Evaluation of coat uniformity and taste-masking efficiency of irregular-shaped drug particles coated in a modified tangential spray fluidized bed processor

Bibliography

• Al-Khattawi A, Mohammed AR. Compressed orally disintegrating tablets: excipients evolution and formulation strategies. Expert Opin Drug Deliv 2013;10:651-63
   PubMed Web of Science ®Google Scholar
• Shahiwala A. Formulation approaches in enhancement of patient compliance to oral drug therapy. Expert Opin Drug Deliv 2011;8:1521-9
   PubMed Web of Science ®Google Scholar
• European Medicines Agency, Committee for Medicinal Products for Human Use (CHMP). Reflection Paper: Formulations of choice for the paediatric population. Adoption by CHMP Sept. 21, 2006. Available From http://www.ema.europa.eu/docs/en_GB/document_library/Scientific_guideline/2009/09/WC500003782.pdf [Last Accessed 14 January 2015]
   Google Scholar
• European Medicines Agency. Guideline on pharmaceutical development of medicines for paediatric use. EMA/CHMP/QWP/805880/2012 Rev. 2, Adoption by CHMP July 2013. Available From http://www.ema.europa.eu/docs/en_GB/document_library/Scientific_guideline/2013/07/WC500147002.pdf [Last Accessed 18 May 2015]
   Google Scholar
• Douroumis D. Orally disintegrating dosage forms and taste-masking technologies. Expert Opin Drug Deliv 2011;8:665-75
   PubMed Web of Science ®Google Scholar
• Sohi H, Sultana Y, Khar RK. Taste masking technologies in oral pharmaceuticals: recent developments and approaches. Drug Dev Ind Pharm 2004;30:429-48
   PubMed Web of Science ®Google Scholar
• Kondo K, Ito N, Niwa T, et al. Design of sustained release fine particles using two-step mechanical powder processing: Particle shape modification of drug crystals and dry particle coating with polymer nanoparticle agglomerate. Int J Pharm 2013;453:523-32
   PubMed Web of Science ®Google Scholar
• Jono K, Ichikawa H, Miyamoto M, et al. A review of particulate design for pharmaceutical powders and their production by spouted bed coating. Powder Technol 2000;113:269-77
   Web of Science ®Google Scholar
• Ishida M, Uchiyama J, Isaji K, et al. A novel approach to a fine particle coating using porous spherical silica as core particles. Drug Dev Ind Pharm 2014;40:1054-64
   PubMed Web of Science ®Google Scholar
• Watano S, Nakamura H, Hamada K, et al. Fine particle coating by a novel rotating fluidized bed coater. Powder Technol 2004;141:172-6
   Web of Science ®Google Scholar
• Kaewklum R, Kuprianov VI. Experimental studies on a novel swirling fluidized-bed combustor using an annular spiral air distributor. Fuel 2010;89:43-52
   Web of Science ®Google Scholar
• Ortega-Casanova J. CFD and correlations of the heat transfer from a wall at constant temperature to an impinging swirling jet. Int J Heat Mass Transfer 2012;55:5836-45
   Web of Science ®Google Scholar
• Özbey M, Söylemez MS. Effect of swirling flow on fluidized bed drying of wheat grains. Energy Convers Manage 2005;46:1495-512
   Web of Science ®Google Scholar
• Heng PWS, Chan LW, Tang ESK. Use of swirling airflow to enhance coating performance of bottom spray fluid bed coaters. Int J Pharm 2006;327:26-35
   PubMed Web of Science ®Google Scholar
• Bouwman AM, Bosma JC, Vonk P, et al. Which shape factor(s) best describe granules? Powder Technol 2004;146:66-72
   Web of Science ®Google Scholar
• Shiino K, Iwao Y, Miyagishima A, et al. Optimization of a novel wax matrix system using aminoalkyl methacrylate copolymer E and ethylcellulose to suppress the bitter taste of acetaminophen. Int J Pharm 2010;395:71-7
   PubMed Web of Science ®Google Scholar
• Turton R. Challenges in the modeling and prediction of coating of pharmaceutical dosage forms. Powder Technol 2008;181:186-94
   Web of Science ®Google Scholar
• Er DZL, Liew CV, Heng PWS. Layered growth with bottom-spray granulation for spray deposition of drug. Int J Pharm 2009;377:16-24
   PubMed Web of Science ®Google Scholar
• Wong PM, Chan LW, Heng PWS. Investigation on side-spray fluidized bed granulation with swirling airflow. AAPS PharmSciTech 2012;14:211-21
   PubMed Web of Science ®Google Scholar
• Tang ESK, Wang LK, Liew CV, et al. Drying efficiency and particle movement in coating-impact on particle agglomeration and yield. Int J Pharm 2008;350:172-80
   PubMed Web of Science ®Google Scholar
• Cuppok Y, Muschert S, Marucci M, et al. Drug release mechanisms from Kollicoat SR: Eudragit NE coated pellets. Int J Pharm 2011;409:30-7
   PubMed Web of Science ®Google Scholar
• Albertini B, Cavallari C, Passerini N, et al. Characterization and taste-masking evaluation of acetaminophen granules: comparison between different preparation methods in a high-shear mixer. Eur J Pharm Sci 2004;21:295-303
   PubMed Web of Science ®Google Scholar
• Maniruzzaman M, Boateng JS, Bonnefille M, et al. Taste masking of paracetamol by hot-melt extrusion: an in vitro and in vivo evaluation. Eur J Pharm Biopharm 2012;80:433-42
   PubMed Web of Science ®Google Scholar
• Suzuki H, Onishi H, Takahashi Y, et al. Development of oral acetaminophen chewable tablets with inhibited bitter taste. Int J Pharm 2003;251:123-32
   PubMed Web of Science ®Google Scholar
• Anand V, Kataria M, Kukkar V, et al. The latest trends in the taste assessment of pharmaceuticals. Drug Discov Today 2007;12:257-65
   PubMed Web of Science ®Google Scholar
• Siewert M, Dressman J, Brown CK, et al. FIP/AAPS guidelines to dissolution/in vitro release testing of novel/special dosage forms. AAPS PharmSciTech 2003;4:43-52
   Google Scholar
• Al-Zoubi N, Koundourellis JE, Malamataris S. FT-IR and Raman spectroscopic methods for identification and quantitation of orthorhombic and monoclinic paracetamol in powder mixes. J Pharm Biomed Anal 2002;29:459-67
   PubMed Web of Science ®Google Scholar
• Perlovich GL, Volkova TV, Bauer-Brandl A. Polymorphism of paracetamol-relative stability of the monoclinic and orthorhombic phase revisited by sublimation and solution calorimetry. J Therm Anal Calorim 2007;89:767-74
   Web of Science ®Google Scholar
• Cima Labs, Inc. Effervescent dosage form with microparticles. US5178878; 1993
   Google Scholar
• Cima Labs, Inc. Rapidly dissolving robust dosage form. US6024981; 2000
   Google Scholar
• Cima Labs, Inc. Pediatric effervescent dosage form. US5223264; 1993
   Google Scholar
• Cima Labs, Inc. Taste masking microparticles for oral dosage forms. US5607697; 1997
   Google Scholar
• Cima Labs, Inc. Taste masking rapid release system. US6740341; 2004
   Google Scholar
• Ethypharm, Inc. Process for manufacturing coated granules with masked taste and immediate release of the active principle. US6660382; 2003
   Google Scholar
• Ethypharm, Inc. Particles with granulated crystalline Ibuprofen. US6951657; 2005
   Google Scholar
• Gattefosse ETS SA. Tablet for crunching with masked taste and instant release of active principle and method for making same. WO0024385; 2000
   Google Scholar
• Gattefosse ETS SA. Method for coating solid particles with a thermofusible agent and resulting coated solid particles. WO0207706; 2002
   Google Scholar
• Gattefosse ETS SA. Method for preparing a pharmaceutical composition with modified release of the active principle comprising a matrix. WO9814176; 2000
   Google Scholar
• Eurand America, Inc. Effervescent microcapsules. US5639475; 1997
   Google Scholar
• Eurand America, Inc. Effervescent microcapsules. US5709886; 1998
   Google Scholar
• Eurand America, Inc. Taste-masked microcapsule compositions and methods of manufacture. US6139865; 2000
   Google Scholar
• Eurand Pharmaceuticals Ltd. Taste masked pharmaceutical compositions prepared by coacervation. WO2006055142; 2006
   Google Scholar
• Guo X, Chang RK, Hussain MA. Ion-exchange resins as drug delivery carriers. J Pharm Sci 2009;98:3886-902
   PubMed Web of Science ®Google Scholar
• Fertin Pharma AS. Stable medicated chewing gum comprising cyclodextrin inclusion complex. WO2009006898; 2009
   Google Scholar
• Loftsson T, Duchene D. Cyclodextrins and their pharmaceutical applications. Int J Pharm 2007;329:1-11
   PubMed Web of Science ®Google Scholar
• McNeil Consumer Products Co. Chewable medicament tablet containing means for taste masking. US4851226; 1989
   Google Scholar
• McNeil Consumer Products Co. Taste masking and sustained release coatings for pharmaceuticals. US5075114; 1991
   Google Scholar
• Elan Corp. P.L.C. Controlled release powder and process for its preparation. US4952402; 1990
   Google Scholar
• Fuisz Technologies Ltd. Process and apparatus for making rapidly dissolving dosage units and product there from. US5622719; 1997
   Google Scholar