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Miscellaneous

Ultraselective antagonists of the d-opioid receptor

, , , , , & show all
Pages 45-47 | Published online: 25 Feb 2005

Reference

  • GUERRINI R et al.: Opioid receptor selectivity alteration by single residue replacement: synthesis and activity profile of [Dmti ]deltorphin B. Eur. J. Pharmacol. (1996) 302:37–42.
  • CAPASSO A et al.: Dmt-Tic-OH, a highly selective and potent 6-opioid dipeptide receptor antagonist after systemic administration in the mouse. Life Sci. (1996) 59:93–98.
  • BALBONI G et al.: Opioid diketopiperazines: synthesis and activity of a prototypic class of opioid antagonists. Biol. Chem. (1997) 378:19–29.
  • BRYANT SD et al.: Opioid diketopiperazines: refinement of the 6 opioid antagonist pharmacophore. Biol. Chem. (1997) 378:107–114.
  • SALVADORI S et al: Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary 6 opioid antagonist activity. J. Med. Chem. (1997) 40:3100–3108.
  • BRYANT SD et al: New 6-opioid antagonists: ideal pharmacological probes. Trends PharmacoL Sci. (In Press).
  • LAZARUS LH et al.: Opioid infidelity: novel opioid peptides with dual high affinity for 6-and µ-receptors. Trends Neurosci. (1996) 19:31–35.

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