Polyester-based microparticles of different hydrophobicity: the patterns of lipophilic drug entrapment and release

References

• Albertsson AC, Srivastava RK. Recent developments in enzyme-catalyzed ring-opening polymerization. Adv Drug Deliv Rev Rev, 2008;60(9):1077–93.
   PubMed Web of Science ®Google Scholar
• Biggs DL, Lengsfeld CS, Hybertson BM, Ng KY, Manning MC, Randolph TW. In vitro and in vivo evaluation of the effects of PLA microparticle crystallinity on cellular response. J Control Release, 2003;92(1–2):147–61.
   PubMed Web of Science ®Google Scholar
• Choi JS, Seo K, Yoo JW. Recent advances in PLGA particulate systems for drug delivery. J Pharma Investig, 2012;42(3):155–63.
   Google Scholar
• Chung TW, Huang YY, Tsai YL, Liu YZ. Effects of solvent evaporation rate on the properties of protein-loaded PLLA and PDLLA microspheres fabricated by emulsion-solvent evaporation process. J Microencapsulation, 2002;19(4):463–71.
   PubMed Web of Science ®Google Scholar
• Cohen LJ. Risperidone. Pharmacotherapy, 1994;14(3):253–65.
   PubMed Web of Science ®Google Scholar
• Costa P, Sousa Lobo JM. Modeling and comparison of dissolution profiles. Eur J Pharm Sci, 2001;13(2):123–33.
   PubMed Web of Science ®Google Scholar
• Dalmoro A, Barba AA, Lamberti M, Mazzeo M, Venditto V, Lamberti G. Random l-lactide/ɛ-caprolactone copolymers as drug delivery materials. J Materials Sci, 2014;49(17):5986–96.
   Web of Science ®Google Scholar
• Danhier F, Ansorena E, Silva JM, Coco R, Le Breton A, Préat V. PLGA-based nanoparticles: An overview of biomedical applications. J Control Release, 2012;161(2):505–22.
   PubMed Web of Science ®Google Scholar
• du Noüy PL. Spontaneous decrease of the surface tension of serum. I. J Exp Med, 1922;35(4):575–97.
   Google Scholar
• Dunne M, Corrigan OI, Ramtoola Z. Influence of particle size and dissolution conditions on the degradation properties of polylactide-co-glycolide particles. Biomaterials, 2000;21(16):1659–68.
   PubMed Web of Science ®Google Scholar
• Ensign LM, Cone R, Hanes J. Oral drug delivery with polymeric nanoparticles: The gastrointestinal mucus barriers. Adv Drug Deliv Rev Rev, 2012;64(6):557–70.
   PubMed Web of Science ®Google Scholar
• Frank A, Rath SK, Venkatraman SS. Controlled release from bioerodible polymers: Effect of drug type and polymer composition. J Control Release, 2005;102(2):333–44.
   PubMed Web of Science ®Google Scholar
• Frelichowska J, Bolzinger MA, Pelletier J, Valour JP, Chevalier Y. Topical delivery of lipophilic drugs from o/w Pickering emulsions. Int J Pharm, 2009;371(1–2):56–63.
   PubMed Web of Science ®Google Scholar
• Fu X, Ping Q, Gao Y. Effects of formulation factors on encapsulation efficiency and release behaviour in vitro of huperzine A-PLGA microspheres. J Microencapsulation, 2005;22(7):705–14.
   PubMed Web of Science ®Google Scholar
• Haley B, Frenkel E. Nanoparticles for drug delivery in cancer treatment. Urologic Oncology, 2008;26(1):57–64.
   PubMed Web of Science ®Google Scholar
• Izumikawa S, Yoshioka S, Aso Y, Takeda Y. Preparation of poly(L-lactide) microspheres of different crystalline morphology and effect of crystalline morphology on drug release rate. J Controlled Release, 1991;15:133–40.
   Web of Science ®Google Scholar
• Karavelidis V, Karavelidis V, Giliopoulos D, Karavas E, Bikiaris D. Nanoencapsulation of a water soluble drug in biocompatible polyesters. Effect of polyesters melting point and glass transition temperature on drug release behavior. European J Pharmaceutical Sci, 2010;41(5):636–43.
   PubMed Web of Science ®Google Scholar
• Kim M, Pack DW. Rhodamine-123 staining in hematopoietic stem cells of young mice indicates mitochondrial activation rather than dye efflux. Blood, 1998;91(11):4106–17.
   PubMed Web of Science ®Google Scholar
• Korzhikov V, Gusevskaya KV, Litvinchuk EN, Vlakh EG, Tennikova TB. Enzyme-mediated ring-opening polymerization of pentadecalactone to obtain biodegradable polymer for fabrication of scaffolds for bone tissue engineering. Int J Polymer Sci, 2013;2013:476748.
   Web of Science ®Google Scholar
• Kowalski A, Duda A, Penczek S. Mechanism of cyclic ester polymerization initiated with tin(II) octoate. 2. macromolecules fitted with tin(II) alkoxide species observed directly in MALDI − TOF spectra. Macromolecules, 2000;33(3):689–95.
   Web of Science ®Google Scholar
• Kuentz M. Lipid-based formulations for oral delivery of lipophilic drugs. Drug Discov Today Technol, 2012;9(2):e97–104.
   Google Scholar
• Kumar A, et al. Efficient ring-opening polymerization and copolymerization of -Caprolactone and ω-pentadecalactone catalyzed by Candida antartica lipase B. Macromolcules, 2000;33:6303–9.
   Web of Science ®Google Scholar
• Lai MK, Tsiang RCC. Microencapsulation of acetaminophen into poly(L-lactide) by three different emulsion solvent-evaporation methods. J Microencapsulation, 2005;22(3):261–74.
   PubMed Web of Science ®Google Scholar
• Li J, Sabliov C. PLA/PLGA nanoparticles for delivery of drugs across the blood-brain barrier. Nanotechnology Rev, 2013;2(3):241–57.
   Web of Science ®Google Scholar
• Miyajima M, Koshika A, Okada J, Ikeda M, Nishimura K. Effect of polymer crystallinity on papaverine release from poly(L-lactic acid) matrix. J Controlled Release, 1997;49(2–3):207–15.
   Web of Science ®Google Scholar
• Odeberg JM, Kaufmann P, Kroon KG, Höglund P. Lipid drug delivery and rational formulation design for lipophilic drugs with low oral bioavailability, applied to cyclosporine. Eur J Pharm Sci, 2003;20(4–5):375–82.
   PubMed Web of Science ®Google Scholar
• Olivier JC. Drug transport to brain with targeted nanoparticles. NeuroRx J. Am Soc Exp NeuroTher, 2005;2(1):108–19.
   Google Scholar
• Pan J, Feng SS. Targeted delivery of paclitaxel using folate-decorated poly(lactide)-vitamin E TPGS nanoparticles. Biomaterials, 2008;29(17):2663–72.
   PubMed Web of Science ®Google Scholar
• Pawar AA, Chen DR, Venkataraman C. Influence of precursor solvent properties on matrix crystallinity and drug release rates from nanoparticle aerosol lipid matrices. Int J Pharm, 2012;430(1–2):228–37.
   PubMed Web of Science ®Google Scholar
• Péan JM, Venier-Julienne MC, Filmon R, Sergent M, Phan-Tan-Luu R, Benoit JP. Optimization of HSA and NGF encapsulation yields in PLGA microparticles. Int J Pharm, 1998;166(1):105–15.
   Web of Science ®Google Scholar
• Porter CJH, Trevaskis NL, Charman WN. Lipids and lipid-based formulations: Optimizing the oral delivery of lipophilic drugs. Nat Rev Drug Discov, 2007;6(3):231–48.
   PubMed Web of Science ®Google Scholar
• Rawat A, Bhardwaj U, Burgess DJ. Comparison of in vitro-in vivo release of Risperdal(®) Consta(®) microspheres. Int J Pharm, 2012;434(1–2):115–21.
   PubMed Web of Science ®Google Scholar
• Stridsberg K, Ryner M, Albertsson A. Controlled ring-opening polymerization: Polymers with designed macromolecular architecture. Adv Polymer Sci, 2002;157:1–25.
   Google Scholar
• Su ZX, Shi Y-N, Teng L-S, Li X, Wang L, Meng Q-F, Teng L-R, Li Y-X. Biodegradable poly(D, L-lactide-co-glycolide) (PLGA) microspheres for sustained release of risperidone: Zero-order release formulation. Pharm Develop Technol, 2011;16(4):377–84.
   PubMed Web of Science ®Google Scholar
• Tamboli V, Mishra GP, Mitra AK. Novel pentablock copolymer (PLA-PCL-PEG-PCL-PLA)-based nanoparticles for controlled drug delivery: Effect of copolymer compositions on the crystallinity of copolymers and in vitro drug release profile from nanoparticles. Colloid Polymer Sci, 2013;291(5):1235–45.
   PubMed Web of Science ®Google Scholar
• Tong R, Coyle VJ, Tang L, Barger AM, Fan TM, Cheng J. Polylactide nanoparticles containing stably incorporated cyanine dyes for in vitro and in vivo imaging applications. Microsc Res Tech, 2010;73(9):901–9.
   PubMed Web of Science ®Google Scholar
• Xiong XY, Tam KC, Gan LH. Release kinetics of hydrophobic and hydrophilic model drugs from pluronic F127/poly(lactic acid) nanoparticles. J Control Release, 2005;103(1):73–82.
   PubMed Web of Science ®Google Scholar
• Zambaux MF, Bonneaux F, Gref R, Dellacherie E, Vigneron C. Preparation and characterization of protein C-loaded PLA nanoparticles. J Control Release, 1999;60(2–3):179–88.
   PubMed Web of Science ®Google Scholar