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Original Research

Synthesis and evaluation of ortho-[18F] fluorocelecoxib for COX-2 cholangiocarcinoma imaging

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Pages 1467-1478 | Published online: 24 May 2018

References

  • HayashiNYamamotoHHiraokaNDifferential expression of cyclooxygenase-2 (COX-2) in human bile duct epithelial cells and bile duct neoplasmHepatology200134463865011584358
  • SiricaAELaiGHZhangZCBiliary cancer growth factor pathways, cyclo-oxygenase-2 and potential therapeutic strategiesJ Gastroenterol Hepatol200116436337211357901
  • SiricaAELaiGHEndoKZhangZCYoonBICyclooxygenase-2 and ERBB-2 in cholangiocarcinoma: potential therapeutic targetsSemin Liver Dis200222330331312360423
  • MarksEIYeeNSMolecular genetics and targeted therapeutics in biliary tract carcinomaWorld J Gastroenterol20162241335134726819503
  • BridgewaterJGallePRKhanSAGuidelines for the diagnosis and management of intrahepatic cholangiocarcinomaJ Hepatol20146061268128924681130
  • Taylor-RobinsonSDToledanoMBAroraSIncrease in mortality rates from intrahepatic cholangiocarcinoma in England and Wales 1968–1998Gut200148681682011358902
  • KhanSATaylor-RobinsonSDToledanoMBBeckAElliottPThomasHCChanging international trends in mortality rates for liver, biliary and pancreatic tumoursJ Hepatol200237680681312445422
  • CasavillaFAMarshJWIwatsukiSHepatic resection and transplantation for peripheral cholangiocarcinomaJ Am Coll Surg199718554294369358085
  • OhtsukaMItoHKimuraFResults of surgical treatment for intrahepatic cholangiocarcinoma and clinicopathological factors influencing survivalBr J Surg200289121525153112445060
  • SmithWLUradeYJakobssonPJEnzymes of the cyclooxygenase pathways of prostanoid biosynthesisChem Rev2011111105821586521942677
  • KhanSADavidsonBRGoldinRDGuidelines for the diagnosis and treatment of cholangiocarcinoma: an updateGut201261121657166922895392
  • SiricaAECholangiocarcinoma: molecular targeting strategies for chemoprevention and therapyHepatology200541151515690474
  • BerthiaumeEPWandsJThe molecular pathogenesis of cholangiocarcinomaSemin Liver Dis200424212713715192786
  • BurrNETalboysRJSavvaSAspirin may prevent cholangiocarcinoma: a case-control study from the United KingdomDigest Dis Sci20145971567157224535250
  • JendrossekVTargeting apoptosis pathways by Celecoxib in cancerCancer Lett2013332231332421345578
  • PreshlockSTredwellMGouverneurVF-18-labeling of arenes and heteroarenes for applications in positron emission tomographyChem Rev2016116271976626751274
  • PrabhakaranJUnderwoodMDParseyRVSynthesis and in vivo evaluation of F-18 -4- 5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl benzene sulfonamide as a PET imaging probe for COX-2 expressionBioorg Med Chem20071541802180717166726
  • ToyokuniTKumarJSDWalshJCSynthesis of 4-(5-F-18 fluoromethyl-3-phenylisoxazol-4-yl)-benzenesulfonamide, a new F-18 fluorinated analogue of valdecoxib, as a potential radiotracer for imaging cyclooxygenase-2 with positron emission tomographyBioorg Med Chem Lett200515214699470216153836
  • UddinMJCrewsBCGhebreselasieKFluorinated COX-2 Inhibitors as Agents in PET Imaging of Inflammation and CancerCancer Prev Res201141015361545
  • RieseJHoffTNordhoffADewittDLReschKKaeverVTransient expression of prostaglandin endoperoxide synthase-2 during mouse macrophage activationJ Leukoc Biol19945544764828145018
  • McCarthyTJSheriffAUGranetoMJTalleyJJWelchMJRadio-synthesis, in vitro validation, and in vivo evaluation of F-18-labeled COX-1 and COX-2 inhibitorsJ Nucl Med200243111712411801714
  • de VriesEFJvan WaardeABuursmaARVaalburgWSynthesis and in vivo evaluation of F-18-desbromo-DuP-697 as a PET tracer for cyclooxygenase-2 expressionJ Nucl Med200344101700170614530489
  • RiniBIWeinbergVDunlapSMaximal COX-2 immunostaining and clinical response to celecoxib and interferon alpha therapy in metastatic renal cell carcinomaCancer2006106356657516369983
  • FabiAMetroGPapaldoPImpact of celecoxib on capecitabine tolerability and activity in pretreated metastatic breast cancer: results of a Phase II study with biomarker evaluationCancer Chemother Pharmacol200862471772518071704
  • JewettDMPotockiJFEhrenkauferREA gas solid-phase microchemical method for the synthesis of acetyl hypofluoriteJ Fluorine Chem1984244477484
  • BiavaMPorrettaGCPoceGCyclooxygenase-2 inhibitors. 1,5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/cyclooxygenase-1 selectivityJ Med Chem200750225403541117915854
  • HusainAAhmadAAlamMMAjmalMAhujaPFenbufen based 3- 5-(substituted aryl)-1,3,4-oxadiazol-2-yl -1-(biphenyl-4-yl)propan-1-ones as safer antiinflammatory and analgesic agentsEur J Med Chem20094493798380419457595
  • HoodWFGierseJKIsaksonPCCharacterization of celecoxib and valdecoxib binding to cyclooxygenaseMol Pharmacol200363487087712644588
  • GierseJKZhangYHoodWFValdecoxib: assessment of cyclooxygenase-2 potency and selectivityJ Pharmacol Exp Ther200531231206121215494548
  • HuangHLYehCNLeeWYI-123 Iodooctyl fenbufen amide as a SPECT tracer for imaging tumors that over-express COX enzymesBiomaterials201334133355336523384791
  • HuangHLHuangYCLeeWYYehCNLinKJYuCSF-18-gluta-thione conjugate as a PET tracer for imaging tumors that overexpress L-PGDS enzymePLoS One20149814
  • YehCNChangCWChungYHSynthesis and characterization of boron fenbufen and its F-18 labeled homolog for boron neutron capture therapy of COX-2 overexpressed cholangiocarcinomaEur J Pharm Sci201710721722928728977
  • YehCNLinKJChenTWCharacterization of a novel rat cholangiocarcinoma cell culture model-CGCCAWorld J Gastroenterol201117242924293221734803
  • ChenSFWuCHLeeYMCaveolin-1 interacts with derlin-1 and promotes ubiquitination and degradation of cyclooxygenase-2 via collaboration with p97 complexJ Biol Chem201328846334623346924089527
  • YehCNMaitraALeeKFJanYYChenMFThioacetamide-induced intestinal-type cholangiocarcinoma in rat: an animal model recapitulating the multi-stage progression of human cholangiocarcinomaCarcinogenesis200425463163614656942
  • MonakhovNKNeistadtELShavlovskilMMShvartsmanALNeifakhSAPhysicochemical properties and isoenzyme composition of hexokinase from normal and malignant human tissuesJ Natl Cancer Inst19786112734276635
  • LiZBCaiWBCaoQZ64Cu-labeled tetrameric and octameric RGD peptides for small-animal PET of tumor alpha(v)beta(3) integrin expressionJ Nucl Med20074871162117117574975
  • JacobsonOWeissIDKiesewetterDOFarberJMChenXYPET of tumor CXCR4 expression with 4-F-18-T140J Nucl Med201051111796180420956475
  • TietzOWuestMMarshallAPET imaging of cyclooxygenase-2 (COX-2) in a pre-clinical colorectal cancer modelEJNMMI Res201661126860293
  • WeberACasiniAHeineAUnexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: new pharmacological opportunities due to related binding site recognitionJ Med Chem200447355055714736236
  • ChungYHHsuPHHuangCWEvaluation of prognostic integrin alpha 2 beta 1 PET tracer and concurrent targeting delivery using focused ultrasound for brain glioma detectionMol Pharm201411113904391425153169