169
Views
29
CrossRef citations to date
0
Altmetric
Drug Profile

Transdermal buprenorphine in the treatment of chronic pain

Pages 315-323 | Published online: 10 Jan 2014

References

  • Staats PS, Johnson RE. New perspectives on the pharmacology of opioids and their use in chronic pain. Prog. Anesthesiol. 16, 235–249 (2002).
  • Grossman SA, Benedetti C, Brock C et al. NCCN Practice Guidelines for Cancer Pain. NCCN Proceedings14, 135–150 (2000).
  • Ferrell B, Casarett D, Epplin J et al. The management of persistent pain in older persons. J. Am. Geriatr. Soc. 50(Suppl. 6), S205–S224 (2002).
  • Welsh J, Copp K, Dunne J et al. Control of pain in patients with cancer. A national clinical guideline. Edinburgh (Scotland). Scottish Intercollegiate Guidelines Network, 2000, 1–6 (1996).
  • Masson AHB. Sublingual buprenorphine versus oral dihydrocodeine in post-operative pain. J. Int. Med. Res.9, 506–510 (1981).
  • Hanks GW. The clinical usefulness of agonist-antagonist opioid analgesics in chronic pain. Drug Alcohol Depend. 20, 339–46 (1987).
  • Heel RC, Brogden RN, Speight TM, Avery GS. Buprenorphine: a review of its pharmacological properties and therapeutic efficacy. Drugs17, 81–119 (1979).
  • Budd K. Buprenorphine and the transdermal system: the ideal match in pain management. Int. J. Clin. Pract.133(Suppl.), 9–14 (2003).
  • Allan L, Hays H, Jensen NH et al. Randomised crossover trial of transdermal fentanyl and sustained release oral morphine for treating chronic non-cancer pain. Br. Med. J. 322, 1154–1158 (2001).
  • Payne R, Mathias SD, Pasta DJ et al. Quality of life and cancer pain: satisfaction and side effects with transdermal fentanyl versus oral morphine. J. Clin. Oncol. 16, 1588–1593 (1998).
  • Grünenthal GmbH. Transtec Scientific Monograph. (2002).
  • Martin WR, Eades CG, Thompson JA et al. The effects of morphine- and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog. J. Pharmacol. Exp. Ther. 197, 517–532 (1976).
  • Lewis JW. Buprenorphine. Drug Alcohol. Depend. 14, 363–372 (1985).
  • Cowan A, Doxey JC, Harry EJR. The animal pharmacology of buprenorphine, an oripavine analgesic agent. Br. J. Pharmacol. 60, 547–554 (1977).
  • Leander JD. Buprenorphine is a potent κ-opioid receptor antagonist in pigeons and mice. Eur. J. Pharmacol. 151, 457–461 (1988).
  • Cowan A, Lewis JW, Macfarlane IR. Agonist and antagonist properties of buprenorphine, a new antinociceptive agent. Br. J. Pharmacol. 60, 537–545 (1977).
  • Evans HC, Easthope SE. Transdermal buprenorphine. Drugs 63, 1999–2010 (2003).
  • Dunn JE, Herz A. In vivo receptor binding of the opiate partial agonist, buprenorphine, correlated with its agonistic and antagonistic actions. Br. J. Pharmacol. 74, 627–633 (1981).
  • Tyers MB. A classification of opiate receptors that mediate antinociception in animals. Br. J. Pharmacol.69, 503–512 (1980).
  • Budd K. High-dose buprenorphine for postoperative analgesia. Anaesthesia36, 900–903 (1981).
  • Walsh SL, Preston KL, Stitzer ML, Cone EJ, Bigelow GE. Clinical pharmacology of buprenorphine: ceiling effects at high doses. Clin. Pharmacol. Ther. 55, 569–580 (1994).
  • Dahan A, Bijl H, Romberg R et al. Full reversal of buprenorphine induced respiratory depression by naloxone. Eur. J. Anaesthesiology (2005) (In Press).
  • Tegeder I, Lotsch J, Geisslinger G. Pharmacokinetics of opioids in liver disease. Clin. Pharmacokinet. 37, 17–40 (1999).
  • Budd K. Buprenorphine: a review. Evidence Based Med. Prac. 1–24 (2002).
  • Böhme K. Buprenorphine in a transdermal therapeutic system – a new option. Clin. Rheumatol. 21(Suppl. 1), S13–S16 (2002).
  • Data on file. Grünenthal. (2003).
  • Sittl R. Buprenorphine transdermal patch: clinical expert report. Grünenthal, GmbH, Germany (2000).
  • Rance MJ, Shillingford JS. The role of the gut in the metabolism of strong analgesics. Biochem. Pharmacol.25, 735–741 (1976).
  • Rance MJ, Shillingford JS. The metabolism of phenolic opiates by rat intestine. Xenobiotica 7(9), 529–536 (1997).
  • Iribarne C, Picart D, Dreano Y, Bail JP, Berthou F. Involvement of cytochrome P450 3A4 in N-dealkylation of buprenorphine in human liver microsomes. Life Sci. 60, 1953–1964 (1977).
  • Ohtani M, Kotaki H, Nishitateno K. Kinetics of resoiratory depression in rats induced by buprenorphine and its metabolite, norbuprenrophine. J. Pharmacol. Exp. Ther. 281(1), 428–433 (1984).
  • Filitz J, Sittl R, Griessinger N, Likar R, Koppert W. Pharmacokinetics of transdermal buprenorphine (Transtec®) in patients with renal insufficiency. Poster presented at EAPC in Aachen. J. Pain Symptom Manage. (2005) (In Press).
  • McQuay HJ, Moore RA, Bullingham RES. Buprenorphine kinetics. In: Advancesin Pain Research and Therapy. Foley KM, Inturrisi CE (Eds). Raven Press, NY, USA, 271–278 (1986).
  • Moore RA, Sear JW, Baldwin D et al. Morphine kinetics during and after renal transplantation in man. Clin. Pharmacol. Ther. 35, 641–645 (1997).
  • Böhme K. Buprenorphine transdermal system (TDS) (delivery rates 35/52.5/70 µg/h) in comparison to sublingual buprenorphine in chronic pain patients. 1st Congress of the Research Network of the European Association for Palliative Care, December 7–9, Berlin, Germany (2000).
  • Böhme K, Likar R. Efficacy and tolerability of a new opioid analgesic formulation, buprenorphine transdermal therapeutic system (TDS), in the treatment of patients with chronic pain. A randomized, double-blind, placebo-controlled study. Pain Clinic 15, 193–202 (2003).
  • Sittl R, Griessinger N, Likar R. Analgesic efficacy and tolerability of transdermal buprenorphine in patients with inadequately controlled chronic pain related to cancer and other disorders: a multicenter, randomized, double-blind, placebo-controlled trial. Clin. Ther. 25, 150–68 (2003).
  • Sorge J, Sittl R. Transdermal buprenorphine in the treatment of chronic pain: results of a Phase III, multicenter, randomized, double-blind, placebo-controlled study. Clin. Ther. 26(11), 1808–1820 (2004).
  • Radbruch L. Buprenorphine TDS: use in daily practice, benefits for patients. Int. J. Clin. Pract. (Suppl. 13), 19–22 (2003).
  • Kopp M. Buprenorphine transdermal system (TDS) in an open long-term study with chronic pain patients. 1st Congress of the Research Network of the European Association for Palliative Care, December 7–9, Berlin, Germany (2000).
  • Vielvoye-Kerkmeer APE. Long-term treatment with buprenorphine TDS in patients with chronic pain. Eur. J. Palliat. Care 10(Suppl. 1), 17–19 (2003).
  • Liedgens H, Ritzdorf I. Efficacy and safety of transdermal buprenorphine demonstrated in a large chronic pain population. Schmerz 17(Suppl. 1), S104–S105 (2003).
  • Twycross RG. Opioid analgesics in cancer pain: current practice and controversies. Cancer Surveys 7, 29–53 (1988).
  • Atkinson RE, Schofield P, Mellor P. The efficacy in sequential use of buprenorphine and morphine in advanced cancer pain. In: Opioids in the Treatment of Cancer Pain. Doyle D (Ed.). Royal Society of Medicine Services, International Congress and Symposium Series. 146, 81–87 (2004).
  • Camba MA, The Opioid Study Group of the Spanish Pain Society. Transdermal buprenorphine for the management of nociceptive chronic pain. Rev. Soc. Esp. Dolor. (Suppl V), 22–30 (1990).
  • Rodriguez-Lopez MJ, The Opioid Study Group of the Spanish Pain Society. Transdermal buprenorphine in the management of neuropathic pain. Rev. Soc. Esp. Dolor. (Suppl. V), 11–21 (2004).
  • Muriel C, The Opioid Study Group of the Spanish Pain Society. Assessment of buprenorphine transdermal patch in patients with cancer pain. Rev. Soc. Esp. Dolor. (Suppl. V), 41–48 (2004).
  • Barutell C de, The Opioid Study Group of the Spanish Pain Society. Buprenorphine and tramadol. Rev. Soc. Esp. Dolor. (Suppl. V), 31–40 (2004).
  • Gonzalez-EscaladaJR, The Opioid Study Group of the Spanish Pain Society. Use of buprenorphine and oral morphine in patients with chronic pain. Rev Soc Esp Dolor (Suppl. V), 3–10 (2004).
  • Gal TJ. Naloxone reversal of buprenorphine-induced respiratory depression. Clin. Pharmacol. Ther. 45, 66–71 (1989).
  • Knape JTA. Early respiratory depression resistant to naloxone following epidural buprenorphine. Anesthesiology 64, 382–384 (1986).
  • Haddox JD, Joranson D, Angarola RT et al. The use of opioids for the treatment of chronic pain: a consensus statement from American Academy of Pain Medicine and American Pain Society www.ampainsoc.org/cgi-bin/print/print.pl (Accessed April 2005)
  • World Health Organization. World Health Organization’s pain relief ladder. www.who.int/cancer/palliative/ painladder/en/ (Accessed April 2005)

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.