Boronated Thymidine Analogues for Boron Neutron Capture Therapy

REFERENCES

• Soloway , A. H. , Tjarks , W. , Barnum , B. A. , Rong , F -G. , Barth , R. F. , Codogni , I. M. and Wilson , J. G. 1998 . The Chemistry of Neutron Capture Therapy . Chemical Reviews , 98 : 1515 – 1562 . [INFOTRIEVE] [CSA]
   PubMed Web of Science ®Google Scholar
• Al-Madhoun , A. S. , Johnsamuel , J. , Yan , J. , Ji , W. , Wang , J. , Zhuo , J -C. , Lunato , A. J. , Woollard , J. E. , Hawk , A. E. , Cosquer , G. Y. , Blue , T. E. , Eriksson , S. and Tjarks , W. 2002 . Synthesis of a Small Library of 3-(Carboranylalkyl)Thymidines and Their Biological Evaluation as Substrates for Human Thymidine Kinases 1 and 2 . Journal of Medicinal Chemistry , 45 : 4018 – 4028 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Byun , Y. , Yan , J. , Al-Madhoun , A. S. , Johnsamuel , J. , Yang , W. , Barth , R. F. , Eriksson , S. and Tjarks , W. 2005 . Synthesis and Biological Evaluation of Neutral and Zwitterionic 3-Carboranyl Thymidine Analogues for Boron Neutron Capture Therapy . Journal of Medicinal Chemistry , 48 : 1188 – 1198 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Johnsamuel , J. , Lakhi , N. , Al-Madhoun , A. S. , Byun , Y. , Yan , J. , Eriksson , S. and Tjarks , W. 2004 . Synthesis of Ethyleneoxide Modified 3-Carboranyl Thymidine Analogues and Evaluation of Their Biochemical, Physicochemical, and Structural Properties . Bioorganic & Medicinal Chemistry , 12 : 4769 – 4781 . [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Lunato , A. J. , Wang , J. , Woollard , J. E. , Anisuzzaman , A. K M. , Ji , W. , Rong , F -G. , Ikeda , S. , Soloway , A. H. , Eriksson , S. , Ives , D. H. , Blue , T. E. and Tjarks , W. 1999 . Synthesis of 5-(Carboranylalkylmercapto)-2'-Deoxyuridines and 3-(Carboranylalkyl)Thymidines and Their Evaluation as Substrates for Human Thymidine Kinases 1 and 2 . Journal of Medicinal Chemistry , 42 : 3378 – 3389 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Al-Madhoun , A. S. , Tjarks , W. and Eriksson , S. 2004 . The Role of Thymidine Kinases in the Activation of Pyrimidine Nucleoside Analogues . Mini-Reviews in Medicinal Chemistry , 4 : 341 – 350 . [INFOTRIEVE] [CSA]
   PubMed Web of Science ®Google Scholar
• Moore , C. , Hernandez-Santiago , B. I. , Hurwitz , S. J. , Tan , C. , Wang , C. and Schinazi , R. F. 2005 . The Boron-Neutron Capture Agent β- d-5-o-Carboranyl-2'-Deoxyuridine Accumulates Preferentially in Dividing Brain Tumor Cells . Journal of Neurooncology , 74 : 275 – 280 . [CROSSREF] [CSA]
   Google Scholar
• Busby , D. C. and Hawthorne , M. F. 1982 . The Crown Ether Promoted Base Degradation of p-Carborane . Inorganic Chemistry , 21 : 4101 – 4103 . [CROSSREF] [CSA]
   Google Scholar
• Barth , R. F. , Yang , W. , Al-Madhoun , A. S. , Johnsamuel , J. , Byun , Y. , Chandra , S. , Smith , D. R. , Tjarks , W. and Eriksson , S. 2004 . Boron-Containing Nucleosides as Potential Delivery Agents for Neutron Capture Therapy of Brain Tumors . Cancer Research , 64 : 6287 – 6295 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Al-Madhoun , A. S. , Johnsamuel , J. , Barth , R. F. , Tjarks , W. and Eriksson , S. 2004 . Evaluation of Human Thymidine Kinase 1 Substrates as New Candidates for Boron Neutron Capture Therapy . Cancer Research , 64 : 6280 – 6286 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Barth , R. F. , Adams , D. M. , Soloway , A. H. , Mechetner , E. B. , Alam , F. and Anisuzzaman , A. K. M. 1991 . Determination of Boron in Tissues and Cells Using Direct-Current Plasma Atomic Emission Spectroscopy . Analytical Chemistry , 63 : 890 – 893 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMed Web of Science ®Google Scholar
• Iida , H. , Yamazaki , N. and Kibayashi , C. 1987 . Total Synthesis of (+)-Nojirimycin and (+)-1-Deoxynojirimycin . Journal of Organic Chemistry , 52 : 3337 – 3342 . [CROSSREF] [CSA]
   Google Scholar
• Fujii , S. , Goto , T. , Ohta , K. , Hashimoto , Y. , Suzuki , T. , Ohta , S. and Endo , Y. 2005 . Potent Androgen Antagonists Based on Carborane as a Hydrophobic Core Structure . Journal of Medicinal Chemistry , 48 : 4654 – 4662 . [INFOTRIEVE] [CROSSREF] [CSA]
   Google Scholar
• Vlieghe , P. , Clerc , T. , Pannecouque , C. , Witvrouw , M. , De Clercq , E. , Salles , J. -P and Kraus , J. -L . 2001 . New 3′-Azido-3′-Deoxythymidin-5′-yl O-(4-Hydroxyalkyl or -Alkenyl or -Alkylepoxide) Carbonate Prodrugs: Synthesis and Anti-HIV Evaluation . Journal of Medicinal Chemistry , 44 : 3014 – 3021 . [INFOTRIEVE] [CROSSREF] [CSA]
   PubMedGoogle Scholar
• Klier , A. H. , Alves , R. J. , Auxiliadora , M. , Prado , F. , De Souza Filho , J. D. and D'Accorso , N. B. 2000 . Synthesis of New Five Membered Nitrogen Containing Heterocycles Bearing d-Galactose Side Chains . Synthetic Communications , 30 : 4361 – 4374 . [CSA]
   Web of Science ®Google Scholar