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Articles

Methacrylic acid-co-butylmethacrylate copolymers: design, characterization and evaluation as encapsulating material for colon targeted formulations

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Pages 34-46 | Received 08 May 2015, Accepted 02 Sep 2015, Published online: 12 Oct 2015

References

  • Langholz E. Current trends in inflammatory bowel disease: the natural history. Ther. Adv. Gastroenterol. 2010;3: 77–86.
  • Baumgart DC, Sandborn WJ. Inflammatory bowel disease: clinical aspects and established and evolving therapies. Lancet. 2007;369:1641–1657.10.1016/S0140-6736(07)60751-X
  • Triantafillidis JK, Nasioulas G, Kosmidis PA. Colorectal cancer and inflammatory bowel disease: epidemiology, risk factors, mechanisms of carcinogenesis and prevention strategies. Anticancer Res. 2009;29:2727–2737.
  • Latella G, Papi C. Crucial steps in the natural history of inflammatory bowel disease. World J. Gastroenterol. 2012;18:3790–3799.10.3748/wjg.v18.i29.3790
  • Munkholm RL Review article: the incidence and prevalence of colorectal cancer in inflammatory bowel disease. Aliment Pharmacol. Ther. 18( Suppl. 2):1–5.
  • Molodecky NA, Soon IS, Rabi DM, et al. Increasing incidence and prevalence of the inflammatory bowel diseases with time, based on systematic review. Gastroenterology. 2012;142:46–54.10.1053/j.gastro.2011.10.001
  • Soon IS, Molodecky NA, Rabi DM, et al. The relationship between urban environment and the inflammatory bowel diseases: a systematic review and meta-analysis. BMC Gastroenterol. 2012;12:51.10.1186/1471-230X-12-51
  • Li Z, de Zhang K, Yi WQ, et al. NF-κB p65 antisense oligonucleotides may serve as a novel molecular approach for the treatment of patients with ulcerative colitis. Arch. Med. Res. 2008;39:729–734.10.1016/j.arcmed.2008.08.001
  • Oslen T, Cui G, Goll R, et al. Infliximab therapy decreases the levels of TNF-alpha and IFN-gamma mRNA in colonic mucosa of ulcerative colitis. Scand. J. Gastroenterol. 2009;44:727–735.
  • Carter MJ, Lobo AJ, Travis SPL. Guidelines for the management of inflammatory bowel disease in adults. Gut. 2004;53:1–6.10.1136/gut.2004.043372
  • Sandborn WJ. Oral 5-ASA therapy in Ulcerative colitis: what are the implications of the new formulations? J. Clin. Gastroenterol. 2008;42:338–344.10.1097/MCG.0b013e3181595b56
  • Sobczak M, Fabisiak A, Murawska N, et al. Current overview of extrinsic and intrinsic factors in etiology and progression of inflammatory bowel diseases. Pharmacol. Rep. 2014;66:766–775.10.1016/j.pharep.2014.04.005
  • Jain NK. Advances in controlled and novel drug delivery. 1st ed. New Delhi: CBS Publishers and Distributors; 2001. p. 89–119.
  • Jain SK, Jain A. Target-specific drug release to the colon. Expert Opin. Drug Delivery. 2008;5:483–498.10.1517/edd.2008.5.issue-5
  • Nemec JW, Bauer W. Acrylic and methacrylic acid polymers. In: Mark HF, Kroschwitz JL, editors. Encyclopedia of polymer science and engineering. 2nd ed. New York (NY): Wiley; 1985.p. 211–234.
  • Jones D. Pharmaceutical applications of polymers for drug delivery. In: Rapra review reports. Vol. 15. UK: Rapra Technology Ltd; 2004. p. 3–4.
  • Thakral SK, Thakral NK, Majumdar DK. Eudragit®: a technology evaluation. Expert Opin. Drug Delivery. 2013;10:131–149.10.1517/17425247.2013.736962
  • Muñoz-Muñoz F, Ruiz JC, Alvarez-Lorenzo C, et al. Novel interpenetrating smart polymer networks grafted onto polypropylene by gamma radiation for loading and delivery of vancomycin. Eur. Polym. J. 2009;45:1859–1867.10.1016/j.eurpolymj.2009.04.023
  • Loughlin RG, Tunney MM, Donnelly RF, et al. Modulation of gel formation and drug-release characteristics of lidocaine-loaded poly(vinyl alcohol)-tetraborate hydrogel systems using scavenger polyol sugars. Eur. J. Pharm. Biopharm. 2008;69:1135–1146.10.1016/j.ejpb.2008.01.033
  • Vijay S, Sati OP, Majumdar DK. Acrylic acid–methyl methacrylate copolymer for oral prolonged drug release. J. Mater. Sci.: Mater. Med. 2010;21:2583–2592.
  • Vijay S, Sati OP, Majumdar DK. Acrylic acid–methyl methacrylate (2.5:7.5/2:8) enteric copolymer for targeted drug delivery. J. Mater. Sci.: Mater. Med. 2010; 22:125–135.
  • Kanevskaya YA, Shchepilov AM, Zubov PI. The effect of the supermolecular structure of coatings of a copolymer of butyl methacrylate and methacrylic acid on durability. Polym. Sci. USSR. 1970;12:2201–2206.10.1016/0032-3950(70)90449-1
  • Konstantinopolskaya MB, Kanevskaya YA, Karyakina MI, et al. The structure of a copolymer of butyl methacrylate and methacrylic acid. Polym. Sci. USSR. 1965:1102–1105.10.1016/0032-3950(65)90386-2
  • Qui X, Song G, Chu X, et al. microencapsulated n-alkane with p (n-butyl methacrylate-co-methacrylic acid) shell as phase change materials for the thermal energy storage. Solar Energy. 2013;91:212–220.
  • Bezuglyi VD, Voskresenskaya IB, Alekseyeva TA, et al. Investigation of the copolymerization of methacrylic acid with methyl acrylate and butyl methacrylate in water–dioxan solvent systems. Polym. Sci. USSR. 1975;17:112–116.10.1016/0032-3950(75)90222-1
  • Scherrer RA, Whitehouse MW. Anti-inflammatory agents. New York (NY): Academic Press; 1974. p. 33.
  • Neil MJ, editor. The Merck index: an encyclopedia of chemicals, drugs and biological. 14th ed. Whitehouse station (NJ). Merck Research Laboratories Division of Merck & Co.; 2006. p. 582.
  • Dooley M, Spencer CM, Dunn CJ. Aceclofenac: a reappraisal of its use in the management of pain and rheumatic disease. Drugs. 2001;61:1351–1378.10.2165/00003495-200161090-00012
  • Meyer JH, Dressman J, Fink AS, et al. Effect of size and density on gastric emptying of indigestible solids. Gastroenterology. 1985;89:805–813.
  • Rodrı́guez M, Vila-Jato JL, Torres D. Design of a new multiparticulate system for potential site specific and controlled drug delivery to the colonic region. J. Controlled Release. 1998;55:67–77.10.1016/S0168-3659(98)00029-7
  • Xiang-HuaQu, QWu, GQChen. In vitro study on hemocompatibility and cytocompatibility of poly(3-hydroxybutyrate-co-3-hydroxyhexanoate). J. Biomater. Sci. Polym. Ed. 2006; 17:1107–1121.10.1163/156856206778530704
  • Chowdhary KPR, Srinivasa RY. Design and in vitro and in vivo evaluation of mucoadhesive microcapsule of glipizide for oral controlled release: a technical note. AAPS Pharm. Sci. Tech. 2003; 4:320–325.
  • Morris GD, Beck PL, Herridg MS, et al. Hapten-induced model of chronic inflammation and ulceration in the rat colon. Gastroenterology. 1989;96:795–803.
  • Krawisz JE, Sharon P, Stenson WF. Quantitative assay for acute intestinal inflammation based on myeloperoxidase activity. Assessment of inflammation in the rat and hamster model. Gastroenterology. 1984;87:1344–1350.
  • Ju RTC, Nixon PR, Patel MV. Drug release from hydrophilic matrices. 1. New scaling laws for predicting polymer and drug release based on the polymer disentanglement concentration and the diffusion layer. J. Pharm. Sci. 1995;84:1455–1463.10.1002/(ISSN)1520-6017
  • Kerbers R, Glamann H. Lösungsmitteleinflüsse auf die copolymerisations parameter des systems methylmethacrylat/acrylsäure [Solvent effects on the reactivity ratios of the system methyl methacrylate / acrylic acid]. Die Makromolekulare Chemie, German. 1967;100:290.10.1002/macp.1967.021000134
  • Thakral S, Thakral NK, Majumdar DK. Eudragit®: a technology evaluation. Expert Opin. Drug Delivery. 2013;10:131–149.10.1517/17425247.2013.736962
  • Ito Y, Casolaro M, Kono K, et al. An insulin-releasing system that is responsive to glucose. J. Controlled Release. 1989;10:195–203.10.1016/0168-3659(89)90063-1
  • Autian J Biological model systems for the testing of the toxicity of biomaterials. Polymers in medicine and surgery. In: Kronethal RL, Oser Z, Martin E, editors. Polymer science and technology. New York (NY): Plenum Press; 1993. p. 181.
  • Maghsoodi M. Physicomechanical properties of naproxen-loaded microparticles prepared from Eudragit L100. AAPS PharmSciTech. 2009;10:120–128.10.1208/s12249-009-9186-5
  • Shargel L, Yu A Applied biopharmaceutics & pharmacokinetics. London, UK: Printice-Hall International Inc.; 1999. p. 173.
  • Peppas NA. Analysis of fickian and non-fickian drug release from polymers. Pharm Acta Helv. 1985;60:110–111.
  • Chueh HR, Zia H, Rhodes CP. Optimization of sotalol floating and bioadhesive extended release tablet formulations. Drug Dev. Ind. Pharm. 1995;21:1725–1747.10.3109/03639049509069261

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