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Review

Drug delivery across the skin

Pages 1887-1937 | Published online: 23 Feb 2005

Bibliography

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  • •Description of a new type of skin permeation enhancer.
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  • •One of the first studies investigating the relationship between the chemistry of an enhancer and its effect on skin permeabil-ity.
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  • BOMMANNAN D, OKUYAMA H, STAUFFER P, GUY RH: Sonophoresis. I. The use of high-frequency ultrasound to enhance transdermal drug delivery. Pharm. Res. (1992) 9(0559–564.
  • MENON GK, BOMMANNAN DB, ELIAS PM: High-frequency sonophoresis: permeation pathways and structural basis for enhanced permeability. Skin. Phar-macol. (1994) 7(3):130–139.
  • MITRAGOTRI S, EDWARDS DA, BLANKSCHTEIN D, LAN-GER R: A mechanistic study of ultrasonically enhanced transdermal drug delivery. J. Pharm. Sci. (1995) 84 (6) 697–706.
  • •A scholarly paper which describes the effect of ultrasound on the skin.
  • MENON GK, PRICE LF, BOMMANNAN B et al Selective obliteration of the epidermal calcium gradient leads to enhanced lamellar body secretion. J Invest. Dermatol. (1994) 102 (5) 789–795
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  • MITRAGOTRI S, BLANKSCHTEIN D, LANGER R: Transder-mal drug delivery using low-frequency sonophoresis. Pharm. Res. (1996) 13(3):411–420.
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  • •Good, review article written by opinion leaders.
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  • GREEN PG, FLANAGAN M, SHROOT B, GUY R: Iontopho-retie drug delivery. In: Pharmaceut. Skin Penetration En-hancement. Walters K, Hadgraft J (Eds.), Marcel Dekker, New York (1993):297–319.
  • SINGH P, MAIBACH HI: Transdermal iontophoresis: pharmacokinetic considerations. Din. Pharmacokinet. (1994) 26(5) 327–334.
  • COSTELLO CT, JESKE AH: Iontophoresis: applications in transdermal medication delivery. Phys, Ther. (1995) 75 (6) :554–563.
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  • BANGA AK CHIEN YW: Hydrogel-based iontotherapeu-tic delivery devices for transdermal delivery of pep-tide/protein drugs. Pharm, Res, (1993) 10(5):697–702.
  • •Good paper.
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  • HEIT MC, MONTEIRO-RIVIERE NA, JAYES FL, RIVIERE JE: Transdermal iontophoretic delivery of luteinizing hor-mone releasing hormone (LHRH): effect of repeated ad-ministration. Pharm, Res. (1994) 11 (7) :1000–1003 .
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  • •Important paper discussing the factors that contribute to ion-tophoretic flow.
  • KIM A, GREEN PG, RAO G, GUY RH: Convective solvent flow across the skin during iontophoresis. Pharm, Res, (1993) 10(9):1315–1320.
  • CRAANE VAN HINSBERG WH, BAX L, FLINTERMAN NH et al.: Iontophoresis of a model peptide across human skin in vitro: effects of iontophoresis protocol, pH and ionic strength on peptide flux and skin impedance. Pharm, Res, (1994) 11(9):1296–300.
  • POTTS RO, GUY RH, FRANCOEUR ML: Routes of ionic per-meability through mammalian skin. Solid States Ionics (1992) 53–56:165–169.
  • KALIA YN, GUY RH: The electrical characteristics of hu-man skin in vivo. Pharm, Res. (1995) 12(10:1605–1613.
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  • •A good introductory paper.
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  • The Dermal Lymphatic Capillaries. Daróczy J (Ed.), Springer, Berlin (1989):2.
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  • •Good summary of a decade of experience with TTS oestra diol.
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  • LANGLEY MS, HEEL RC: Transdermal clonidine. A pre-liminary review of its pharmacodynamic properties and therapeutic efficacy. Drugs (1988) 35 (2):123–142.
  • •An early review of the performance of TTS clonidine in the praxis.
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  • •A useful review of the, somewhat disputed, anti-emetic treat-ment TTS.
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  • •A useful review article.
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