145
Views
4
CrossRef citations to date
0
Altmetric
Research Article

Thermal sintering: a novel technique used in the design, optimization and biopharmaceutical evaluation of propranolol HCl gastric floating tablets

, , , &
Pages 33-45 | Received 18 Jun 2012, Accepted 23 Oct 2012, Published online: 15 Jan 2013

References

  • Hornsby PR, Maxwell AS. Mechanism of sintering between polypropylene beads. J Mater Sci 1992;27:2525–7
  • German RM. Sintering theory and practice. New York: Wiley-Interscience; 1996
  • Singh R, Poddar SS, Chivate A. Sintering of wax for controlled release from pellets. AAPS PharmSciTech 2007;8:74
  • Siegel R, Cohen J, Brown L, Langer R. Sintered polymers for sustained macromolecular drug release. In Anderson J, Kin SW, eds. Recent advances in drug delivery systems. New York: Plenum; 1982:52
  • Sreenivasa Rao B, Ramana Murthy KV, Seshasayana A, et al. Design and evaluation of ethylene vinyl acetate sintered matrix tablets. Indian J Pharm Sci 2003;65:496
  • Ramana Murthy KV, Rao BS, Seshasayana A, et al. Studies on release of rifampicin from sintered matrix tablets. Indian J Pharm Sci 2001;65:371–8
  • Ramana Murthy KV, Rao BS, Madhuri K, et al. Preparation and evaluation of carnauba wax powder as an excipient for oral controlled release formulations. Int J Pharm Excipients 2000;Oct:251–254
  • Tripathi KD. Antihypertensive drugs: essentials of medical pharmacology. 5th ed. New Delhi: Jaypee Brothers; 2003:235–6
  • Williams DA, Temke TL. Foyes: principles of medicinal chemistry. International student edition. Philadelphia, PA: Lippincott Williams and Wilkins; 2002:489–93
  • Stone FW, Stratta JJS. Ethylene oxide polymers. Encycl Polym Sci Technol 1967;6:103–45
  • Srikanth MV, Sunil SA, Sreenivasa Rao N, et al. Design and in vitro evaluation of effervescent gastric floating drug delivery systems of propanolol HCl. Invest Clin 2012;53:60–70
  • Srikanth MV, Sreenivasa Rao N, Sunil SA, et al. Formulation and evaluation of gastro retentive floating drug delivery system of ofloxacin. Drug Invest Today 2011;3:7–9
  • USP 24 NF 19. United States pharmacopoeial convention. Philadelphia, PA: National Publishing; 2000:1429
  • Lazarus J, Cooper J. Absorption, testing, and clinical evaluation of oral prolonged action drugs. J Pharm Sci 1961;50:715–32
  • Wagner JG. Interpretation of percent dissolved-time plots derived from in vitro testing of conventional tablets and capsules. J Pharm Sci 1969;58:1253–7
  • Higuchi T. Mechanism of sustained action medication: theoretical analysis of rate release of solid drugs dispersed in solid matrices. J Pharm Sci 1963;52:1145–9
  • Korsmeyer R, Gurny R, Peppas N. Mechanisms of solute release from porous hydrophilic polymers. Int J Pharm 1983;15:25–35
  • Hixson AW, Crowell JH. Dependence of reaction velocity upon surface and agitation (I) theoretical consideration. Ind Eng Chem 1931;23:923–31
  • World Health Organization. ICH harmonized tripartite guideline on stability testing of new drug substances and products. Q1A (R2). Geneva: World Health Organization; 2003
  • Srikanth MV, Janaki Ram B, Sunil SA, et al. Development and validation of HPLC method for estimation of propranolol HCl in human plasma. J Sci Ind Res 2012;71:120–3
  • Shailesh P, Laxmanbhai P, Chhaganbhai P. Floating matrix tablets of domperidone formulation and optimization using simplex lattice design. Iranian J Pharm Res 2011;10:447–55
  • Wan LSC, Heng PWS, Wong LF. Relationship between swelling and drug release in a hydrophilic matrix. Drug Dev Ind Pharm 1993;19:1201–10
  • Colombo P, Bettini R, Santi P, et al. Analysis of the swelling and release mechanisms from drug delivery systems with emphasis on drug solubility and water transport. J Control Release 1996;39:231–7
  • Uhumwangho MU, Latha K, Sunil SA, et al. Formulation of gastro-retentive floating tablets of diltiazem hydrochloride with carnauba wax by melt granulation technique. J Pharm Allied Sci 2010;7:979–86
  • Srikanth MV, Uhumwangho MU, Sreenivasa Rao N, et al. Formulation and evaluation of gastro retentive floating drug delivery system for propranolol HCl. J Pharm Allied Sci 2011;8:1339–48
  • Bhosale UV, Kusum Devi V, Nimisha J, Swamy PV. Effect of polymer concentration and viscosity grade on atenolol release from gastric floating drug delivery systems. Indian J Pharm Educ Res 2010;44:267–73
  • Srikanth MV, Janaki Ram B, Sunil SA, et al. Gastroretentive drug delivery systems: novel approaches and its evaluation – a review. Int J Pharm Sci Rev Res 2011;10:203–16
  • Wagner JG, Nelson E. Percent absorbed time plots derived from blood level and/or urinary excretion data. J Pharm Sci 1963;52:610–13

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.