Fast dissolving electrospun polymeric films of anti-diabetic drug repaglinide: formulation and evaluation

References

• Sharma D, Singh JN, Sharma SS. Effects of 4-phenyl butyric acid on high glucose-induced alterations in dorsal root ganglion neurons. Neurosci Lett. 2016;635:83–89.
   PubMed Web of Science ®Google Scholar
• Shomali M. Diabetes treatment in 2025: can scientific advances keep pace with prevalence? Therapeut Adv Endocrinol. 2012;3(5):163–173.
   PubMedGoogle Scholar
• Sharma D, Bhattacharya P, Kalia K, et al. Diabetic nephropathy: new insights into established therapeutic paradigms and novel molecular targets. Diabetes Res Clin Pract. 2017;128:91–108.
   PubMed Web of Science ®Google Scholar
• Wysowski DK, Armstrong G, Governale L. Rapid increase in the use of oral antidiabetic drugs in the United States, 1990–2001. Diabetes Care. 2003;26(6):1852–1855.
   PubMed Web of Science ®Google Scholar
• Mandić Z, Gabelica V. Ionization, lipophilicity and solubility properties of repaglinide. J Pharm Biomed Anal. 2006;41(3):866–871.
   PubMed Web of Science ®Google Scholar
• Gadadare R, Mandpe L, Pokharkar V. Ultra rapidly dissolving repaglinide nanosized crystals prepared via bottom-up and top-down approach: influence of food on pharmacokinetics behavior. AAPS PharmSciTech. 2015;16(4):787–799.
   PubMed Web of Science ®Google Scholar
• Varshosaz J, Minayian M, Ahmadi M, et al. Enhancement of solubility and antidiabetic effects of Repaglinide using spray drying technique in STZ-induced diabetic rats. Pharm Dev Technol. 2017;22(6):754–763.
   PubMed Web of Science ®Google Scholar
• Chatap VK, Patil SD. In-vitro and in-vivo consideration of repaglinide immediate-release tablet: assessment of porous acetostarch as a promising carrier for dissolution rate enhancement. Food Sci Technol. 2016;4(4):78–88.
   Google Scholar
• Shinde UA, Modani SH, Singh KH. Design and development of repaglinide microemulsion gel for transdermal delivery. AAPS PharmSciTech. 2018;19(1):315–325.
   PubMed Web of Science ®Google Scholar
• Desai NS, Bramhane DM, Nagarsenker MS. Repaglinide–cyclodextrin complexes: preparation, characterization and in vivo evaluation of antihyperglycemic activity. J Incl Phenom Macrocycl Chem. 2011;70(1-2):217–225.
   Web of Science ®Google Scholar
• Vuddanda PR, Mathew AP, Velaga S. Electrospun nanofiber mats for ultrafast release of ondansetron. React Funct Polym. 2016;99:65–72.
   Web of Science ®Google Scholar
• Preis M, Woertz C, Kleinebudde P, et al. Oromucosal film preparations: classification and characterization methods. Expert Opin Drug Deliv. 2013;10(9):1303–1317.
   PubMed Web of Science ®Google Scholar
• Chowdhury T, de P, el-Sherbini N, et al. Management of adults with diabetes on the haemodialysis unit: summary of new guidance from the Joint British Diabetes Societies (JBDS) and the Renal Association. Br J Diabetes. 2016;16:2.
   Web of Science ®Google Scholar
• Kamble RN, Gaikwad S, Maske A, et al. Fabrication of electrospun nanofibres of BCS II drug for enhanced dissolution and permeation across skin. J Adv Res. 2016;7(3):483–489.
   PubMed Web of Science ®Google Scholar
• Liu Z-P, Zhang L-L, Yang Y-Y, et al. Preparing composite nanoparticles for immediate drug release by modifying electrohydrodynamic interfaces during electrospraying. Powder Technol. 2018;327:179–187.
   Web of Science ®Google Scholar
• Thakkar S, Misra M. Electrospun polymeric nanofibers: new horizons in drug delivery. Eur J Pharm Sci. 2017;107:148–167.
   PubMed Web of Science ®Google Scholar
• Vadlamudi MK, Dhanaraj S. Significance of excipients to enhance the bioavailability of poorly water-soluble drugs in oral solid dosage forms: a review. IOP Conf Ser Mater Sci Eng. 2017;263(2):22–23.
   Google Scholar
• Huang W, Yang Y, Zhao B, et al. Fast dissolving of ferulic acid via electrospun ternary amorphous composites produced by a coaxial process. Pharmaceutics. 2018;10(3):115.
   Web of Science ®Google Scholar
• Wang Q, Yu D-G, Zhang L-L, et al. Electrospun hypromellose-based hydrophilic composites for rapid dissolution of poorly water-soluble drug. Carbohydrate Polym. 2017;174:617–625.
   PubMed Web of Science ®Google Scholar
• Li J-J, Yang Y-Y, Yu D-G, et al. Fast dissolving drug delivery membrane based on the ultra-thin shell of electrospun core-shell nanofibers. Eur J Pharmaceut Sci. 2018;122:195–204.
   PubMed Web of Science ®Google Scholar
• Yu D-G, Li J-J, Williams GR, et al. Electrospun amorphous solid dispersions of poorly water-soluble drugs: a review. J Controlled Rel. 2018;292:91.
   PubMed Web of Science ®Google Scholar
• Brough C, Miller DA, Keen JM, et al. Use of polyvinyl alcohol as a solubility-enhancing polymer for poorly water soluble drug delivery (part 1). AAPS PharmSciTech. 2016;17(1):167–179.
   PubMedGoogle Scholar
• Brough C, Miller DA, Ellenberger D, et al. Use of polyvinyl alcohol as a solubility enhancing polymer for poorly water-soluble drug delivery (part 2). AAPS PharmSciTech. 2016;17(1):180–190.
   PubMedGoogle Scholar
• Sareen S, Mathew G, Joseph L. Improvement in solubility of poor water-soluble drugs by solid dispersion. Int J Pharma Investig. 2012;2(1):12.
   PubMedGoogle Scholar
• Khadka P, Ro J, Kim H, et al. Pharmaceutical particle technologies: an approach to improve drug solubility, dissolution and bioavailability. Asian J Pharm Sci. 2014;9(6):304–316.
   Google Scholar
• Huang M, Hou Y, Li Y, et al. High performances of dual network PVA hydrogel modified by PVP using borax as the structure-forming accelerator. Des Monomers Polym. 2017;20(1):505–513.
   PubMed Web of Science ®Google Scholar
• Anup N, Thakkar S, Misra M. Formulation of olanzapine nanosuspension based orally disintegrating tablets (ODT); comparative evaluation of lyophilization and electrospraying process as solidification techniques. Adv Powder Technol. 2018;29(8):1913–1924.
   Web of Science ®Google Scholar
• Thakkar S, Sharma D, Misra M. Comparative evaluation of electrospraying and lyophilization techniques on solid state properties of Erlotinib nanocrystals: assessment of in-vitro cytotoxicity. Eur J Pharmaceut Sci. 2018;111:257–269.
   PubMed Web of Science ®Google Scholar
• Sharma K, Sharma D, Sharma M, et al. Astaxanthin ameliorates behavioral and biochemical alterations in in-vitro and in-vivo model of neuropathic pain. Neurosci Lett. 2018;674:162–170.
   PubMed Web of Science ®Google Scholar
• Desai N, Nagarsenker M. Design and evaluation of self-nanoemulsifying pellets of repaglinide. AAPS PharmSciTech. 2013;14(3):994–1003.
   PubMed Web of Science ®Google Scholar
• Zhu Z, Yang T, Zhao Y, et al. A simple method to improve the dissolution of repaglinide and exploration of its mechanism. Asian J Pharm Sci. 2014;9(4):218–225.
   Google Scholar
• Liu J, Xiao Y, Allen C. Polymer–drug compatibility: a guide to the development of delivery systems for the anticancer agent, ellipticine. J Pharm Sci. 2004;93(1):132–143.
   PubMed Web of Science ®Google Scholar
• Zupančič Š, Sinha-Ray S, Sinha-Ray S, et al. Controlled release of ciprofloxacin from core–shell nanofibers with monolithic or blended core. Mol Pharmaceutics. 2016;13(4):1393–1404.
   PubMed Web of Science ®Google Scholar
• Yu D-G, Branford-White C, White K, et al. Dissolution improvement of electrospun nanofiber-based solid dispersions for acetaminophen. Aaps Pharmscitech. 2010;11(2):809–817.
   PubMed Web of Science ®Google Scholar
• Li X, Kanjwal MA, Lin L, et al. Electrospun polyvinyl-alcohol nanofibers as oral fast-dissolving delivery system of caffeine and riboflavin. Colloids Surf B. 2013;103:182–188.
   PubMed Web of Science ®Google Scholar
• El-Aziz AA, El-Maghraby A, Taha NA. Comparison between polyvinyl alcohol (PVA) nanofiber and polyvinyl alcohol (PVA) nanofiber/hydroxyapatite (HA) for removal of Zn2+ ions from wastewater. Arab J Chem. 2017;10(8):1052–1060.
   Web of Science ®Google Scholar
• Santibenchakul S, Chaiyasith S, Pecharapa W. Effect of PVP concentration on microstructure and physical properties of electrospun SnO2 nanofibers. Integr Ferroelectrics. 2016;175(1):130–137.
   Web of Science ®Google Scholar
• Zeng J, Yang L, Liang Q, et al. Influence of the drug compatibility with polymer solution on the release kinetics of electrospun fiber formulation. J Control Release. 2005;105(1-2):43–51.
   PubMed Web of Science ®Google Scholar
• Ghosal K, Chandra A, Praveen G, et al. Electrospinning over solvent casting: tuning of mechanical properties of membranes. Sci Rep. 2018;8(1):5058.
   PubMedGoogle Scholar
• Korbag I, Mohamed Saleh S. Studies on mechanical and biodegradability properties of PVA/lignin blend films. Int Res J Environ. 2016;73(1):18–24.
   Google Scholar
• Irfan M, Rabel S, Bukhtar Q, et al. Orally disintegrating films: a modern expansion in drug delivery system. Saudi Pharm J. 2016;24(5):537–546.
   PubMed Web of Science ®Google Scholar
• Yu T, Wu C, Chang C, et al. Effects of crystalline morphologies on the mechanical properties o. Express Polym Lett. 2012;6(4):318–328.
   Web of Science ®Google Scholar
• Shete G, Pawar YB, Thanki K, et al. Oral bioavailability and pharmacodynamic activity of hesperetin nanocrystals generated using a novel bottom-up technology. Mol Pharmaceutics. 2015;12(4):1158–1170.
   PubMed Web of Science ®Google Scholar
• Valleri M, Mura P, Maestrelli F, et al. Development and evaluation of glyburide fast dissolving tablets using solid dispersion technique. Drug Dev Ind Pharm. 2004;30(5):525–534.
   PubMed Web of Science ®Google Scholar
• Mondal D, Mollick MMR, Bhowmick B, et al. Effect of poly (vinyl pyrrolidone) on the morphology and physical properties of poly (vinyl alcohol)/sodium montmorillonite nanocomposite films. Pro Nat Sci Mater. 2013;23(6):579–587.
   Web of Science ®Google Scholar