Publication Cover
Drying Technology
An International Journal
Volume 35, 2017 - Issue 12
318
Views
17
CrossRef citations to date
0
Altmetric
Articles

Formulation and evaluation of solid self-microemulsifying drug delivery system of chlorthalidone by spray drying technology

, ORCID Icon, &

References

  • Swarbrick, J. Encyclopedia of Pharmaceutical Technology, 3rd ed.; Informa Healthcare: New York, 2007, 1732–1802.
  • Kalepu, S.; Manthina, M.; Padavala, V. Oral lipid-based drug delivery systems – an overview. Acta Pharmaceutica Sinica B 2003, 3(6), 361–372.
  • Bajaj, A.; Rao, M.; Khole, I.; Munjapara. G. Self-nanoemulsifying drug delivery system of cefpodoxime proxetil containing tocopherol polyethylene glycol succinate. Drug Development and Industrial Pharmacy 2013, 39(5), 635–645.
  • Government of India, Indian Pharmacopoeia Commision, Ministry of Health and Family Welfare. Indian Pharmacopoeia, Vols.1 and 3; Controller of Publications, Ghaziabad, 2010, 1076–1077.
  • Florey, K. Analytical Profile of Drug Substances, Vol.14, 1st ed.; Academic Press, Elsevier: London, 2005, 1–33.
  • Krishnamoorthy, B.; Raghavan, C.; Selvan, N.; Rahman, S. Self-emulsifying drug delivery system: Optimization and its prototype for various compositions of oils, surfactants and co-surfactants. Journal of Pharmacy Research 2013, 6(5), 510–514.
  • Pouton, C. Lipid formulations for oral administration of drugs: Non-emulsifying, self-emulsifying and self-microemulsifying drug delivery systems. European Journal of Pharmaceutical Sciences 2000, 11(2), 93–98.
  • Kohli, K.; Chopra, S.; Dhar, D.; Arora, S.; Khar, R. Self-emulsifying drug delivery systems: An approach to enhance oral bioavailability. Drug Discovery Today 2010, 15(21–22), 958–965.
  • Gursoy, N.G.; Benita, S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomedicine & Pharmacotherapy 2004, 58, 173–182.
  • Kawabata, Y.; Wada, K.; Nakatani, M.; Yamada, S.; Onoue, S. Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: Basic approaches and practical applications. International Journal of Pharmaceutics 2011, 420(1), 1–10.
  • Mette, G.; Mullertz, A.; Nielsen, J.; Pedersen G. Bioavailability of seocalcitol II: Development and characterization of self-microemulsifying drug delivery systems (SMEDDS) for oral administration containing medium and long chain triglycerides. European Journal of Pharmaceutical Sciences 2006, 8, 233–242.
  • Parakh, D.; Patil, M.; Shinde, G. Self micro-emulsifying drug delivery system: Approach to improve solubility and permeability. International Journal of Institutional Pharmacy and Life Sciences 2015, 5(4), 21–37.
  • Müllertz, A.; Ogbonna, A.; Ren, S.; Rades, T. New perspectives on lipid and surfactant based drug delivery systems for oral delivery of poorly soluble drugs. Journal of Pharmacy and Pharmacology 2010, 62(11), 1622–1636.
  • Mu, H.; Holm, R.; Müllertz, A. Lipid-based formulations for oral administration of poorly water-soluble drugs. International Journal of Pharmaceutics 2013, 453(1), 215–224.
  • Tang, J.; Sun, J.; He, Z. Self-emulsifying drug delivery systems: Strategy for improving oral delivery of poorly soluble drugs. Current Drug Therapeutics 2007, 2, 85–93.
  • Shen, H.; Zhong, M. Preparation and evaluation of self-microemulsifying drug delivery systems (SMEDDS) containing atorvastatin. Journal of Pharmacy and Pharmacology 2006, 58(9), 1183–1191.
  • Patel, D.; Sawant, K. Self microemulsifying drug delivery system: Formulation, development, and biopharmaceutical evaluation of lipophilic drugs. Current Drug Delivery 2009, 6, 419–424.
  • Rahman, M.; Harwansh, R.; Mirza, M.; Hussain, S.; Hussain A. Oral lipid based drug delivery system (LBDDS) formulation, characterization and application a review. Current Drug Delivery 2011, 8, 330–345.
  • Dixit, A.; Rajput, S.; Patel, S. Preparation and bioavailability assessment of SMEDDS containing valsartan. AAPS PharmSciTech 2010, 11(1), 314–321.
  • Komura, T.; Gurley, B.; Khan, M.; Reddy, I. Self-emulsifying drug delivery systems (SEDDS) of coenzyme Q 10: Formulation development and bioavailability assessment. International Journal of Pharmaceutics 2001, 212, 233–246.
  • Birchal, V.S.; Passos, M.L.; Wildhagen, G.R.S.; Mujumdar, A.S. Effect of spray dryer operating variables on the whole milk powder quality. Drying Technology 2005, 23, 611–636.
  • Huang, L.; Kumar, K.; Mujumdar, A.S. A parametric study of the gas flow patterns and drying performance of co-current spray dryer: Results of a computational fluid dynamics study. Drying Technology 2003, 22(6), 957–978.
  • Huang, L.; Kumar, K.; Mujumdar, A.S. Simulation of a spray dryer fitted with a rotary disk atomizer using a three-dimensional computational fluid dynamic model. Drying Technology 2004, 22(6), 1489–1515.
  • Liu, C.; Desai, K.G.H.; Tang, X.; Chen, X. Drug release kinetics of spray dried chitosan microspheres. Drying Technology 2006, 24, 769–776.
  • Mujumdar, A.S. Research and developments in drying: Recent trends and future prospectus. Drying Technology 2004, 22(1&2), 1–26.
  • Goula, A.M.; Adamopoulos, K.G. Spray drying performance of a laboratory spray dryer for tomato powder preparation spray drying performance of laboratory. Drying Technology 2007, 21(7), 37–41.
  • Re, M.I. Formulating drug delivery systems by spray drying. Drying Technology 2006, 24, 433–446.
  • Jangam, S.V.; Thorat, B.N. Optimization of spray drying of ginger extract optimization of spray drying of ginger extract. Drying Technology 2010, 28, 1426–1434.
  • Kawabata, Y.; Wada, K.; Nakatani, M.; Yamada, S.; Onoue, S. Formulation design for poorly water soluble drugs based on biopharmaceutics classification system: Basic approaches and practical applications. International Journal of Pharmaceutics 2011, 420, 1–10.
  • Dharankar, S.; Parakh, D.; Patil, M.; Kshirsagar S. Spray-dried solid self-emulsifying delivery system of ketoprofen: Development and its characterization. Drying Technology 2015, 33, 2002–2011.
  • Reiss, H. Entropy induced dispersion of bulk liquids. Journal of Colloid and Interface Science 1975, 53, 61–70.
  • Re, M. Microencapsulation by spray drying. Drying Technology 1998, 16(6), 1195–1236.
  • Nath, S.; Satpathy, G.A. Systematic approach for investigation of spray drying processes. Drying Technology 1998, 16(6), 1173–1193.
  • Maria, I. Formulating drug delivery systems by spray drying. Drying Technology 2006, 24, 433–446.
  • Mujumdar, A. Aspects of computer simulation of liquid fuelled combustors. Drying Technology 2010, 3, 311–342.
  • Saifee, M.; Zarekar, S.; Rao, V.U.; Zaheer, Z.; Soni, R.; Burande, S. Formulation and in vitro evaluation of solid- self- emulsifying drug delivery system (SEDDS) of glibenclamide. American Journal of Advanced Drug Delivery 2013, 1(3), 323–340.
  • Elnaggar, Y.; El-Massik, M.; Abdallah. O. Self-nanoemulsifying drug delivery systems of tamoxifen citrate: Design and optimization. International Journal of Pharmaceutics 2009, 380(1–2), 133–141.
  • Villar, A.; Naverosb, B.; Campmany, A.; Naveros, B.; Trenchs, M.; Rocabert, C.; Bellowa, L. Design and optimization of self-nanoemulsifying drug delivery systems (SNDDS) for enhanced dissolution of gemfibrozil. International Journal of Pharmaceutics 2012, 431(1–2), 161–175.
  • Hu, X.; Chen, L.; Chen, D.; Zhang, J.; Liu, Z.; Wub, W.; Song, H. Sirolimus solid self-microemulsifying pellets: Formulation development, characterization and bioavailability evaluation. International Journal of Pharmaceutics 2012, 438(1–2), 123–133.
  • Balakrishnan, P.; Lee, B.; Oha, D.; Kim, J.; Lee, Y.; Kim, D.; Jee, J.; Lee, Y.; Woo, J.; Yonga, C.; Choiaet, H. Enhanced oral bioavailability of coenzyme Q 10 by self-emulsifying drug delivery systems. International Journal of Pharmaceutics 2009, 374, 66–72.
  • Basalious, E.; Shawky, N.; Badr-Eldin, S. SNEDDS containing bioenhancers for improvement of dissolution and oral absorption of lacidipine. I: Development and optimization. International Journal of Pharmaceutics 2010, 391(1–2), 203–211.
  • Tang, B.; Cheng G.; Gu, J.; Xu, C. Development of solid self-emulsifying drug delivery systems: Preparation techniques and dosage forms. Drug Discovery Today 2007, 13(13–14), 606–612.
  • Oh, D.; Kang, J.; Kim, D.; Lee, B.; Kim, J.; Yong, C.; Choi, H. Comparison of solid self-microemulsifying drug delivery system (solid SMEDDS) prepared with hydrophilic and hydrophobic solid carrier. International Journal of Pharmaceutics 2011, 420(2), 412–418.
  • Milović, M.; Djuriš, J.; Djekić, L.; Vasiljević, D.; Ibrić, S. Characterization and evaluation of solid self-microemulsifying drug delivery systems with porous carriers as systems for improved carbamazepine release. International Journal of Pharmaceutics 2012, 436(1–2), 58–65.
  • Wang, Z.; Sun, J.; Wang, Y.; Liu, X.; Liu, Y.; Fu, Q.; Meng, P.; He, Z. Solid self-emulsifying nitrendipine pellets: Preparation and in-vitro/in-vivo evaluation. International Journal of Pharmaceutics 2010, 383, 1–6.
  • Abdelwahed, W.; Degobert, G.; Stainmesse, S.; Fessi. H. Freeze-drying of nanoparticles: Formulation, process and storage considerations. Advanced Drug Delivery Review 2006, 58, 1688–1713.
  • Katteboina, S.; Chandrashekhar, P.; Balaji, S. Approaches for the development of solid self-emulsifying drug delivery systems and dosage forms. Asian Journal of Pharmaceutical Sciences 2009, 4(4), 240–253.
  • Qureshi, M.; Chitneni, M.; Wong, G. Enhancement of solubility and therapeutic potential of poorly soluble lovastatin by SMEDDS formulation adsorbed on directly compressed spray dried magnesium aluminometasilicate liquid loadable tablets: A study in diet induced hyperlipidemic rabbits. Asian Journal of Pharmaceutical Sciences 2015, 10(1), 40–56.
  • Piao, Z.; Choe, J.; Teak, K.; Rhee, Y.; Lee. B. Formulation and in-vivo human bioavailability of dissolving tablets containing a self-nanoemulsifying itraconazole solid dispersion without precipitation in simulated gastrointestinal fluid. European Journal of Pharmaceutical Sciences 2014, 51, 67–74.
  • Abdalla, A.; Klein, S.; Mäder, K. A new self-emulsifying drug delivery system (SEDDS) for poorly soluble drugs: Characterization, dissolution, in-vitro digestion and incorporation into solid pellets. European Journal of Pharmaceutical Sciences 2008, 35(5), 457–464.
  • Hamoudi, M.; Fattal, E.; Gueutin, C.; Nicolas, V.; Bochot, A. Beads made of cyclodextrin and oil for the oral delivery of lipophilic drugs: In vitro studies in simulated gastro-intestinal fluids. International Journal of Pharmaceutics 2011, 416(2), 507–514.
  • Patil, P.; Paradkar. A. Porous polystyrene beads as carriers for self-emulsifying system containing loratadine. AAPS PharmSciTech 2006, 7(1), 1–7.
  • Faisal, W.; O’Hora, T.; O’Driscoll, C.; Griffin, B. A novel lipid-based solid dispersion for enhancing oral bioavailability of lycopene in-vivo evaluation using a pig model. International Journal of Pharmaceutics 2013, 453(2), 307–314.
  • Tran, T.; Tran, P.; Lee, B. Dissolution-modulating mechanism of alkalizers and polymers in a nanoemulsifying solid dispersion containing ionizable and poorly water-soluble drug. European Journal of Pharmaceutics and Biopharmaceutics 2009, 72(1), 83–90.
  • Park, M.; Balakrishnan, P.; Yang, S. 2013. Polymeric nanocapsules with SEDDS oil-core for the controlled and enhanced oral absorption of cyclosporine. International Journal of Pharmaceutics 2013, 441(1–2), 757–764.
  • Qi, X.; Wang, L.; Zhu, L.; Hu, Z.; Zhang, J. Self-double-emulsifying drug delivery system (SEDDS): A new way for oral delivery of drugs with high solubility and low permeability. International Journal of Pharmaceutics 2011, 409(1–2), 245–251.
  • Banker, G.S.; Rhodes, C.T. Modern Pharmaceutics, 4th ed.; Informa Healthcare: New York, 2009, 112–143.
  • Parakh, D.; Patil, M.; Dashputre, N.; Kshirsagar, S. Development of self micro-emulsifying drug delivery system of mebendazole by spray drying technology: characterization, in-vitro and in-vivo evaluation. Drying Technology 2015, 34(9), 1023–1042.
  • Ahmad, J.; Kohli, K.; Mir, S.; Amin, S. Formulation of self-nanoemulsifying drug delivery system for telmisartan with improved dissolution and oral bioavailability formulation of self-nanoemulsifying drug delivery system for telmisartan with improved dissolution and oral bioavailability. Journal of Dispersion Science and Technology 2011, 32, 958–968.
  • Seo, Y.; Kim, D.; Ramasamy, T.; Kim, J.; Marasini, N.; Oh, Y.; Kim, D.; Kim, J.; Yong, C. Development of docetaxel-loaded solid self-nanoemulsifying drug delivery system (SNEDDS) for enhanced chemotherapeutic effect. International Journal of Pharmaceutics 2013, 452(1–2), 412–420.
  • Patel, K.; Patel, B. Enhancement of oral bioavailability of valsartan by using solid self-emulsifying drug delivery system. International Journal of Universal Pharmacy and BioSciences 2014, 3(3), 141–156.
  • Baboota, S.; Shakeel, F.; Ahuja, A.; Ali, J.; Sheikh, S. Design development and evaluation of novel nanoemulsion formulations for transdermal potential of celecoxib. Acta Pharma 2007, 57, 315–332.
  • Chaudhari, S.; Kolhe, S.; Ratnaparakhi, M.; Ranpise, A. Study of oral lipid based formulation through design and evaluation of solid self emulsified drug delivery system. International Journal of Pharmaceutical and Phytopharmacological Research 2013, 3(2), 97–103.
  • Singh, A.; Chaurasiya, A.; Awasthi, A.; Mishra, G.; Asati, D.; Khar, K.; Mukherjee, R. Oral bioavailability enhancement of exemestane from self-microemulsifying drug delivery system (SMEDDS). AAPS PharmSciTech 2009, 10(3), 906–916.
  • Parakh, D.; Patil, M. Comparison of in-vitro dissolution profiles of marketed dicyclomine hydrochloride tablets. An International Journal of Advances in Pharmaceutical Sciences 2014, 5(3), 2109–2119.
  • Agarwal, V.; Alayoubi, A.; Siddiqui, A.; Sami Nazzal, S. Powdered self-emulsified lipid formulations of meloxicam as solid dosage forms for oral administration. Drug Development and Industrial Pharmacy 2012, 1, 1–9.
  • Wu, H.; Long, X.; Yuan, F.; Chen, L.; Pan, S. Combined use of phospholipid complexes and self-emulsifying microemulsions for improving the oral absorption of a BCS class IV compound, baicalin. Acta Pharmaceutica Sinica B 2014, 4(3), 217–226.
  • Akhtar, N.; Talegaonkar, S.; Khar, R.; Jaggi, M. A validated stability-indicating LC method for estimation of etoposide in bulk and optimized self-nano emulsifying formulation: Kinetics and stability effects. Saudi Pharmaceutical Journal 2013, 21, 103–111.
  • Yin, Y.; Cui, F.; Mua, C.; Choi, M.; Kim, J.; Chung, S.; Shim, C.; Kim, D. Docetaxel microemulsion for enhanced oral bioavailability: Preparation and in-vitro and in-vivo evaluation. Journal of Controlled Release 2009, 140(2), 86–94.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.