A novel approach to a fine particle coating using porous spherical silica as core particles

References

• Christine C, Jackson JS, Zhi HL, et al. A feasibility study on pellet coating using a high-speed quasi-continuous coater. AAPS Pharm Sci Tech 2012;13:1276–86
   PubMed Web of Science ®Google Scholar
• Kage H, Abe R, Hattanda R, et al. Effect of solid circulation rate on coating efficiency and agglomeration in circulating fluidized bed type coater. Powder Technol 2003;130:203–10
   Web of Science ®Google Scholar
• Lustrik M, Dreu R, Sibanc R, Srcic S. Comparative study of the uniformity of coating thickness of pellets coated with a conventional Wurster chamber and a swirl generator-equipped Wurster chamber. Pharm Dev Technol 2012;17:268–76
   PubMed Web of Science ®Google Scholar
• Ichikawa H, Fujioka K, Adeyeye MC, Fukumori Y. Use of ion-exchange resins to prepare 100 mm-sized microcapsules with prolonged drug-release by the Wurster process. Int J Pharm 2001;216:67–76
   PubMed Web of Science ®Google Scholar
• Jono K, Ichikawa H, Miyamoto M, Fukumori Y. A review of particulate design for pharmaceutical powders and their production by spouted bed coating. Powder Technol 2000;113:269–77
   Web of Science ®Google Scholar
• Hakim LF, Portman JL, Casper MD, Weimer AW. Aggregation behavior of nanoparticles in fluidized beds. Powder Technol 2005;160:149–60
   Web of Science ®Google Scholar
• Tsutsumi A, Nakamoto S, Mineo T, Yoshida K. A novel fluidized-bed coating of fine particles by rapid expansion of supercritical fluid solutions. Powder Technol 1995;85:275–8
   Web of Science ®Google Scholar
• Hemati M, Cherif R, Saleh K, Pont V. Fluidized bed coating and granulation: influence of process-related variables and physicochemical properties on the growth kinetics. Powder Technol 2003;130:18–34
   Web of Science ®Google Scholar
• Roy P, Khanna R, Subbarao D. Granulation time in fluidized bed granulators. Powder Technol 2010;199:95–9
   Web of Science ®Google Scholar
• Hede PD, Bach P, Jensen AD. Small-scale top-spray fluidised bed coating: Granule impact strength, agglomeration tendency and coating layer morphology. Powder Technol 2007;176:156–67
   Web of Science ®Google Scholar
• Ishikawa T, Mukai B, Shiraishi S, et al. Preparation of rapidly disintegrating tablet using new types of microcrystalline cellulose (PH-M series) and low substituted-hydroxypropylcellulose or spherical sugar granules by direct compression method. Chem Pharm Bull 2001;49:134–9
   PubMed Web of Science ®Google Scholar
• Kimura1 S, Iwao1 Y, Ishida M, et al. Optimal conditions to prepare fine globular granules with a multi-functional rotor processor. Int J Pharm 2010;391:244–7
   PubMedGoogle Scholar
• Muschert S, Siepmann F, Cuppok Y, et al. Improved long term stability of aqueous ethylcellulose film coatings: importance of the type of drug and starter core. Int J Pharm 2009;368:138–45
   PubMed Web of Science ®Google Scholar
• El-Malah Y, Nazzal S. Novel use of Eudragit® NE 30D/Eudragit® L 30D-55 blends as functional coating materials in time-delayed drug release applications. Int J Pharm 2008;357:219–27
   PubMed Web of Science ®Google Scholar
• Yoshida T, Tasaki H, Maeda A, et al. Salting-out taste-masking system generates lag time with subsequent immediate release. Int J Pharm 2009;365:81–8
   PubMed Web of Science ®Google Scholar
• Dakshinamurthy DC, Richard AG, Sarala P, Tarun KM. Controlled release multiple layer coatings. Drug Dev Ind Pharm 2010;36:200–8
   PubMed Web of Science ®Google Scholar
• Shimizu T, Sugaya M, Nakano Y, et al. Formulation study for lansoprazole fast-disintegrating tablet. III. Design of rapidly disintegrating tablets. Chem Pharm Bull 2003;51:1121–7
   PubMed Web of Science ®Google Scholar
• Muschert S, Siepmann F, Leclercq B, et al. Prediction of drug release from ethylcellulose coated pellets. J Control Release 2009;135:71–9
   PubMed Web of Science ®Google Scholar
• Maejima T, Kubo M, Osawa T, et al. Application of Tumbling Melt Granulation (TMG) method to prepare controlled-release fine granules. Chem Pharm Bull 1998;46:534–6
   PubMed Web of Science ®Google Scholar
• Ichikawa H, Tokumitsu H, Jono K, et al. Coating of pharmaceutical powders by fluidized bed process. VI. Microencapsulation using blend and composite latices of copoly(ethyl acrylate-methyl methacrylate-2-hydroxyethyl methacrylate). Chem Pharm Bull 1994;42:1308–14
   Web of Science ®Google Scholar
• Fukumori Y, Ichikawa H, Yamaoka Y, et al. Effect of additives on the physical properties of fine ethyl cellulose microcapsules prepared by the Wurster process. Chem Pharm Bull 1991;39:164–9
   Web of Science ®Google Scholar
• Fukumori Y, Ichikawa H, Yamaoka Y, et al. Microgranulation and encapsulation of pulverized pharmaceutical powders with ethyl cellulose by the Wurster process. Chem Pharm Bull 1991;39:1806–12
   Web of Science ®Google Scholar
• Fukumori Y, Ichikawa H, Jono K, et al. Effect of additives on the agglomeration in aqueous coating with hydroxylpropyl cellulose. Chem Pharm Bull 1993;41:725–30
   Web of Science ®Google Scholar
• Yuasa H, Nakano T, Kanaya Y. Suppression of agglomeration in fluidized bed coating I. Suppression of agglomeration by adding NaCl. Int J Pharm 1997;158:195–201
   Google Scholar
• Guignon B, Regalado E, Duquenoy A, Dumoulin E. Helping to choose operating parameters for a coating fluid bed process. Powder Technol 2003;130:193–8
   Web of Science ®Google Scholar
• Nakano T, Yuasa H. Suppression of agglomeration in fluidized bed coating. IV. Effects of sodium citrate concentration on the suppression of particle agglomeration and the physical properties of HPMC film. Int J Pharm 2001;215:3–12
   PubMed Web of Science ®Google Scholar
• Hede PD, Bach P, Jensen AD. Fluidized-bed coating with sodium sulfate and PVA-TiO2, 2. Influence of coating solution viscosity, stickiness, pH, and droplet diameter on agglomeration. Ind Eng Chem Res 2009;48:1905–13
   Web of Science ®Google Scholar
• Nimkulrat S, Suchiva K, Phinyocheep P, Puttipipatkhachorn S. Influence of selected surfactants on the tackiness of acrylic polymer films. Int J Pharm 2004;287:27–37
   PubMed Web of Science ®Google Scholar
• Cervera MF, Heinämäki J, Räsänen E, et al. Determination of tackiness of chitosan film-coated pellets exploiting minimum fluidization velocity. Int J Pharm 2004;281:119–27
   PubMedGoogle Scholar
• Shimizu T, Nakano Y, Morimoto S, et al. Formulation study for lansoprazole fast-disintegrating tablet. I. Effect of compression on dissolution behavior. Chem Pharm Bull 2003;51:942–7
   PubMed Web of Science ®Google Scholar
• Heng P, Wan L, Tan Y. Relationship between aggregation of HPMC coated spheroids and tackiness/viscosity/additives of the coating formulations. Int J Pharm 1996;138:57–66
   Web of Science ®Google Scholar
• Lin SY, Chen KS, Run-Chu L. Organic esters of plasticizers affecting the water absorption, adhesive property, glass transition temperature and plasticizer permanence of Eudragit acrylic films. J Control Release 2000;68:343–50
   PubMed Web of Science ®Google Scholar
• Chan LW, Wong TW, Chua PC, et al. Anti-tack action of polyvinylpyrrolidone on hydroxypropylmethylcellulose solution. Chem Pharm Bull 2003;51:107–12
   Google Scholar
• Pan X, Shichao YE, Zhang Z, et al. A study of spray granulation in vibrated fluidized bed with internal heating tubes. Front Chem Eng China 2009;3:78–82
   Google Scholar
• Barletta D, Donsi G, Ferrari G, et al. The effect of mechanical vibration on gas fluidization of a fine aeratable powder. Chem Eng Res Des 2008;86:359–69
   Web of Science ®Google Scholar
• Watano S, Nakamura H, Hamada K, et al. Fine particle coating by a novel rotating fluidized bed coater. Powder Technol 2004;141:172–6
   Web of Science ®Google Scholar
• Dreu R, Luštrik M, Perpar M, et al. Fluid-bed coater modifications and study of their influence on the coating process of pellets. Drug Dev Ind Pharm 2012;38:501–11
   PubMed Web of Science ®Google Scholar
• Verraedt E, Mooter G, Martens JA. Novel amorphous microporous silica spheres for controlled release applications. J Pharm Sci 2011;100:4295–301
   PubMed Web of Science ®Google Scholar
• Ito F, Shudo K, Yamaguchi K. Total synthesis of (±)-hyrtiazepine. Tetrahedron 2011;67:1805–11
   Web of Science ®Google Scholar
• Abdullah EC, Geldart D. The use of bulk density measurements as flowability indicators. Powder Technol 1999;102:151–65
   Web of Science ®Google Scholar
• Hamashita T, Nakagawa Y, Aketo T, Watano S. Granulation of core particles suitable for film coating by agitation fluidized bed I. Optimum formulation for core particles and development of a novel friability test method. Chem Pharm Bull 2007;55:1169–74
   PubMed Web of Science ®Google Scholar
• Nagel KM, Peck GE. Investigating the effects of excipients on the powder flow characteristics. Drug Dev Ind Pharm 2003;29:277–87
   PubMed Web of Science ®Google Scholar
• Quispe-Condori S, Saldaña MDA, Temelli F. Microencapsulation of flax oil with zein using spray and freeze drying. LWT-Food Sci Technol 2011;40:1880–7
   Google Scholar
• Hede PD, Bach P, Jensen AD. Small-scale top-spray fluidised bed coating: Granule impact strength, agglomeration tendency and coating layer morphology. Powder Technol 2007;176:156–67
   Web of Science ®Google Scholar
• Schaafsma SH, Vonk P, Segers P, Kossen NWF. Description of agglomerate growth. Powder Technol 1998;97:183–90
   Web of Science ®Google Scholar
• Ehlers H, Liu A, Räikkönen H, et al. Granule size control and targeting in pulsed spray fluid bed granulation. Int J Pharm 2009;377:9–15
   PubMed Web of Science ®Google Scholar
• Iveson SM, Litster JD. Growth regime map for liquid-bound granules. AIChE J 1998;44:1510–18
   Web of Science ®Google Scholar
• Airaksinen S, Karjalainen M, Shevchenko A, et al. Role of water in the physical stability of solid dosage formulations. J Pharm Sci 2005;94:2147–65
   PubMed Web of Science ®Google Scholar
• Ronsse F, Depelchin J, Pieters JG. Particle surface moisture content estimation using population balance modeling in fluidised bed agglomeration. J Food Eng 2012;109:347–57
   Web of Science ®Google Scholar
• Langrish TAG, Kockel TK. The assessment of a characteristic drying curve for milk powder for use in computational fluid dynamics modelling. Chem Engr J 2001;84:69–74
   Web of Science ®Google Scholar
• Abberger T. The effect of powder type, free moisture and deformation behaviour of granules on the kinetics of fluid bed granulation. Eur J Pharm Biopharm 2001;52:327–36
   PubMed Web of Science ®Google Scholar
• Abberger T, Seo A, Schæfer T. The effect of droplet size and powder particle size on the mechanisms of nucleation and growth in fluid bed melt agglomeration. Int J Pharm 2002;249:185–97
   PubMed Web of Science ®Google Scholar
• Martin JT, Anthony JH. Dry powder inhaler formulation. Respir Care 2005;50:1209–27
   PubMedGoogle Scholar
• Yeo THC, Tan IAW, Abdullah MO. Development of adsorption air-conditioning technology using modified activated carbon -- A review. Renew Sust Energ Rev 2012;16:3355–63
   Web of Science ®Google Scholar
• Umprayn K, Mendes RW. Hygroscopicity and moisture adsorption on kinetics of pharmaceutical solids: a review. Drug Dev Ind Pharm 1987;13:653–93
   Web of Science ®Google Scholar
• Ennis BJ. A microlevel-based characterization of granulation phenomena. Powder Technol 1991;65:257–72
   Web of Science ®Google Scholar
• Hartung A, Knoell M, Schmidt U, Langguth P. Relevance of air-to-liquid mass ratio effect on final granule properties of an Enalapril maleate formulation. Drug Dev Ind Pharm 2012;38:12–8
   PubMed Web of Science ®Google Scholar
• Xua J, Bovetb LL, Zhao K. Taste masking microspheres for orally disintegrating tablets. Int J Pharm 2008;359:63–9
   PubMedGoogle Scholar
• Tzika M, Alexandridou S, Kiparissides C. Evaluation of the morphological and release characteristics of coated fertilizer granules produced in a Wurster fluidized bed. Powder Technol 2003;132:16–24
   Web of Science ®Google Scholar