116
Views
4
CrossRef citations to date
0
Altmetric
Original Research

Evaluation of in vivo behavior of controlled and pulsatile release pastilles using pharmacokinetic and γ-scintigraphic techniques

, MPharm PhD, , MPharm PhD & , MPharm PhD
Pages 1333-1345 | Published online: 28 Aug 2012

Bibliography

  • Shukla D, Chakraborty S, Singh S, Mishra B. Lipid based oral multiparticulate formulations – Advantages, technological advances and industrial applications. Expert Opin Drug Deliv 2011;8:207-24
  • Shukla D, Chakraborty S, Singh S, Mishra B. Pastillation: a novel technology for development of oral lipid based multiparticulate controlled release formulation. Powder Technol 2011;209:65-72
  • Shukla D, Chakraborty S, Mishra B. In vitro and in vivo evaluation of multilayered pastilles for chronotherapeutic management of nocturnal asthma. Expert Opin Drug Deliv 2012;9:9-18
  • Shukla D, Chakraborty S, Singh S, Mishra B. Doxofylline: a promising methylxanthine derivative for the treatment of asthma and chronic obstructive pulmonary disease. Expert Opin Pharmacother 2009;10:2343-56
  • Davis SS, Hardy JG, Fara JW. Transit of pharmaceutical dosage forms through the small intestine. Gut 1986;27:886-92
  • Dressman JB, Berardi RR, Elta GH, Absorption of flurbiprofen in the fed and fasted state. Pharm Res 1992;9:901-7
  • Snape WJ Jr, Battle WM, Schwartz SS, Metoclopramide to treat gastroparesis due to diabetes mellitus: a double-blind, controlled trial. Ann Intern Med 1982;96:444-6
  • Wilding IR, Davis SS, O’Hagan DT. Optimizing gastrointestinal delivery of drugs. Bailliere's Clin Gastroenterol 1994;8:255-70
  • Damle B, Ullah I, Doll W, Pharmacokinetics and gamma scintigraphy evaluation of two enteric coated formulations of didanosine in healthy volunteers. Br J Clin Pharmacol 2002;54:255-61
  • Wilding IR, Coupe AJ, Davis SS. The role of gamma scintigraphy in oral drug delivery. Adv Drug Deliv Rev 1991;7:87-117
  • Davis SS, Hardy JG, Newman SP, Wilding IR. Gamma scintigraphy in the evaluation of pharmaceutical dosage forms. Eur J Nuclear Med 1992;19:971-86
  • Rastogi R, Sultana Y, Aqil M, Alginate microspheres of isoniazid for oral sustained drug delivery. Int J Pharm 2007;334:71-7
  • Digenis GA. The utilization of short-lived radionuclide in the assessment of formulation and in vivo disposition of drugs. In: Wilson CG, Hardy JG, editors. Radionuclide imaging in drug research. Croom Helm; London: 1982. p. 103-43
  • Digenis GA, Parr AF, Jay M. Neutron activation methods for evaluation of pharmaceutical dosage forms. In: Hardy JG, Davis SS, Wilson CG, editors. Drug delivery to the gastrointestinal tract. Ellis Horwood press; Chichester, England: 1989. p. 111-19
  • Digenis GA, Sandefer EP. Gamma scintigraphy and neutron activation techniques in the in vivo assessment of orally administered dosage forms. Crit Rev Ther Drug Carrier Syst 1991;7:309-45
  • Digenis GA, Sandefer EP, Page RC, Doll WJ. Gamma scintigraphy: an evolving technology in pharmaceutical formulation development - Part 1. Pharm Sci Technol Today 1998;1:100-7
  • Fell JT, Digenis GA. Imaging and behaviour of solid oral dosage forms in vivo. Int J Pharm 1984;22:1-16
  • Spiller RC. Where do all the tablets go in 1986? Gut 1986;27:879-85
  • Wilson CG, Washington N. Assessment of disintegration and dissolution of dosage forms in vivo using gamma scintigraphy. Drug Dev Ind Pharm 1988;14:211-18
  • Digenis GA, Sandefer EP, Page RC, Doll WJ. Gamma scintigrapy: an evolving technology in pharmaceutical formulation development - Part 2. Pharm Sci Technol Today 1998;1:160-5
  • Casey DL, Beihn RM, Digenis GA, Shabhu MB. Method for monitoring hard gelatin capsule disintegration times in humans using external scintigraphy. J Pharm Sci 1976;65:1412-13
  • Theodorakis MC, Digenis GA, Beihn RM, Rate and pattern of gastric emptying in human using 99 mTc-labeled triethylenetetraamine- polystyrene resin. J Pharm Sci 1980;69:568-71
  • Harris D, Fell JT, Sharma HL, Taylor DC. GI transit of potential bioadhesive formulations in man: a scintigraphic study. J Control Release 1990;12:45-53
  • Christian PE, Moore JG, Sorenson JA, Effects of meal size and correction technique on gastric emptying time: studies with two tracers and opposed detectors. J Nucl Med 1980;9:883-5
  • Palin KJ, Whalley DR, Wilson CG, Determination of gastric-emptying profiles in the rat: influence of oil structure and volume. Int J Pharm 1982;12:315-22
  • Haruta S, Kawai K, Jinnouchi S, Evaluation of absorption kinetics of orally administered theophylline in rats based on gastrointestinal transit monitoring by gamma scintigraphy. J Pharm Sci 2000;90:464-73
  • Goggin JM, Hoskinson JJ, Butine MD, Scintigraphic assessment of gastric emptying of canned and dry diets in healthy cats. Am J Ver Res 1998;59:388-92
  • Gannu R, Bandari S, Sudke SG, Development and validation of a stability-indicating RP-HPLC method for analysis of doxofylline in human serum. Application of the method to a pharmacokinetic study. Acta Chromatographica 2007;9:149-60
  • Meier J, Nuesch E, Schmidt R. Pharmacokinetic criteria for the evaluation of retard formulations. Eur J Clin Pharmacol 1974;76:429-32
  • Ma N, Xu L, Wang Q, Development and evaluation of new sustained-release floating microspheres. Int J Pharm 2008;358:82-90
  • Atyabi F, Sharma HL, Mohammad HAH, Fell JT. In vivo evaluation of a novel gastric retentive formulation based on ion exchange resins. J Control Release 1996;42:105-13
  • Jain SK, Agrawal JP, Jain NK. A novel calcium silicate based microspheres of repaglinide: in vivo investigations. J Control Release 2006;113:111-16
  • Bressolle F, Bromet-Petit M, Audran M. Validation of liquid chromatographic and gas chromatographic methods applications to pharmacokinetics. J Chromatogr B 1996;686:3-10
  • Jayasagar G, Krishna Kumar M, Chandrasekhar K, Validated HPLC method for the determination of celecoxib in human serum and its application in a clinical pharmaceutical study. Pharmazie 2002;57:619-21

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.