81
Views
2
CrossRef citations to date
0
Altmetric
Original Research

Synthesis, antimicrobial, and antiproliferative activities of substituted phenylfuranylnicotinamidines

, &
Pages 1133-1146 | Published online: 11 Mar 2016

References

  • KennedyBO’ConnorBKornBGibbonsNO’ConnorTKeaneJMulti-drug resistant tuberculosis: experiences of two tertiary referral centresIr Med J2011104618218522111396
  • KuttyNTreating children without antibiotics in primary healthcareOman Med J201126530330522125722
  • LevySBFactors impacting on the problem of antibiotic resistanceJ Antimicrob Chemother2002491253011751763
  • LindMJPrinciples of cytotoxic chemotherapyMedicine20083611923
  • SummersLAThe Bipyridinium HerbicidesLondonAcademic Press1980
  • World Health OrganizationWHO Model List of Essential MedicinesGenevaWorld Health Organization102013 Retrieved April 22, 2014. Available from: http://apps.who.int/iris/bitstream/10665/112738/1/9789240692671_eng.pdfAccessed February 18, 2016
  • LibmanMDMillerMARichardsGKAntistaphylococcal activity of pentamidineAntimicrob Agents Chemother1990349179517962285292
  • WerbovetzKDiamidines as antitrypanosomal, antileishmanial and antimalarial agentsCurr Opin Investig Drugs200672147157
  • PathakMKDhawanDLindnerDJBordenECFarverCYiTPen-tamidine is an inhibitor of PRL phosphatases with anticancer activityMol Cancer Ther20021141255126412516958
  • SmithJStewartBJGlaysherSThe effect of pentamidine on melanomaAnticancer Drugs201021218118519966562
  • LansiauxATaniousFMishalZDistribution of furamidine analogues in tumor cells targeting of the nucleus or mitochondria depending on the amidine substitutionCancer Res200262247219722912499262
  • AntonySMarchandCStephenAGNovel high-throughput electrochemiluminescent assay for identification of human tyrosyl-DNA phosphodiesterase (Tdp1) inhibitors and characterization of furamidine (NSC 305831) as an inhibitor of Tdp1Nucleic Acids Res200735134474448417576665
  • IsmailMABrunREasterbrookJDTaniousFAWilsonWDBoykinDWSynthesis and antiprotozoal activity of aza-analogues of furamidineJ Med Chem200346224761476914561095
  • WenzlerTBoykinDWIsmailMAHallJETidwellRRBrunRNew treatment option for second-stage African sleeping sickness: in vitro and in vivo efficacy of aza analogs of DB289Antimicrob Agents Chemother200953104185419219620327
  • ThuitaJKWolfKKMurillaGASafety, pharmacokinetic, and efficacy studies of oral DB868 in a first stage vervet monkey model of human African trypanosomiasisPLoS Negl Trop Dis201376e223023755309
  • WenzlerTYangSBraissantOBoykinDWBrunRWangMZPharmacokinetics, Trypanosoma brucei gambiense, efficacy, and time of drug action of DB829, a preclinical candidate for treatment of second-stage human African trypanosomiasisAntimicrob Agents Chemother201357115330534323959303
  • ThuitaJKWolfKKMurillaGAChemotherapy of second stage human African trypanosomiasis: comparison between the parenteral diamidine DB829 and its oral prodrug DB868 in vervet monkeysPLoS Negl Trop Dis201592e000340925654243
  • YoussefMMAl-OmairMAIsmailMASynthesis, DNA affinity, and antimicrobial activity of 4-substituted phenyl-2,2′-bichalcophenes and aza-analoguesMed Chem Res20122140744082
  • HussinWAIsmailMAEl-SayedWMNovel 4-substituted phenyl-2,2′-bichalcophenes and aza-analogues as antibacterial agents: a structural activity relationshipDrug Des Devel Ther20137185193
  • El-SayedWMHussinWAIsmailMAEfficacy of two novel 2,2′-bifurans to inhibit methicillin-resistant Staphylococcus aureus infection in male mice in comparison to vancomycinDrug Des Devel Ther20126279287
  • HussinWAIsmailMAAlzahraniAMEl-SayedWMEvaluation of the biological activity of novel monocationic fluoroaryl-2,2′- bichalcophenes and their analoguesDrug Des Devel Ther20148963972
  • El-SayedWMHussinWAAntimutagenic and antioxidant activity of novel 4-substituted phenyl-2,2′-bichalcophenes and aza-analogsDrug Des Devel Ther201377381
  • IsmailMAArafaRKYoussefMMEl-SayedWMAnticancer, antioxidant activities and DNA affinity of novel monocationic bithiophenes and analoguesDrug Des Devel Ther2014816591672
  • BauerWKirbyWMSherrisJCTurckMJAntibiotic susceptibility testing by a standardized single disk methodClinic Pathol1966454493496
  • YoussefMMMahmoudAAAl-FaiyzYSAntimicrobial and antioxidant activities of Artemisia abyssinica extracts and DNA degradation effectsAsian J Biochem20151013141
  • CLSI/NCCLSMethods for Dilution Antimicrobial Susceptibility Tests for Bacteria That Grow Aerobically, Approved Standard7th edWayne, PACLSI2006
  • SkehanPStorengRScudieroDNew colorimetric cytotoxicity assay for anticancer-drug screeningJ Natl Cancer Inst19908213110711122359136
  • McCaffreyTAAgarwalLAWekslerBBA rapid fluorometric DNA assay for the measurement of cell density and proliferation in vitroIn Vitro Cell Dev Biol19882432472523280545
  • MonksAScudieroDSkehanPFeasibility of a high-flux anticancer drug screen using a diverse panel of cultured human tumor cell linesJ Natl Cancer Inst199183117577662041050
  • SayedARYoussefMMAl-FaiyzYSSynthesis, characterization, and biological evaluation of novel thiadiazoline sulfonamides and metal complexesJ Appl Sci2015156884893
  • SambrookJFritschEFManiatisTMolecular Cloning: A Laboratory ManualCold Spring Harbor, NYCold Spring Harbor Laboratory Press1989
  • BridgesSMSalinMLDistribution of iron-containing superoxide dismutase in vascular plantsPlant Physiol198168227527816661901
  • Al-OmairMASayedARYoussefMMSynthesis of novel triazoles, tetrazine, thiadiazoles and their biological activitiesMolecules2015202591261025648599
  • GreenLCWagnerDAGlogowskiJSkipperPLWishnokJSTannenbaumSRAnalysis of nitrate, nitrite, and [15N] nitrate in biological fluidsAnal Biochem198212611311387181105
  • SreejayanNRaoMNANitric oxide scavenging by curcuminoidsJ Pharm Pharmacol19974911051079120760
  • CrayJABellANWBhagannaPMswakaAYTimsonDJHallsworthJEHydrophobic substances induce water stress in microbial cellsMicrob Biotechnol2013645349223336673
  • CrayJAStevensonABallPChaotropicity: a key factor in product tolerance of biofuel-producing microorganismsCurr Opin Biotechnol20153322825925841213
  • OyaizuMStudies on product of browning reaction prepared from glucose amineJpn J Nutr198644307315
  • MoncadaSPalmerRMHiggsEANitric oxide: physiology, pathophysiology, and pharmacologyPharmacol Rev19914321091421852778