Efficient Transformation of Thymidine into 2′,3′-Didehydro-2′,3′-Dideoxy-Thymidine (D4T) Involving Opening of a 2,3′-Anhydro Derivative by Phenylselenol

References

• Barré-Sinoussi , F. , Chermann , J. C. , Rey , F. , Nugeyre , M. T. , Chamaret , S. , Gruest , J. , Dauguet , C. , Axler-Blin , C. , Vezinet-Brun , F. , Rouzioux , C. , Rozenbaum , W. and Montagnier , L. 1983 . Science , 220 : 868
   PubMed Web of Science ®Google Scholar
• Nasr , M. , Litterts , C. and Mc Growan . 1990 . J. Antiviral Res. , 14 : 125
   PubMed Web of Science ®Google Scholar
• De Las Heras , F. G. , Camarasa , M. J. and Fiandor , J. R. P. 1990 . Chem. Syn. Antib. , Edited by: Luckac , C. Vol. 320 , Heidelberg, Berlin : Springer-Verlag .
   Google Scholar
• Balzarini , J. and De Clercq , E. 1990 . “ Pharmacochemistry Library ” . In Design of Anti-AIDS Drugs , Edited by: De Clercq , E. Vol. 14 , 141 – 174 . Amsterdam : Elsevier .
   Google Scholar
• Huryn , D. M. and Okabe , M. 1992 . Chem. Rev. , 92 : 1745
   Web of Science ®Google Scholar
• De Clercq , E. 1988 . Adv. Drug. Res. , 17 : 1
   Google Scholar
• Mansuri , M. M. , Starett , J. E. Jr. , Ghazzouli , I. , Hitchcock , M. J. M. and Sterzycki , R. Z.
   Google Scholar
• Brankovan , V. , Lin , T.-S. , August , E. M. , Prusoff , W. H. , Sommadossi , J.-P. and Martin , J. C. 1989 . J. Med. Chem. , 32 : 461
   PubMed Web of Science ®Google Scholar
• Vial , J. M. , Agback , P. and Chattopadhyaya , J. 1990 . Nucleosides & Nucleotides , 9 : 245
   Web of Science ®Google Scholar
• Czernecki , S. and Valéry , J.-M. 1990 . J. Chem. Soc. Chem. Commun. , 801
   Google Scholar
• Horwitz , J. P. , Chua , J. , Da Rooge , M. , Noel , M. and Klundt , I. L. 1966 . J. Org. Chem. , 31 : 205
   PubMed Web of Science ®Google Scholar
• Martin , J. C. , Mansuri , M. M. , Starett , J. E. , Sommadossi , J.-P. , Brankovan , V. , Ghazzouli , I. , Ho , H.-T. and Hitchcock , M. J. M. 1989 . Nucleosides & Nucleotides. , 8 : 841
   Web of Science ®Google Scholar
• Mansuri , M. M. , Starett , J. E. Jr. , Wos , J. A. , Tortolani , D. R. , Brodfuehrer , P. R. , Howell , H. G. and Martin , J. C. 1989 . J. Org. Chem. , 54 : 4780
   Web of Science ®Google Scholar
• Chu , C. K. , Bhadti , V. S. , Doboszewski , P. , Gu , Z. P. , Kosugi , V. , Pullaiah , K. C. and Van Roey , P. 1989 . J. Org. Chem. , 54 : 2217
   Web of Science ®Google Scholar
• Cosford , N. D. P. and Schinazi , R. F. 1991 . J. Org. Chem. , 56 : 2161
   Web of Science ®Google Scholar
• Cosford , N. D. P. and Schinazi , R. F. 1993 . Nucleosides & Nucleotides , 12 : 149
   Web of Science ®Google Scholar
• Paulmier , C. 1986 . Selenium Reagents and Intermediates in Organic Synthesis , Oxford : Pergamon Press . Vol. 5
   Google Scholar
• Haraguchi , K. , Tanaka , H. , Maeda , H. , Itoh , Y. , Saito , S. and Miyasaka , T. 1991 . J. Org. Chem. , 56 : 5401
   Web of Science ®Google Scholar
• Vargeese , C. and Abushanab , E. 1992 . Nucleosides & Nucleotides , 11 : 1549
   Web of Science ®Google Scholar
• Grieco , P. A. and Miyashita , M. 1974 . J. Org. Chem. , 39 : 120
   Web of Science ®Google Scholar