459
Views
53
CrossRef citations to date
0
Altmetric
Research Article

Evaluation of Critical Formulation Factors in the Development of a Rapidly Dispersing Captopril Oral Dosage Form

, , , , , & show all
Pages 967-979 | Published online: 10 Aug 2003

References

  • Seager H. Drug delivery products and the Zydis fast dissolving dosage form. J. Pharm. Pharmacol 1998; 50(4)375–382
  • Johannessen T., Kristensen P. On-demand therapy in gastroesophageal reflux disease: a comparison of the early effects of single doses of fast dissolving famotidine wafers and ranitidine tablets. Clin. Ther. 1997; 19(1)73–81
  • The fifth report of the joint national committee on detection, evaluation, and treatment of high hlood pressure (JNC V). Arch. Intern. Med. 1993; 153(2)154–183
  • Nur A.O., Zhang J.S. Recent progress in sustained/controlled oral delivery of captopril: an overview. Int. J. Pharm. 2000; 194(2)139–146
  • Ohman K.P., Kagedal B., Larsson R., Kalberg E.B. Pharmacokinetics of captopril and its effect on blood pressure during acute and chronic administration and in relation to food intake. J. Cardiovasc. Pharm. 1985; 7: S20–S24
  • Ceyhan B., Karaaslan Y., Caymaz O., Oto A., Oram E., Oram A., Ugurlu S. Comparison of sublingual captopril and sublingual nifedifine in hypertensive emergencies. Jpn. J. Pharmacol. 1990; 52: 189–193
  • Angeli P., Chiesa M., Caregaro L., Merkel C., Sacerdoti D., Rondana M., Gatta A. Comparison of sublingual captopril and nifedipine in immediate treatment of hypertensive emergencies. Arch. Intern. Med. 1991; 151: 678–682
  • Karachalios G.N., Chrioskos N., Kintziou H., Perogianopouos K., Kehagioglow K. Treatment of hypertensive crisis with sublingual captopril. Curr. Ther. Res. 1990; 48(1)5–9
  • Haude M., Steffen W., Erbel R., Meyer J. Sublingual administration of captopril versus nitroglycerin in patients with severe heart failure. Int. J. Cardiology 1990; 27: 351–359
  • Al-Furaih T.A., McElnay J.C., Elborn J.S., Rusk R., Scott M.G., McMahon J., Nicholls D.P. Sublingual captopril—a pharmacokinetic and pharmacodynamic evaluation. Eur. J. Clin. Pharmacol. 1991; 40: 393–398
  • McElnay J.C., Al-Furaih T.A., Hughes C.M., Scott M.G., Nicholls D.P. A pharmacokinetic and pharmacodynamic evaluation of buffered sublingual captopril in patients with congestive heart failure. Eur. J. Clin. Pharmacol. 1996; 49(6)471–476
  • Kearney P., Wong S.K. Method for Making Freeze Dried Drug Dosage Forms. US Patent 5,631,023, May 20, 1997
  • Green R., Kearney P. Process for Preparing Fast Dispersing Solid Oral Dosage Form. US Patent 5,976,577, November 2, 1999
  • Mizumoto T., Masuda Y., Fukui M. Intrabuccally Dissolving Compressed Moldings and Production Process Thereof. US Patent 5,576,014, November 19, 1996
  • Dijkgraaf B.L.J., Muhlenbruch A. Granulate for the Preparation of Fast-Disintegrating and Fast-Dissolving Compositions Containing A High Amount of Drug. US Patent 5,837,292, November 17, 1998
  • Khankari R.K., Hontz J., Chastain S.J., Katzner L. Rapidly Dissolving Robust Dosage Form. US Patent 6,024,981, February 15, 2000
  • Pather S.I., Robinson J.R., Eichman J.D., Khankari R.K., Hontz J., Gupte S.V. Effervescent Drug Delivery System for Oral Administration. US Patent 6,391,335, May 21, 2002
  • Fuisz R.C. Rapidly Dispersible Compositions Containing Polydextrose. US Patent 5,501,858, March 26, 1996
  • Myers G.L., Battist G.E., Fuisz R.C. Process and Apparatus for Making Rapidly Dissolving Dosage Units and Product Therefrom. US Patent 5,866,163, February 2, 1999
  • Sachs E.M., Haggerty J.S., Cima M.J., Williams P.A. Three-Dimensional Printing Techniques. US Patent 5,204,055, April 20, 1993
  • Cima M.J., Sachs E., Cima L.G., Yoo J., Khanuja S., Borland S.W., Wu B., Giordano R.A. Computer-derived microstructures by 3D printing: Bio- and Structural Materials. Solid Freeform Fabrication Symposium Proceedings. Univ. of Texas, 1994; 181–190
  • Wu B.M., Borland S.W., Giordano R.A., Cima L.G., Sachs E.M., Cima M.J. Solid freeform fabrication of drug delivery devices. J. Control. Release 1996; 40: 77–87
  • Katstra W.E., Palazzolo R.D., Rowe C.W., Giritlioglu B., Teung P., Cima M.J. Oral dosage forms fabricated by three dimensional printing. J. Control. Release 2000; 66(1)1–9
  • Rowe C.W., Katstra W.E., Palazzolo R.D., Giritlioglu B., Teung P., Cima M.J. Multimechanism oral dosage forms fabricated by three dimensional printing. J. Control. Release 2000; 66(1)11–17
  • Lin S., Chao P., Chien Y.W., Sayani A., Kumar S., Mason M., West T., Yang A., Monkhouse D.C. In vitro and in vivo evaluations of biodegradable implants for hormone replacement therapy: effect of system design and PK-PD relationship. AAPS Pharm. Sci. Tech. 2001; 2(3), Article 16
  • Yoo J., Kumar S., Rowe C.W., Monkhouse D.C., Shanahan G., Kang A. Factors influencing the dispersion of rapidly dissolving oral dosage forms fabricated by the TheriForm™ process. AAPS Pharm. Sci. 1999; 1(1), 1998 AAPS Annual Meeting Supplement
  • Rowe C.W., Wang C., Monkhouse D. TheriForm technology. Modified-Release Drug Delivery Technology, M.J. Rathbone, J. Hadgraft, M.S. Roberts. Marcel Dekker, Inc. 2002; 77–87
  • Yoo J., Kumar S., Monkhouse D. Dosage Form Exhibiting Rapid Disperse Properties, Methods of Use and Process for the Manufacture of Same. US Patent 6,471,992, October 29, 2002
  • Pereira C.M., Tam Y.K. Simplified determination of captopril in plasma by high performance liquid chromatography. J. Chromatogr. 1988; 425: 208–213
  • Tsai T., San Y.P., Ho H.S., Wu J.S., Sheu M.T. Film-forming polymer-granulated excipients as the matrix materials for controlled release dosage form. J. Control. Release 1998; 51(2–3)289–299
  • Draper N.R., Smith H. Selecting the best regression equation. Applied Regression Analysis, 2nd Ed. Wiley, New York 1981; 225–311
  • Seta Y., Higuchi F., Kawahar Y., Nishimura K., Okada R. Design and preparation of captopril sustained-release dosage forms and their biopharmaceutical properties. Int. J. Pharm. 1988; 29: 245–254
  • Allen L.V., Erickson M.A. Stability of baclofen, captopril, diltiazem hydrochloride, dipyramide, and flecainide acetate in extemporaneously compounded oral liquids. Am. J. Health-Syst. Ph. 1996; 53(18)2179–2184
  • Yoo J. Comprehensive report on the development and process scale up of pseudoephedrine HCl TheriFlash™ dosage form. Internal Communications, Therics, Inc. 1999, On file

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.