831
Views
27
CrossRef citations to date
0
Altmetric
Research Article

Evaluation about wettability, water absorption or swelling of excipients through various methods and the correlation between these parameters and tablet disintegration

, , , &
Pages 1417-1425 | Received 07 Aug 2017, Accepted 28 Feb 2018, Published online: 06 Apr 2018

References

  • Desai PM, Liew CV, Heng PW. Review of disintegrants and the disintegration phenomena. J Pharm Sci. 2016;105:2545–2555.
  • Slavkova M, Breitkreutz J. Orodispersible drug formulations for children and elderly. Eur J Pharm Sci. 2015;75:2–9.
  • Guyot-Herman AM. Tablet disintegration and disintegrating agents. STP Pharma Sci. 1992;2445–462.
  • Chamsai B, Sriamornsak P. Novel disintegrating microcrystalline cellulose pellets with improved drug dissolution performance. Powder Technol. 2013;233:278–285.
  • Sieber D, Lazzari A, Quodbach J, et al. Applicability of two automated disintegration apparatuses for rapidly disintegrating (mini)tablets. Pharm Dev Technol. 2017;22:198–205.
  • Yoshida M, Hazekawa M, Haraguchi T, et al. Evaluation of the palatabilities in 10 different famotidine orally disintegrating tablets by combination of disintegration device and taste sensor. Drug Dev Industr Pharm. 2015;41:1387–1392.
  • Quodbach J, Kleinebudde P. A critical review on tablet disintegration. Pharm Dev Technol. 2016;21:763–774.
  • Markl D, Zeitler JA. A review of disintegration mechanisms and measurement techniques. Pharm Res. 2017;34:890–917.
  • Quodbach J, Kleinebudde P. Systematic classification of tablet disintegrants by water uptake and force development kinetics. J Pharm Pharmacol. 2014;66:1429–1438.
  • Yamamoto Y, Fujii M, Watanabe K, et al. Effect of powder characteristics on oral tablet disintegration. Int J Pharm. 2009;365:116–120.
  • Yoshinori O, Kosugi A, Hamaguchi M, et al. A comparative study of disintegration actions of various disintegrants using Kohonen’s self-organizing maps. J Drug Deliv Sci Technol. 2018;43:141–148.
  • Chaheen M, Soulairol I, Bataille B, et al. Chitin’s functionality as a novel disintegrant: benchmarking against commonly used disintegrants in different physicochemical environments. J Pharm Sci. 2017;106:1839–1848.
  • Wang C, Huang H, Jia M, et al. Formulation and evaluation of nanocrystalline cellulose as a potential disintegrant. Carbohydr Polym. 2015;130:275–279.
  • Kamiya T, Kondo H, Hiroma H, et al. Impact of process parameters on Mg–St content and tablet surface wettability in the external lubrication method for a rotary tablet press. Adv Powder Technol. 2016;27:193–198.
  • Alghunaim A, Kirdponpattara S, Newby BZ. Techniques for determining contact angle and wettability of powders. Powder Technol. 2016;287:201–215.
  • Kirdponpattara S, Phisalaphong M, Newby BM. Applicability of Washburn capillary rise for determining contact angles of powders/porous materials. J Colloid Interf Sci. 2013;397:169–176.
  • Hammes MV, Englert AH, Noreña CPZ, et al. Effect of water activity and gaseous phase relative humidity on microcrystalline cellulose water contact angle measured by the Washburn technique. Colloids Surf A Physicochem Eng Asp. 2016;500:118–126.
  • Bormashenko E. Contact angles of rotating sessile droplets. Colloids Surf A Physicochem Eng Asp. 2013;432:38–41.
  • Hooper P, Lasher J, Alexander KS, et al. A new modified wetting test and an alternative disintegration test for orally disintegrating tablets. J Pharm Biomed Anal. 2016;120:391–396.
  • Harada T, Narazaki R, Nagira S, et al. Evaluation of the disintegration properties of commercial famotidine 20 mg orally disintegrating tablets using a simple new test and human sensory test. Chem Pharm Bull. 2006;54:1072–1075.
  • Iwao Y, Tanaka S, Uchimoto T, et al. An easy-to-use approach for determining the disintegration ability of disintegrants by analysis of available surface area. Int J Pharm. 2013;448:1–8.
  • Bele MH, Derle DV. Mechanism of disintegrant action of polacrilin potassium: swelling or wicking? Acta Pharm Sinica B. 2012;2:70–76.
  • Ken Welch MS. Simultaneous measurement of drug release and liquid uptake in pharmaceutical tablets. J Pharm Sci. 2003;92:1242–1249.
  • Thoorens G, Krier F, Leclercq B, et al. Microcrystalline cellulose, a direct compression binder in a quality by design environment—a review. Int J Pharm. 2014;473:64–72.
  • Gamble JF, Chiu W-S, Tobyn M. Investigation into the impact of sub-populations of agglomerates on the particle size distribution and flow properties of conventional microcrystalline cellulose grades. Pharm Dev Technol. 2010;16:542–548.
  • Elkomy MH, El Menshawe SF, Abou-Taleb HA, et al. Loratadine bioavailability via buccal transferosomal gel: formulation, statistical optimization, in vitro/in vivo characterization, and pharmacokinetics in human volunteers. Drug Deliv. 2017;24:781–791.
  • Rodriguez Amado JR, Prada AL, Duarte JL, et al. Development, stability and in vitro delivery profile of new loratadine-loaded nanoparticles. Saudi Pharm J. 2017;25:1158–1168.
  • Heshmati M, Piri M. Experimental investigation of dynamic contact angle and capillary rise in tubes with circular and noncircular cross sections. Langmuir. 2014; 30:14151–14162.
  • Ji L, Shi B. A novel method for determining surface free energy of powders using Washburn’s equation without calculating capillary factor and contact angle. Powder Technol. 2015;271:88–92.
  • Holysz ECaL. Use of the Washburn equation for surface free energy determination. Langmuir. 1992;8:710–716.
  • Yang B, Xu L, Wang Q, et al. Modulation of the wettability of excipients by surfactant and its impacts on the disintegration and release of tablets. Drug Dev Ind Pharm. 2016;42:1945–1955.
  • Alghunaim A, Zhang Newby B-m. Influence of tube wettability on water contact angle of powders determined by capillary rise. Colloids Surf A Physicochem Eng Asp. 2016;492:79–87.
  • Dai Y, Meng Q, Mu W, et al. Recent advances in the applications and biotechnological production of mannitol. J Funct Foods. 2017;36:404–409.
  • Chen XY, Chen C, Zhang ZJ, et al. Synthesis and capacitive performance of nitrogen doped porous carbons derived from sodium carboxymethyl starch. Powder Technol. 2013;246:201–209.
  • Kawashima Y, Takeuchi H, Hino T. Low-substituted hydroxypropylcellulose as a sustained-drug release matrix base or disintegrant depending on its particle size and loading in formulation. Pharm Res. 1993;10:351–355.
  • Pabari R, Ramtoola Z. Effect of a disintegration mechanism on wetting, water absorption, and disintegration time of orodispersible tablets. J Young Pharm. 2012;4:157–163.
  • Quodbach J, Kleinebudde P. Performance of tablet disintegrants: impact of storage conditions and relative tablet density. Pharm Dev Technol. 2014;20:762–768.
  • Kim B, La Flamme K, Peppas NA. Dynamic swelling behavior of pH-sensitive anionic hydrogels used for protein delivery. J Appl Polym Sci. 2003;89:1606–1613.
  • Harada T, Narazaki R, Nagira S, et al. Evaluation of disintegration properties of orally rapidly disintegrating tablets using a novel disintegration tester. Chem Pharm Bull. 2006;60:1240–1248.
  • Nyström CAG, Duberg M, Karehill PG. Bonding surface area and bonding mechanism - two important factors for the understanding of powder compactability. Drug Dev Industr Pharm. 1993;19:2143–2196.
  • Quodbach J, Moussavi A, Tammer R, et al. Tablet disintegration studied by high-resolution real-time magnetic resonance imaging. J Pharm Sci. 2014;103:249–255.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.