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Patent Evaluations

Indole-2-carboxamide derivatives: a patent evaluation of WO2015036412A1

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Bibliography

  • Papers of special note have been highlighted as either of interest (●) or of considerable interest (●●) to readers.
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● Atypical antipsychotics act through stimulation of neurogenesis.

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●● Development of one of the most promising class of small-molecule neurogenesis inducers.

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●● Report on first small-molecule neurogenesis inducer in clinical testing, Phases Ia and Ib.

  • Jagasia R, Jakob-Roetne R, Peters J-U, et al. Preparation of indol-carboxamide derivatives as neurogenic agents. WO2015036412A1. 2015.

● The evaluated patent application.

  • Ceccarelli SM, Jagasia R, Jakob-Roetne R, et al. Preparation of benzisoxazoles as modulators of neurogenesis. WO2014016267A1. 2014.
  • Ceccarelli SM, Jagasia R, Jakob-Roetne R, et al. Preparation of benzimidazoles as CNS active agents. WO2014053409A1. 2014.
  • Ceccarelli SM, Jagasia R, Jakob-Roetne R, et al. Neurogenesis-stimulating isoquinoline derivatives. WO2014177596A1. 2014.
  • Ceccarelli SM, Jagasia R, Jakob-Roetne R, et al. Preparation of 1,7-naphthyridine derivatives as neurogenesis stimulators for treatment of neurological diseases and neuropsychiatric disorders. WO2015014768A1. 2015.
  • Ceccarelli SM, Jagasia R, Jakob-Roetne R, et al. Preparation of substituted 1,6-naphthyridines. WO2014079787A1. 2014.
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