146
Views
4
CrossRef citations to date
0
Altmetric
Research Articles

The effect of some acrylic polymers on dissolution of celecoxib solid dispersion formulations

ORCID Icon, ORCID Icon &
Pages 788-796 | Received 16 Mar 2021, Accepted 17 Jun 2021, Published online: 15 Jul 2021

References

  • Alonzo DE, Zhang GGZ, Zhou D, Gao Y, Taylor LS. 2010. Understanding the behavior of amorphous pharmaceutical systems during dissolution. Pharm Res. 27(4):608–618.
  • Andrews GP, Abu-Diak O, Kusmanto F, Hornsby P, Hui Z, Jones DS. 2010. Physicochemical characterization and drug-release properties of celecoxib hot-melt extruded glass solutions. J Pharm Pharmacol. 62(11):1580–1590.
  • Babu NJ, Nangia A. 2011. Solubility advantage of amorphous drugs and pharmaceutical cocrystals. Cryst Growth Des. 11(7):2662–2679.
  • Baird JA, Taylor LS. 2012. Evaluation of amorphous solid dispersion properties using thermal analysis techniques. Adv Drug Deliv Rev. 64(5):396–421.
  • Brouwers J, Brewster ME, Augustijns P. 2009. Supersaturating drug delivery systems: the answer to solubility-limited oral bioavailability? J Pharm Sci. 98(8):2549–2572.
  • Chawla G, Gupta P, Thilagavathi R, Chakraborti AK, Bansal AK. 2003. Characterization of solid-state forms of celecoxib. Eur J Pharm Sci. 20(3):305–317.
  • Cilurzo F, Minghetti P, Selmin F, Casiraghi A, Montanari L. 2003. Polymethacrylate salts as new low-swellable mucoadhesive materials. J Controll Release. 88(1):43–53.
  • Dahan A, Miller JM. 2012. The solubility-permeability interplay and its implications in formulation design and development for poorly soluble drugs. AAPS J. 14(2):244–251.
  • Fouad EA, El-Badry M, Mahrous GM, Alanazi FK, Neau SH, Alsarra IA. 2011. The use of spray-drying to enhance celecoxib solubility. Drug Dev Ind Pharm. 37(12):1463–1472.
  • Frank DS, Matzger AJ. 2019. Effect of polymer hydrophobicity on the stability of amorphous solid dispersions and supersaturated solutions of a hydrophobic pharmaceutical. Mol Pharm. 16(2):682–688.
  • Gao P, Guyton ME, Huang T, Bauer JM, Stefanski KJ, Lu Q. 2004. Enhanced oral bioavailability of a poorly water soluble drug PNU-91325 by supersaturatable formulations. Drug Dev Ind Pharm. 30(2):221–229.
  • Gupta P, Kakumanu VK, Bansal AK. 2004. Stability and solubility of celecoxib-PVP amorphous dispersions: a molecular perspective. Pharm Res. 21(10):1762–1769.
  • Gupta P, Thilagavathi R, Chakraborti AK, Bansal AK. 2005. Role of molecular interaction in stability of celecoxib-PVP amorphous systems. Mol Pharm. 2(5):384–391.
  • Homayouni A, Sadeghi F, Nokhodchi A, Varshosaz J, Garekani HA. 2014. Preparation and characterization of celecoxib solid dispersions; comparison of poloxamer-188 and PVP-K30 as carriers. Iran J Basic Med Sci. 17(5):322–331.
  • Homayouni A, Sadeghi F, Nokhodchi A, Varshosaz J, Garekani HA. 2015. Preparation and characterization of celecoxib dispersions in Soluplus®: comparison of spray drying and conventional methods. Iran J Pharm Res. 14(1):35–50.
  • Homayouni A, Sadeghi F, Varshosaz J, Garekani HA, Nokhodchi A. 2014. Comparing various techniques to produce micro/nanoparticles for enhancing the dissolution of celecoxib containing PVP. Eur J Pharm Biopharm. 88(1):261–274.
  • Hsieh YL, Box K, Taylor LS. 2014. Assessing the impact of polymers on the pH-induced precipitation behavior of poorly water soluble compounds using synchrotron wide angle X-ray scattering . J Pharm Sci. 103(9):2724–2735.
  • Ilevbare GA, Liu H, Edgar KJ, Taylor LS. 2013. Maintaining supersaturation in aqueous drug solutions: impact of different polymers on induction times. Cryst Growth Des. 13(2):740–751.
  • Janssens S, Van den Mooter G. 2009. Review: physical chemistry of solid dispersions. J Pharm Pharmacol. 61(12):1571–1586.
  • Kiew TY, Cheow WS, Hadinoto K. 2015. Preserving the supersaturation generation capability of amorphous drug-polysaccharide nanoparticle complex after freeze drying. Int J Pharm. 484(1–2):115–123.
  • Lam M, Ghafourian T, Nokhodchi A. 2019. Liqui-pellet: the emerging next-generation oral dosage form which stems from liquisolid concept in combination with pelletization technology. AAPS PharmSciTech. 20(6):231.
  • Lee JH, Kim MJ, Yoon H, Shim CR, Ko HA, Cho SA, Lee D, Khang G. 2013. Enhanced dissolution rate of celecoxib using PVP and/or HPMC-based solid dispersions prepared by spray drying method. J Pharm Investig. 43(3):205–213.
  • Lin-Vien D, Colthup NB, Fateley WG, Grasselli JG. 1991. The handbook of infrared and Raman characteristic frequencies of organic molecules. San-Diego: Academic Press.
  • Maghsoodi M, Nokhodchi A, Azhdarzadeh Oskuei M, Heidari S. 2019. Formulation of cinnarizine for stabilization of its physiologically generated supersaturation. AAPS PharmSciTech. 20(3):139.
  • Maghsoodi M, Nokhodchi A, Babi HI. 2020. Rational selection of formulation components to improve dissolution of Dipyridamole. J Drug Deliv Sci Technol. 55:101467. doi.org/10.1016/j.jddst.2019.101467.
  • Matsushita T, Fecht HJ, Wunderlich RK, Egry I, Seetharaman S. 2009. Studies of the thermophysical properties of commercial CMSX-4 alloy. J Chem Eng Data. 54(9):2584–2592.
  • Morgen M, Bloom C, Beyerinck R, Bello A, Song W, Wilkinson K, Steenwyk R, Shamblin S. 2012. Polymeric nanoparticles for increased oral bioavailability and rapid absorption using celecoxib as a model of a low-solubility, high-permeability drug. Pharm Res. 29(2):427–440.
  • Mosquera-Giraldo LI, Borca CH, Parker AS, Dong Y, Edgar KJ, Beaudoin SP, Slipchenko LV, Taylor LS. 2018. Crystallization inhibition properties of cellulose esters and ethers for a group of chemically diverse drugs: experimental and computational insight. Biomacromolecules. 19(12):4593–4606.
  • Moustafine RI, Margulis EB, Sibgatullina LF, Kemenova VA, Mooter GV. 2008. Comparative evaluation of interpolyelectrolyte complexes of chitosan with Eudragit® L100 and Eudragit® L100-55 as potential carriers for oral controlled drug delivery. Eur J Pharm Biopharm. 70(1):215–225.
  • Moustafine RI, Zaharov IM, Kemenova VA. 2006. Physicochemical characterization and drug release properties of Eudragit E PO/Eudragit L 100-55 interpolyelectrolyte complexes . Eur J Pharm Biopharm. 63(1):26–36.
  • Paradkar AR, Chauhan B, Yamamura S, Pawar AP. 2003. Preparation and characterization of glassy celecoxib. Drug Dev Ind Pharm. 29(7):739–744.
  • Raina SA, Alonzo DE, Zhang GGZ, Gao Y, Taylor LS. 2014. Impact of polymers on the crystallization and phase transition kinetics of amorphous nifedipine during dissolution in aqueous media. Mol Pharm. 11(10):3565–3576.
  • Raina SA, Zhang GGZ, Alonzo DE, Wu J, Zhu D, Catron ND, Gao Y, Taylor LS. 2014. Enhancements and limits in drug membrane transport using supersaturated solutions of poorly water soluble drugs. J Pharm Sci. 103(9):2736–2748.
  • Shono Y, Jantratid E, Janssen N, Kesisoglou F, Mao Y, Vertzoni M, Reppas C, Dressman JB. 2009. Prediction of food effects on the absorption of celecoxib based on biorelevant dissolution testing coupled with physiologically based pharmacokinetic modeling. Eur J Pharm Biopharm. 73(1):107–114.
  • Thakral S, Thakral NK, Majumdar DK. 2013. Eudragit®: a technology evaluation. Expert Opin Drug Deliv. 10(1):131–149.
  • Warren DB, Benameur H, Porter CJH, Pouton CW. 2010. Using polymeric precipitation inhibitors to improve the absorption of poorly water-soluble drugs: a mechanistic basis for utility. J Drug Target. 18(10):704–731.
  • Williams HD, Trevaskis NL, Charman SA, Shanker RM, Charman WN, Pouton CW, Porter CJH. 2013. Strategies to address low drug solubility in discovery and development. Pharmacol Rev. 65(1):315–499.
  • Xie T, Taylor LS. 2016. Dissolution performance of high drug loading celecoxib amorphous solid dispersions formulated with polymer combinations. Pharm Res. 33(3):739–750.
  • Yokoi Y, Yonemochi E, Terada K. 2005. Effects of sugar ester and hydroxypropyl methylcellulose on the physicochemical stability of amorphous cefditoren pivoxil in aqueous suspension. Int J Pharm. 290(1–2):91–99.
  • Yoo S, Krill SL, Wang Z, Telang C. 2009. Miscibility/stability considerations in binary solid dispersion systems composed of functional excipients towards the design of multi-component amorphous systems. J Pharm Sci. 98(12):4711–4723.
  • Yoshida T, Kurimoto I, Umejima H, Watanabe S, Sako K, Kikuchi A. 2013. Effects of dissolved state of aminoalkyl methacrylate copolymer E/HCl on solubility enhancement effect for poorly water-soluble drugs. Colloid Polym Sci. 291(5):1191–1199.
  • Yoshida T, Kurimoto I, Yoshihara K, Umejima H, Ito N, Watanabe S, Sako K, Kikuchi A. 2012. Aminoalkyl methacrylate copolymers for improving the solubility of tacrolimus. I: evaluation of solid dispersion formulations. Int J Pharm. 428(1–2):18–24.
  • Zimmermann A, Millqvist-Fureby A, Elema MR, Hansen T, Müllertz A, Hovgaard L. 2009. Adsorption of pharmaceutical excipients onto microcrystals of siramesine hydrochloride: effects on physicochemical properties. Eur J Pharm Biopharm. 71(1):109–116.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.