Physicochemical Characterization and Dissolution Study of Solid Dispersions of Lovastatin with Polyethylene Glycol 4000 and Polyvinylpyrrolidone K30

REFERENCES

• Chiou W.L., Riegalman S. Pharmaceutical applications of solid dispersion systems. J. Pharm. Sci. 1971; 60: 1281–1302
   PubMed Web of Science ®Google Scholar
• Serajuddin A.T.M. Solid dispersions of poorly water-soluble drugs: Early promises, subsequent problems, and recent breakthroughs. J. Pharma. Sci. 1999; 88: 1058–1066
   PubMed Web of Science ®Google Scholar
• Leuner C., Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. Biopharm. 2000; 50: 47–60
   PubMed Web of Science ®Google Scholar
• Sekiguchi K., Obi N. Studies on absorption of eutectic mixtures. I. A comparison of the behaviour of eutectic mixture of sulfathiazole and that of ordinary sulfathiazole in man. Chem. Pharm. Bull. 1961; 9: 866–872
   Web of Science ®Google Scholar
• Margarit M.V., Rodri´guez I.C., Cerezo A. Physical characteristics and dissolution kinetics of solid dispersions of ketoprofen and polyethylene glycol 6000. Int. J. Pharm. 1994; 108: 101–107
   Web of Science ®Google Scholar
• Mura P., Faucci M.T., Manderioli A., Bramanti G., Parrini P. Thermal behavior and dissolution properties of naproxen from binary and ternary solid dispersions. Drug Dev. Ind. Pharm. 1999; 25: 257–264
   PubMed Web of Science ®Google Scholar
• El-Gazayerly O.N. Characterization and evaluation of tenoxicam coprecipitates. Drug Dev. Ind. Pharm. 2000; 26: 925–930
   PubMed Web of Science ®Google Scholar
• Ryh-Nam P., Jing-Huey C., Russel R.C. Enhancement of dissolution and bioavailability of piroxicam in solid dispersions systems. Drug Dev. Ind. Pharm. 2000; 26: 989–994
   PubMed Web of Science ®Google Scholar
• Craig D.Q.M. The mechanism of drug release from solid dispersion in water-soluble polymers. Int. J. Pharm. 2002; 231: 131–144
   PubMed Web of Science ®Google Scholar
• Taylor L.S., Zografi G. Spectroscopic characterization interactions between PVP and indomethacin in amorphous molecular dispersions. Pharm. Res. 1997; 14: 1691–1698
   PubMed Web of Science ®Google Scholar
• Yamashita K., Nakate T., Okimoto K., Ohike A., Tokunaga Y., Ibuki R., Higaki K., Kimura T. Establishment of new preparation method for solid dispersion formulation of tacrolimus. Int. J. Pharm. 2003; 267: 79–91
   PubMed Web of Science ®Google Scholar
• Susumu H., Takeshi H., Naho F., Akira K., Etsuo Y., Katsuhide T. Effects of water content in physical mixture and heating temperature on crystallinity of troglitazone-PVP K30 solid dispersions prepared by closed melting method. Int. J. Pharm. 2005; 302: 103–112
   PubMed Web of Science ®Google Scholar
• Teresa M. M., Victoria M. M., Gloria E. S. Characterization and solubility study of solid dispersions of flunarizine and polyvinylpyrrolidone. Il Farmaco. 2002; 57: 723–727
   PubMedGoogle Scholar
• Franco M., Trapani G., Latrofa A., Tullio C., Provenzano M.R., Serra M., Muggironi M., Biggio G., Liso G. Dissolution properties and anticonvulsant activity of phenytoin-polyethylene glycol 6000 and -polyvinylpyrrolidone K-30 solid dispersions. Int. J. Pharm. 2001; 225: 63–73
   PubMed Web of Science ®Google Scholar
• Van den Mooter G., Augustijns P., Blaton N., Kinget R. Physicochemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30. Int. J. Pharm. 1998; 164: 67–80
   Web of Science ®Google Scholar
• Melgardt M.V., Dale E.W., Jakkie G., Amol K. X-ray powder diffraction determination of the relative amount of crystalline acetaminophen in solid dispersions with PVP. Int. J. Pharm. 1998; 163: 219–224
   Google Scholar
• Arias M.J., Moyano J.R., Gines J.M. Study by DSC and HSM of the oxazepam PEG 6000 and oxazepam-D-mannitol systems: application to the preparation of solid dispersions. Thermochimica Acta. 1998; 321: 33–41
   Web of Science ®Google Scholar
• MacDonald J.S., Gerson R.J., Kornburst D.J., Kloss M.W., Prahalada S., Berry P.H., Alberts A.W., Bokelman D.L. Preclinical evaluation of lovastatin. Am. J. Cardiol. 1998; 62(15)16J–27J, Review
   Google Scholar
• Slater E.E., MacDonald J.S. Mechanism of action and biological profile of HMG CoA reductase inhibitors: A new therapeutic alternative. Drugs. 1998; 36(Suppl. 3)72–82
   Google Scholar
• Gerald S.B., Dean K.E., Micheal J.K. G.B. HarryLovastatin. Analytical Profiles of Drug Substances and Excipients, . Academic press, Inc, New York 1992; 21: 277–315
   Google Scholar
• Frances C., Veiga M.D., Espanol O.M., Cadorniga R. Preparation, characterization and dissolution of ciprofloxacin/PEG 6000 binary systems. Int. J. Pharm. 1991; 77: 193–198
   Web of Science ®Google Scholar
• Christian L., Jennifer D. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. Biopharm. 2000; 50: 47–60
   PubMed Web of Science ®Google Scholar
• Moore J.W., Flanner H. Mathematical comparison of dissolution profiles. Pharm. Technol. 1996; 20(6)64–74
   Google Scholar
• Barzegar-Jalali M., Maleki N., Garjani A., Khandar A.A., Haji-Hosseinloo M., Jabbari R.C, Dasmalchi S. Enhancement of dissolution rate and anti-inflammatory effects of piroxicam using solvent deposition technique. Drug Dev. Ind. Pharm. 2002; 28: 681–686
   PubMed Web of Science ®Google Scholar
• Tang L., Khan S.U., Muhmmad N.A. Evaluation and selection of bio-relevant dissolution media for a poorly water soluble new chemical entity. Pharm. Dev. Technol. 2001; 6: 531–540
   PubMed Web of Science ®Google Scholar
• Reppas C., Nicolaides E. J.B. Dressman, H. Lennernäs“Analysis of drug dissolution data'. Oral Drug Absorption Prediction and Assessment, . Marcel Dekker, Inc, New York 2000; 229–254
   Google Scholar
• Vueba M.L., Batista de Carvalho L.A.E., Veiga F., Sousa J.J., Pina M.E. Influence of cellulose ether polymers on ketoprofen release from hydrophilic matrix tablets. Eur. J. Pharm. Biopharm. 2004; 58: 51–59
   PubMed Web of Science ®Google Scholar
• Aulton M.E. Pharmaceutical Technology. Pharmaceutics: The Science of Dosage Form Design. Churchill Livingstone, London 1988; 600–616
   Google Scholar