Preparation and Evaluation of Fast Dissolving Ibuprofen-Polyethylene Glycol 6000 Solid Dispersions

REFERENCES

• Adeyeye C. M., Price J. C. Development and evaluation of sustained-release ibuprofen-wax microspheres. II. In vitro dissolution studies. Pharm. Res. 1994; 11: 575–579
   PubMed Web of Science ®Google Scholar
• Anastasiadou C., Henry S., Legendre B., Souleau C., Duchene D. Solid dispersions: comparison of prepared melts and coprecipitates of diazepam and polyoxyethylene glycol 4000. Drug Dev. Ind. Pharm. 1983; 9: 103–115
   Web of Science ®Google Scholar
• Bowden S. T. The Phase Rule and Phase Reactions:Theoretical and Practical. MacMillan Press, London 1938
   Google Scholar
• Canaparo R., Muntoni E., Zara G. P., Della P. C., Berno E., Costa M., Eandi M. Determination of ibuprofen in human plasma by high-performance liquid chromatography: validation and application in pharmacokinetic study. Biomed. Chromatogr. 2000; 14: 219–226
   PubMed Web of Science ®Google Scholar
• Carstensen J. T. Melting point diagrams and eutectics. Advanced Pharmaceutical Solids. Marcel Dekker, New York 2001; 170–189
   Google Scholar
• Corrigan O. I. Mechanisms of dissolution of fast release solid dispersions. Drug Dev. Ind. Pharm. 1985; 11: 697–724
   Web of Science ®Google Scholar
• Craig D. Q. M. The mechanisms of drug release from solid dispersions in water-soluble polymers. Int. J. Pharm. 2002; 231: 131–144
   PubMed Web of Science ®Google Scholar
• Craig D. Q. M. Polyethylene glycols and drug release. Drug Dev. Ind. Pharm. 1990; 16: 2501–2506
   Web of Science ®Google Scholar
• Ford J. L., Rubeinstein M. J. H. Phase equlibria and dissolution rates of indomethacin-polyethylene glycol 6000 solid dispersions. Pharm. Acta Helv. 1978; 53: 93–98
   Google Scholar
• Geisslinger G., Dietzel K., Bezler H., Nuernberg B., Brune K. Therapeutically relevant differences in the pharmacokinetical and pharmaceutical behavior of ibuprofen lysinate as compared to ibuprofen acid. Int. J. Clin. Pharmacol. Ther. Tox. 1989; 27: 324–328
   PubMed Web of Science ®Google Scholar
• Ghorab M. K., Adeyeye M. C. Enhancement of ibuprofen, dissolution via wet granulation with beta-cyclodextrin. Pharm. Dev. Tech. 2001; 6: 305–314
   PubMed Web of Science ®Google Scholar
• Lacoulonche F., Chauvet A., Masse J., Egea M. A., Garcia M. L. An investigation of FB interactions with poly(ethylene glycol) 6000, poly(ethylene glycol) 4000 and poly-epsilon-caprolactone by thermoanalytical and spectroscopic methods and modeling. J. Pharm. Sci. 1998; 87: 543–551
   PubMed Web of Science ®Google Scholar
• Lacoulonche F., Manderioli A., Bramanti G., Ceccarelli L. Properties of solid dispersions of naproxen in various polyethylene glycols. Drug Dev. Ind. Pharm. 1996; 22: 909–916
   Web of Science ®Google Scholar
• Laska E. M., Sunshine A., Marrero I., Olson N., Siegel C., McCormick N. The correlation between blood levels of ibuprofen and clinical analgesic response. Clin. Pharmacol. Ther. 1986; 40: 1–7
   PubMed Web of Science ®Google Scholar
• Law D., Wang W., Schmitt E. A., Qiu Y., Steven L. K., Fort J. J. Properties of rapidly dissolving eutectic mixtures of poly(ethylene glycol) and fenofibrate: the eutectic microstructure. J. Pharm. Sci. 2003; 92: 505–515
   PubMed Web of Science ®Google Scholar
• Law D., Wang W., Schmitt E. A., Michelle A. L. Prediction of poly (ethylene) glycol-drug eutectic compositions using an index based on the van't Hoff equation. Pharm. Res. 2002; 19: 315–321
   PubMed Web of Science ®Google Scholar
• Law D., Krill S. L., Schmitt E. A., Fort J. J., Qiu Y., Wang W., Porter W. R. Physicochemical considerations in the preparation of amorphous ritonavir/PEG 8000 solid dispersions. J. Pharm. Sci. 2001; 90: 1015–1025
   PubMed Web of Science ®Google Scholar
• Moter G. V., Augustijns P., Blaton N., Kinget R. Physicochemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30. Int. J. Pharm. 1998; 164: 67–80
   Web of Science ®Google Scholar
• Mura P., Manderioli A., Bramanti G., Ceccarelli L. Properties of solid dispersions of naproxen in various polyethylene glycols. Drug Dev. Ind. Pharm. 1996; 22: 909–916
   Web of Science ®Google Scholar
• Murtha J. L., Ando H. Y. Synthesis of the cholesteryl ester prodrugs cholesteryl ibuprofen and cholesteryl flufenamate and their formulation into phospholipid microemulsions. J. Pharm. Sci. 1994; 83: 1222–1228
   PubMed Web of Science ®Google Scholar
• Passerini N., Gonzalez-Rodriguez M. L., Cavallari C., Rodriguez L., Albertini B. Preparation and characterisation of ibuprofen-poloxamer 188 granules obtained by melt granulation. Eur. J. Pharm. Sci. 2002; 15: 71–78
   PubMed Web of Science ®Google Scholar
• Podolinsky V. V., Taran Y. Influence of adsorption on structure formation in eutectic systems. J. Cryst. Growth. 1981; 52: 82–87
   Web of Science ®Google Scholar
• Potthast H., Dressman J. B., Junginger H. E., Midha K. K., Oeser H., Shah V. P., Vogelpoel H., Barends D. M. Biowaiver monographs for immediate release solid oral dosage forms: ibuprofen. J. Pharm. Sci. 2005; 94: 2121–2131
   PubMed Web of Science ®Google Scholar
• Rabasco A. M., Ginés J. M., Fernández-Arévalo M., Holgado M. A. Dissolution rate of diazepam from polyethylene glycol 6000 solid dispersions. Int. J. Pharm. 1991; 67: 201–205
   Web of Science ®Google Scholar
• Seo A., Holm P., Kristensen H. G., Schæfer T. The preparation of agglomerates containing solid dispersions of diazepam by melt agglomeration in a high shear mixer. Int. J. Pharm. 2003; 259: 161–171
   PubMed Web of Science ®Google Scholar
• Serajuddin A. T. M. Solid dispersion of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs. J. Pharm. Sci. 1999; 88: 1058–1066
   PubMed Web of Science ®Google Scholar
• Sudha R. V., Zeren W., Stefanie H., Steven L. K. Factors affecting the formation of eutectic solid dispersions and their dissolution behavior. J. Pharm. Sci. 2007; 96: 294–304
   PubMed Web of Science ®Google Scholar
• Vasil'ev M. E. Classification of the phase diagrams of binary metallic systems according to atomic interaction forces. Russ. Phys. Chem. 1964; 38: 473–476
   Google Scholar
• Verheyen S., Blaton N., Kinget R., Mooter G. V. Mechanism of increased dissolution of diazepam and temazepam from polyethylene glycol 6000 solid dispersions. Int. J. Pharm. 2002; 249: 45–58
   PubMed Web of Science ®Google Scholar
• Vilhelmsen T., Eliasen H., Schæfer T. Effect of a melt agglomeration process on agglomerates containing solid dispersions. Int. J. Pharm. 2005; 303: 132–142
   PubMed Web of Science ®Google Scholar
• Zerrouk N., Chemtob C., Arnaud P., Toscani S., Dugue J. In vitro and in vivo evaluation of carbamazepine-PEG 6000 solid dispersions. Int. J. Pharm. 2002; 225: 49–62
   Web of Science ®Google Scholar