References
- Albert A., Gledhil W. Improved synthesis of aminoacridines. IV. Substituted 9-aminoacridines. J. Soc. Chem. Ind. (1945); 64: 169
- Heilbronn E. Inhibition of cholinesterases by tetrahydro-aminoacridine. Acta Chem. Scand. (1961); 15: 1386
- Shaw F. H., Bendy G. A. The pharmacology of some new anticholinesterases. Aust. J. Exp. Biol. Med. Sci. (1953); 31: 573
- Shaw F. H., Bently G. A. Morphine antagonism. Aust. J. Exp. Biol. Med. Sci. (1955); 33: 143
- Kaul P. N. Enzyme inhibition by tetrahydroaminoacridine. J. Pharm. Pharmacol. (1962); 14: 243
- Summers W. K., Kaufman K. R., Altman F., Jr., Fisher J. M. THA: A review of the literature and its use in treatment of five overdose patients. Clin. Toxicol. (1980); 16: 268
- Giacobini E., Becker R. “Current Research in Alzheimer Therapy”. Taylor and Francis, New York 1988
- Summers W. K., Majovski L. V., Marsh G. M., Tachiki K., Kling A. Oral tetrahydroaminoacridine in long-term treatment of senile dementia, Alzheimer type. N. Engl. J. Med. (1986); 315: 1241
- Amshey J. W., Steinberg G. M., Miller R. B. A screening program for selective inhibitors of the phosphorylation of acetylcholinesterase. Department of the Army, Aberdeen Proving Ground, MD (1973), Edgewood Arsenal Technical Report, EB-TR-73014
- Bajgar J, Potocka J, Fusek J., Hrdina V. Some possibilities of protection against acetylcholinesterase inhibition by organophosphates in vivo. Sb. Ved. Pr. Lek Fak Univ. Karlovy Hradci Kralove (1984); 27: 425
- Galli A, Mori F. Effectiveness of l,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication. Arch. Toxicol. (1991); 65: 330
- De La Hoz D., Doctor B, Rolston J. S., Rush R. S, Wolfe A D. A simplified procedure for the purification of large quantities of fetal bovine serum acetylcholinesterase. Life Sci. (1986); 39: 195
- Ellman G. L, Courtney K. D., Andres V., Jr., Featherstone R. M. A new and rapid colorimetric determination of acetylcholinesterase activity. Biochem. Pharm. (1961); 7: 88
- Keijer J H, Wolring G. Z., DeJong LP. A. Effect of pH, temperature and ionic strength on the aging of phosphonylated cholinesterases. Biochem. Biophys. Acta (1974); 334: 146
- Finney D J. Probit Analysis. Cambridge University Press, Cambridge 1971
- Bliss C. I. Fisher's Exact Test for 2 x 2 Tables. “Statistics in Biology”. McGraw-Hill, New York (1967); Vol I: 63
- Sanberg P R, Hagenmeyer S. H.M., Henault A. Automated measurement of multivariant locomotor behavior in rodents. Neurobehav. Tox. Teratol. (1985); 7: 87
- Number Cruncher Statistical System. J.L. Hintze, Kaysville, UT (1987), version 5.01
- Kuribara H, Haraguchi H., Tadokoro S. Comparison between discrete lever press and shuttle avoidance responses in mice: Acquisition process and psychoactive drugs. Jap. J. Pharmacol. (1985); 38: 141
- Romano J. A, Mterry R., MMurrow L., Mays M. Z. Protection from lethality and behavioral incapacitation resulting from intoxication by soman (pinacolyl methylphosphono fluoridate) and treatment with atropine sulfate and 2-PAM chloride in the guinea pig, caviaprocellus. Drug Chem. Tox. (1991); 14: 21
- Nielsen A. J, Mena E. E, Williams I. H., Noccerini M R, Liston D. Correlation of brain levels of 9-amino-l,2,3,4-tetrahydroacridine in vitro. Eur. J. Pharmacol. (1989); 173: 53
- Natori K., Okazaki Y., Irie T., Katstube J. Pharmacological and biochemical assessment of SM-10888, a novel cholinesterase inhibitor. Jap. J. Pharmac (1990); 53: 145
- Hunter A. J., Murray T. K., Jones J. A., Cross A. J., Green A. R. The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro. Br. J. Pharmacol. (1989); 98: 79
- Marquis J. K. Pharmacological significance of acetylcholinesterase inhibition by tetrahydroaminoacridine. Biochem. Pharm. (1990); 40: 1071
- Patoč ka J., Bajgar J., Bielavsky J., Fusek J. Kinetics of inhibition of cholinesterases by 1,2,3,4-tetrahydroaminoacridine in vitro. Coll. Czech. Chem. Commun. (1976); 41: 816
- Dawson R. M. Reversibility of the inhibition of acetylcholinesterase by tacrine. Neurosci. Letters (1990); 118: 85
- Potoč ka J., Bajgar J. The reactivation of o-isoproplymethyl-phosphonylated acetylcholinesterase and its modification by some non-acylating ligands. Sb. Ved. Pr. Lek. Fak. Univ. Karlovy Hradci Kralove (1984); 27: 477
- Wu C. S., Yang J. T. Tacrine protection of acetylcholinesterase form inactivation by diisopropylfluorophosphate: A circular dichroism study. Mol. Pharmacol. (1989); 35: 85
- Steinberg G. M., Mednick M. L., Maddox J., Rice R., Cramer J. A hydrophobic binding site in acetylcholinesterase. J. Med. Chem. (1975); 18: 1056
- Freeman S. E., Dawson R. M. Tacrine: A pharmacological review. Prog. Neurobiol. (1991); 36: 257
- Dawson R. M. Tacrine slows the rate of ageing of sarin-inhibited acetylcholinesterase. Neurosci. Letters (1989); 100: 227
- Deyi X., Linxiu W., Shuqiu P. The inhibition and protection of cholinesterase by physostigmine and pyridostigmine against soman poisoning in vivo. Fundam. Appl. Toxicol. (1981); 1: 217
- Departments of the Army, the Navy, and the Air Force. “Treatment of Chemical Agent Casualties and Conventional Military Chemical Injuries”. U.S. Government Printing Office, Washington, DC (1990), Army FM 8–285