, characterization, in vitro and ex vivo evaluation . Colloids Surf. A 392 : 145 – 155 .
   Web of Science ®Google Scholar
• Jannin , V. , J. Musakhanian , and D. Marchaud . 2008 . Approaches for the development of solid and semi-solid lipid-based formulations . Adv. Drug Del. Rev. 2008 , 60 : 734 – 746 .
   PubMed Web of Science ®Google Scholar
• Kallakunta , V. R. , S. Bandari , R. Jukanti , and P. R. Veerareddy . 2012. Oral self-emulsifying powder of lercanidipine hydrochloride: Formulation and evaluation. Powder Technol. 221:375–382.
   Web of Science ®Google Scholar
• Mahmoud , E. A. , E. R. Bendas , and M. I. Mohamed . 2009 . Preparation and evaluation of self-nanoemulsifying tablets of carvedilol . AAPS PharmSciTech 10 : 183 – 192 .
   PubMed Web of Science ®Google Scholar
• Martin , A. 1993 . Physical pharmacy, 4th ed . Philadelphia : Lippincott Williams & Wilkins .
   Google Scholar
• Mashru , P. P. , V. B. Sutariya , M. G. Sankalia , and P. P. Parikh . 2005 . Development and evaluation of fast-dissolving film of salbutamol sulphate . Drug Dev. Ind. Pharm. 31 : 25 – 34 .
   PubMed Web of Science ®Google Scholar
• Maurya , D. P. , Y. Sultana , M. Aqil , B. P. Panda , and A. F. Ali . 2011 . Formulation and optimization of alkaline extracted ispaghula husk microscopic reservoirs of isoniazid by box-behnken statistical design . J. Dispersion Sci. Technol. 32 : 424 – 432 .
   Web of Science ®Google Scholar
• Mukherjee , T. , and F. M. Plakogiannis . 2010 . Development and oral bioavailability assessment of a supersaturated self-microemulsifying drug delivery system (SMEDDS) of albendazole . J. Pharm. Pharmacol. 62 : 1112 – 1120 .
   PubMed Web of Science ®Google Scholar
• Mustafa , G. , Z. I. Khan , T. Bansal , and S. Talegaonkar . 2009 . Preparation and characterization of oil in water nano-reservoir systems for improved oral delivery of atorvastatin . Curr. Nanosci. 5 : 428 – 440 .
   Web of Science ®Google Scholar
• Myung , J. K. , Y. J. Soo , H. S. Woo , S. P. Jun , C. Sung-Up , et al. . 2011 . Immediate release of ibuprofen from Fujicalin-based fast dissolving self-emulsifying tablets . Drug Dev. Ind. Pharm. 37 : 1298 – 1305 .
   PubMed Web of Science ®Google Scholar
• Nazzal , S. , and M. A. Khan . 2006 . Controlled release of a self-emulsifying formulation from a tablet dosage form: Stability assessment and optimization of some processing parameters . Int. J. Pharm. 315 : 110 – 121 .
   PubMed Web of Science ®Google Scholar
• Nekkanti , V. , P. Karatgi , R. Prabhu , and R. Pillai . 2010 . Solid self-microemulsifying formulation for candesartan cilexetil . AAPS PharmSciTech 11 : 9 – 17 .
   PubMed Web of Science ®Google Scholar
• Newton , J. M. , M. R. Pinto , and F. Podczeck . 2007 . The preparation of pellets containing a surfactant or a mixture of mono- and di-glycerides by extrusion/spheronization . Eur. J. Pharm. 30 : 333 – 342 .
   Web of Science ®Google Scholar
• Noyes , A. , and W. Whitney . 1987 . The rate of solution of solid substances in their own solutions . J. Am. Chem. Soc. 19 : 930 – 934 .
   Google Scholar
• Patel , N. V. , J. K. Patel , and S. H. Shah . 2010 . Box Behnken experimental design in the development of pectin-compritol ATO 888 compression coated colon targeted drug delivery of mesalamine . Acta Pharm. 60 : 39 – 54 .
   PubMed Web of Science ®Google Scholar
• Singh , B. , R. Kumar , and N. Ahuja . 2005 . Optimizing drug delivery systems using systematic “design of experiments.” Part I: Fundamental aspects . Crit. Rev. Ther. Drug Carrier Syst. 22 : 27 – 105 .
   PubMed Web of Science ®Google Scholar
• Singh , K. K. , K. K. Srinivasan , K. Gowthamarajan , D. S. Singare , D. Prakash , and N. B. Gaikwad . 2011 . Investigation of preparation parameters of nanosuspension by top-down media milling to improve the dissolution of poorly water-soluble glyburide . Eur. J. Pharm. Biopharm. 78 : 441 – 446 .
   PubMed Web of Science ®Google Scholar
• Villar , A. M. S. , B. C. Naveros , A. C. C. Campmany , M. A. Trenchs , C. B. Rocabert , and L. H. Bellow . 2012 . Design and optimization of self-nanoemulsifying drug delivery systems (SNEDDS) for enhanced dissolution of gemfibrozil . Int. J. Pharm. 431 : 161 – 175 .
   PubMed Web of Science ®Google Scholar
• Yi , T. , J. Wan , H. Xu , et al. . 2008 . A new solid self-microemulsifying formulation prepared by spray-drying to improve the oral bioavailability of poorly water soluble drugs . Eur. J. Pharm. Biopharm. 70 : 439 – 444 .
   PubMed Web of Science ®Google Scholar
• Yinghui , W. , Y. Xiaoli , S. Xiaoguang , P. Xuan , B. Qiang , L. Minchen , G. Manman , and L. Fanzhu . 2012 . Enhanced oral bioavailability of silybin by a supersaturatable self-emulsifying drug delivery system (S-SEDDS) . Colloids Surf. A 396 : 22 – 28 .
   Web of Science ®Google Scholar
• Yosra , S. R. E. , A. E. Magda , and Y. A. Ossama . 2009 . Self-nanoemulsifying drug delivery systems of tamoxifen citrate: Design and optimization . Int. J. Pharm. 380 : 133 – 141 .
   PubMed Web of Science ®Google Scholar
• Zhao , Y. , C. Wang , A. H. L. Chow , K. Ren , T. Gong , Z. Zhang , and Y. Zheng . 2010 . Self-nanoemulsifying drug delivery system (SNEDDS) for oral delivery of Zedoary essential oil: Formulation and bioavailability studies . Int. J. Pharm. 283 : 170 – 177 .
   Web of Science ®Google Scholar
• Zidan , A. S. , and M. Mokhtar . 2011 . Multivariate optimization of formulation variables influencing flurbiprofen proniosomes characteristics . J. Pharm. Sci. 100 : 2212 – 2221 .
   PubMed Web of Science ®Google Scholar