Ibuprofen-loaded centrifugally spun microfibers for quick relief of inflammation in rats

References

• Rainsford K. Ibuprofen: pharmacology, efficacy and safety. Inflammopharmacology. 2009;17(6):275–342.
   PubMedGoogle Scholar
• Irvine J, Afrose A, Islam N. Formulation and delivery strategies of ibuprofen: challenges and opportunities. Drug Dev Ind Pharm. 2018;44(2):173–183.
   PubMed Web of Science ®Google Scholar
• Gryczke A, Schminke S, Maniruzzaman M, et al. Development and evaluation of orally disintegrating tablets (ODTs) containing ibuprofen granules prepared by hot melt extrusion. Colloids Surf B Biointerfaces. 2011;86(2):275–284.
   PubMed Web of Science ®Google Scholar
• Klueglich M, Ring A, Scheuerer S, et al. Ibuprofen extrudate, a novel, rapidly dissolving ibuprofen formulation: relative bioavailability compared to ibuprofen lysinate and regular ibuprofen, and food effect on all formulations. J Clin Pharmacol. 2005;45(9):1055–1061.
   PubMed Web of Science ®Google Scholar
• Szabó P, Kállai-Szabó B, Sebe I, et al. Preformulation study of fiber formation and formulation of drug-loaded microfiber based orodispersible tablets for in vitro dissolution enhancement. Int J Pharm. 2014;477(1–2):643–649.
   PubMed Web of Science ®Google Scholar
• Casian T, Borbás E, Ilyés K, et al. Electrospun amorphous solid dispersions of meloxicam: influence of polymer type and downstream processing to orodispersible dosage forms. Int J Pharm. 2019;569:118593.
   PubMed Web of Science ®Google Scholar
• Hussain A, Mahmood F, Arshad MS, et al. Personalised 3D printed fast-dissolving tablets for managing hypertensive crisis: in-vitro/in-vivo studies. Polymers. 2020;12(12):3057.
   Web of Science ®Google Scholar
• Nasir S, Hussain A, Abbas N, et al. Improved bioavailability of oxcarbazepine, a BCS class II drug by centrifugal melt spinning: in-vitro and in-vivo implications. Int J Pharm. 2021;604:120775.
   PubMed Web of Science ®Google Scholar
• Mirzaeei S, Mohammadi G, Fattahi N, et al. Formulation and physicochemical characterization of cyclosporine microfiber by electrospinning. Adv Pharm Bull. 2019;9(2):249–254.
   PubMed Web of Science ®Google Scholar
• Nagy ZK, Balogh A, Drávavölgyi G, et al. Solvent-free melt electrospinning for preparation of fast dissolving drug delivery system and comparison with solvent-based electrospun and melt extruded systems. J Pharm Sci. 2013;102(2):508–517.
   PubMed Web of Science ®Google Scholar
• Hu X, Liu S, Zhou G, et al. Electrospinning of polymeric nanofibers for drug delivery applications. J Control Release. 2014;185:12–21.
   PubMed Web of Science ®Google Scholar
• Salvagnini C, Roback A, Momtaz M, et al. Surface functionalization of a poly (butylene terephthalate) (PBT) melt-blown filtration membrane by wet chemistry and photo-grafting. J Biomater Sci Polym Ed. 2007;18(12):1491–1516.
   PubMed Web of Science ®Google Scholar
• Dasdemir M, Maze B, Anantharamaiah N, et al. Influence of polymer type, composition, and interface on the structural and mechanical properties of core/sheath type bicomponent nonwoven fibers. J Mater Sci. 2012;47(16):5955–5969.
   Web of Science ®Google Scholar
• Marano S, Barker SA, Raimi-Abraham BT, et al. Development of micro-fibrous solid dispersions of poorly water-soluble drugs in sucrose using temperature-controlled centrifugal spinning. Eur J Pharm Biopharm. 2016;103:84–94.
   PubMed Web of Science ®Google Scholar
• Ma PX, Zhang R. Synthetic nano‐scale fibrous extracellular matrix. J Biomed Mater Res. 1999;46(1):60–72.
   PubMed Web of Science ®Google Scholar
• Ikegame M, Tajima K, Aida T. Template synthesis of polypyrrole nanofibers insulated within one-dimensional silicate channels: hexagonal versus lamellar for recombination of polarons into bipolarons . Angew Chem Int Ed Engl. 2003;42(19):2154–2157.
   PubMed Web of Science ®Google Scholar
• Chen J, Pan H, Yang Y, et al. Self-assembled liposome from multi-layered fibrous mucoadhesive membrane for buccal delivery of drugs having high first-pass metabolism. Int J Pharm. 2018;547(1–2):303–314.
   PubMed Web of Science ®Google Scholar
• Padron S, Patlan R, Gutierrez J, et al. Production and characterization of hybrid BEH‐PPV/PEO conjugated polymer nanofibers by forcespinning™. J Appl Polym Sci. 2012;125(5):3610–3616.
   Web of Science ®Google Scholar
• Marano S, Barker SA, Raimi-Abraham BT, et al. Microfibrous solid dispersions of poorly water-soluble drugs produced via centrifugal spinning: unexpected dissolution behavior on recrystallization. Mol Pharm. 2017;14(5):1666–1680.
   PubMed Web of Science ®Google Scholar
• Morrow EA, Terban MW, Thomas LC, et al. Effect of amorphization method on the physicochemical properties of amorphous sucrose. J Food Eng. 2019;243:125–141.
   Web of Science ®Google Scholar
• Labuza TP, Labuza PS. Influence of temperature and relative humidity on the physical states of cotton candy. J Food Process Preserv. 2004;28(4):274–287.
   Web of Science ®Google Scholar
• Ouiazzane S, Messnaoui B, Abderafi S, et al. Modeling of sucrose crystallization kinetics: the influence of glucose and fructose. J Cryst Growth. 2008;310(15):3498–3503.
   Web of Science ®Google Scholar
• Hussain A, Smith G, Khan KA, et al. Solubility and dissolution rate enhancement of ibuprofen by co-milling with polymeric excipients. Eur J Pharm Sci. 2018;123:395–403.
   PubMed Web of Science ®Google Scholar
• Kearney AS, Gabriel DL, Mehta SC, et al. Effect of polyvinylpyrrolidone on the crystallinity and dissolution rate of solid dispersions of the antiinflammatory CI-987. Int J Pharm. 1994;104(2):169–174.
   Web of Science ®Google Scholar
• Teng C, Li H, Liu J, et al. Effect of high molecular weight PPTA on liquid crystalline phase and spinning process of aramid fibers. Polymers. 2020;12(5):1206.
   Web of Science ®Google Scholar
• Chavan H, Chhabra G, Gujarathi N, et al. Comparative study of in-process and finished products quality control test for tablet and capsules according to pharmacopoeias. Asian J Pharm Res Dev. 2018;6(3):60–68.
   Google Scholar
• Young H-Y, Luo Y-L, Cheng H-Y, et al. Analgesic and anti-inflammatory activities of [6]-gingerol. J Ethnopharmacol. 2005;96(1–2):207–210.
   PubMed Web of Science ®Google Scholar
• Muzaffar K, Nayik GA, Kumar P. Stickiness problem associated with spray drying of sugar and acid rich foods: a mini review. J Nutr Food Sci. 2015;s12(S12):1.
   Google Scholar
• Samprasit W, Akkaramongkolporn P, Ngawhirunpat T, et al. Fast releasing oral electrospun PVP/CD nanofiber mats of taste-masked meloxicam. Int J Pharm. 2015;487(1–2):213–222.
   PubMed Web of Science ®Google Scholar
• Yang M, Xie S, Li Q, et al. Effects of polyvinylpyrrolidone both as a binder and pore-former on the release of sparingly water-soluble topiramate from ethylcellulose coated pellets. Int J Pharm. 2014;465(1–2):187–196.
   PubMed Web of Science ®Google Scholar
• Szabó P, Sebe I, Stiedl B, et al. Tracking of crystalline-amorphous transition of carvedilol in rotary spun microfibers and their formulation to orodispersible tablets for in vitro dissolution enhancement. J Pharm Biomed Anal. 2015;115:359–367.
   PubMed Web of Science ®Google Scholar
• Poller B, Strachan C, Broadbent R, et al. A minitablet formulation made from electrospun nanofibers. Eur J Pharm Biopharm. 2017;114:213–220.
   PubMed Web of Science ®Google Scholar
• Bai Y, Wang D, Zhang Z, et al. Testing of fast dissolution of ibuprofen from its electrospun hydrophilic polymer nanocomposites. Polym Test. 2021;93:106872.
   Web of Science ®Google Scholar
• Kazarian S, Martirosyan G. Spectroscopy of polymer/drug formulations processed with supercritical fluids: in situ ATR–IR and Raman study of impregnation of ibuprofen into PVP. Int J Pharm. 2002;232(1–2):81–90.
   PubMed Web of Science ®Google Scholar
• Einfal T, Planinšek O, Hrovat K. Methods of amorphization and investigation of the amorphous state. Acta Pharm. 2013;63(3):305–334.
   PubMed Web of Science ®Google Scholar
• Lee SY, Yu G, Kim IW. Effects of polymeric additives on the crystallization and release behavior of amorphous ibuprofen. J Nanomater. 2013;2013:1–7.
   Web of Science ®Google Scholar
• Smith G, Hussain A, Bukhari NI, et al. Correlation between molecular dynamics and physical stability of two milled anhydrous sugars: lactose and sucrose. Int J Pharm. 2018;551(1–2):184–194.
   PubMed Web of Science ®Google Scholar