Formulation of solid self-nanoemulsifying drug delivery systems using N-methyl pyrrolidone as cosolvent

References

• Ren S, Mu H, Alchaer F, et al. Optimization of self nanoemulsifying drug delivery system for poorly water-soluble drug using response surface methodology. Drug Dev Ind Pharm 2013;39:799–806
   PubMed Web of Science ®Google Scholar
• Merisko-Liversidge E, Liversidge GG. Nanosizing for oral and parenteral drug delivery: a perspective on formulating poorly-water soluble compounds using wet media milling technology. Adv Drug Deliv Rev 2011;63:427–40
   PubMed Web of Science ®Google Scholar
• Lei Y, Lu Y, Qi J, et al. Solid self-nanoemulsifying cyclosporin A pellets prepared by fluid-bed coating: preparation, characterization and in vitro redispersibility. Int J Nanomedicine 2011;6:795–805
   PubMed Web of Science ®Google Scholar
• Kuentz M. Lipid-based formulations for oral delivery of lipophilic drugs. Drug Discov Today Technol 2012;9:97–104
   Google Scholar
• Miller JM, Beig A, Carr RA, et al. A win-win solution in oral delivery of lipophilic drugs: supersaturation via amorphous solid dispersions increases apparent solubility without sacrifice of intestinal membrane permeability. Mol Pharm 2012;9:2009–16
   PubMed Web of Science ®Google Scholar
• Hao L, Wang X, Zhang D, et al. Studies on the preparation, characterization and pharmacokinetics of Amoitone B nanocrystals. Int J Pharm 2012;433:157–64
   PubMed Web of Science ®Google Scholar
• Zhang M, Li H, Lang B, et al. Formulation and delivery of improved amorphous fenofibrate solid dispersions prepared by thin film freezing. Eur J Pharm Biopharm 2012;82:534–44
   PubMed Web of Science ®Google Scholar
• Zhao G, Duan J, Xie Y, et al. Effects of solid dispersion and self-emulsifying formulations on the solubility, dissolution, permeability and pharmacokinetics of isorhamnetin, quercetin and kaempferol in total flavones of Hippophae rhamnoides L. Drug Dev Ind Pharm 2013;39:1037–45
   PubMed Web of Science ®Google Scholar
• Naylor A, Lewis AL, Ilium L. Supercritical fluid-mediated methods to encapsulate drugs: recent advances and new opportunities. Ther Deliv 2011;2:1551–65
   PubMedGoogle Scholar
• Su FY, Lin KJ, Sonaje K, et al. Protease inhibition and absorption enhancement by functional nanoparticles for effective oral insulin delivery. Biomaterials 2012;33:2801–11
   PubMed Web of Science ®Google Scholar
• Guo JJ, Yue PF, Lv JL, et al. Development and in vivo/in vitro evaluation of novel herpetrione nanosuspension. Int J Pharm 2013;441:227–33
   PubMed Web of Science ®Google Scholar
• Tan BJ, Liu Y, Chang KL, et al. Perorally active nanomicellar formulation of quercetin in the treatment of lung cancer. Int J Nanomedicine 2012;7:651–61
   PubMed Web of Science ®Google Scholar
• Zheng W, Jain A, Papoutsakis D, et al. Selection of oral bioavailability enhancing formulations during drug discovery. Drug Dev Ind Pharm 2012;38:235–47
   PubMed Web of Science ®Google Scholar
• Mercuri A, Passalacqua A, Wickham MS, et al. The effect of composition and gastric conditions on the self-emulsification process of ibuprofen-loaded self-emulsifying drug delivery systems: a microscopic and dynamic gastric model study. Pharm Res 2011;28:1540–51
   PubMed Web of Science ®Google Scholar
• Mohsin K. Design of lipid-based formulations for oral administration of poorly water-soluble drug fenofibrate: effects of digestion. AAPS PharmSciTech 2012;13:637–46
   PubMed Web of Science ®Google Scholar
• Shahba AA, Mohsin K, Alanazi FK. Novel self-nanoemulsifying drug delivery systems (SNEDDS) for oral delivery of cinnarizine: design, optimization, and in-vitro assessment. AAPS PharmSciTech 2012;13:967–77
   PubMed Web of Science ®Google Scholar
• Patil SS, Venugopal E, Bhat S, et al. Microstructural elucidation of self-emulsifying system: effect of chemical structure. Pharm Res 2012;29:2180–8
   PubMed Web of Science ®Google Scholar
• Kang MJ, Jung SY, Song WH, et al. Immediate release of ibuprofen from Fujicalin®-based fast dissolving self-emulsifying tablets. Drug Dev Ind Pharm 2011;37:1298–305
   PubMed Web of Science ®Google Scholar
• Chen ZQ, Liu Y, Zhao JH, et al. Improved oral bioavailability of poorly water-soluble indirubin by a supersaturatable self-microemulsifying drug delivery system. Int J Nanomedicine 2012;7:1115–25
   PubMed Web of Science ®Google Scholar
• Singh B, Singh R, Bandyopadhyay S, et al. Optimized nanoemulsifying systems with enhanced bioavailability of carvedilol. Colloids Surf B Biointerfaces 2013;101:465–74
   PubMed Web of Science ®Google Scholar
• Do TT, Speybroeck MV, Mols R, et al. The conflict between in vitro release studies in human biorelevant media and the in vivo exposure in rats of the lipophilic compound Fenofibrate. Int J Pharm 2011;414:118–24
   PubMed Web of Science ®Google Scholar
• Mukherjee T, Plakogiannis FM. Effects of process parameters on solid self-microemulsifying particles in a laboratory scale fluid bed. Pharm Dev Technol 2012;17:511–20
   PubMed Web of Science ®Google Scholar
• Quan Q, Kim DW, Marasini N, et al. Physicochemical characterization and in vivo evaluation of solid self-nanoemulsifying drug delivery system for oral administration of docetaxel. J Microencapsul 2013;30:307–14
   PubMed Web of Science ®Google Scholar
• Gupta S, Chavhan S, Sawant KK. Self-nanoemulsifying drug delivery system for adefovir dipivoxil: design, characterization, in vitro and ex vivo evaluation. Colloids Surf A: Physicochem Eng Aspects 2011;392:145–55
   Web of Science ®Google Scholar
• Zvonar A, Bolko K, Gasperlin M. Microencapsulation of self-microemulsifying systems: optimization of shell-formation phase and hardening process. Int J Pharm 2012;437:294–302
   PubMed Web of Science ®Google Scholar
• Beg S, Jena SS, Patra H, et al. Development of solid self-nanoemulsifying granules (SSNEGs) of ondansetron hydrochloride with enhanced bioavailability potential. Colloids Surf B Biointerfaces 2013;101:414–23
   PubMed Web of Science ®Google Scholar
• Tarantino R, Bishop E, Cen FC, et al. N-Methyl-2-pyrrolidone as a cosolvent: relationship of cosolvent effect with solute polarity and the presence of proton-donating groups on model drug compounds. J Pharm Sci 1994;83:1213–16
   PubMed Web of Science ®Google Scholar
• Sanghvi R, Narazaki R, Machatha SG, et al. Solubility improvement of drugs using N-methyl pyrrolidone. AAPS PharmSciTech 2008;9:366–76
   PubMed Web of Science ®Google Scholar
• Sasaki J, Otonari T, Uchida Y, et al. Effect of pravastatin and atorvastatin on HDL cholesterol and glucose metabolism in patients with dyslipidemia and glucose intolerance: the PRAT study. J Atheroscler Thromb 2013;20:368–79
   PubMed Web of Science ®Google Scholar
• Jin D, Wu Y, Zhao L, et al. Atorvastatin reduces serum HMGB1 levels in patients with hyperlipidemia. Exp Ther Med 2012;4:1124–6
   PubMed Web of Science ®Google Scholar
• Yang Z, Lee MJ, Zhao Y, et al. Metabolism of tocotrienols in animals and synergistic inhibitory actions of tocotrienols with atorvastatin in cancer cells. Genes Nutr 2012;7:11–18
   PubMed Web of Science ®Google Scholar
• Wani TA, Ahmad A, Zargar S, et al. Use of response surface methodology for development of new microwell-based spectrophotometric method for determination of atrovastatin calcium in tablets. Chem Cent J 2012;6:134–42
   PubMed Web of Science ®Google Scholar
• Vaculikova E, Grunwaldova V, Kral V, et al. Preparation of candesartan and atorvastatin nanoparticles by solvent evaporation. Molecules 2012;17:13221–34
   PubMed Web of Science ®Google Scholar
• Chadha R, Kuhad A, Arora P, et al. Characterisation and evaluation of pharmaceutical solvates of atorvastatin calcium by thermoanalytical and spectroscopic studies. Chem Cent J 2012;6:114. doi:10.1186/1752-153X-6-114
   PubMed Web of Science ®Google Scholar
• Ali KA, Mukherjee B, Bandyopadhyay AK. Formulation development and in vitro evaluation of solidified self-microemulsion in the form of tablet containing atorvastatin calcium. Drug Dev Ind Pharm 2013;39:1742–9
   PubMed Web of Science ®Google Scholar
• Lv HX, Zhang ZH, Hui-Jiang Waddad AY, et al. Preparation, physicochemical characteristics and bioavailability studies of an atorvastatin hydroxypropyl-beta-cyclodextrin complex. Pharmazie 2012;67:46–53
   PubMed Web of Science ®Google Scholar
• Raza K, Negi P, Takyar S, et al. Novel dithranol phospholipid microemulsion for topical application: development, characterization and percutaneous absorption studies. J Microencapsul 2011;28:190–9
   PubMed Web of Science ®Google Scholar
• Venkatesh G, Majid MI, Mansor SM, et al. In vitro and in vivo evaluation of self-microemulsifying drug delivery system of buparvaquone. Drug Dev Ind Pharm 2010;36:735–45
   PubMed Web of Science ®Google Scholar
• Bandyopadhyay S, Katare OP, Singh B. Optimized self nano-emulsifying systems of ezetimibe with enhanced bioavailability potential using long chain and medium chain triglycerides. Colloids Surf B Biointerfaces 2012;100:50–61
   PubMed Web of Science ®Google Scholar
• Mandawgade SD, Sharma S, Pathak S, et al. Development of SMEDDS using natural lipophile: application to β-artemether delivery. Int J Pharm 2008;362:179–83
   PubMed Web of Science ®Google Scholar
• Wang Y, Sun J, Zhang T, et al. Enhanced oral bioavailability of tacrolimus in rats by selfmicroemulsifying drug delivery systems. Drug Dev Ind Pharm 2011;37:1225–30
   PubMed Web of Science ®Google Scholar
• Abdelbary G, Amin M, Salah S. Self nano-emulsifying simvastatin based tablets: design and in vitro/in vivo evaluation. Pharm Dev Technol 2013;18:1294–304
   PubMed Web of Science ®Google Scholar
• Kanuganti S, Jukanti R, Veerareddy PR, et al. Paliperidone-loaded self-emulsifying drug delivery systems (SEDDS) for improved oral delivery. J Dispersion Sci Technol 2012;33:506–15
   Web of Science ®Google Scholar
• Ahmad J, Kohli K, Mir SR, et al. Formulation of self-nanoemulsifying drug delivery system for telmisartan with improved dissolution and oral bioavailability. J Dispersion Sci Technol 2011;32:958–68
   Web of Science ®Google Scholar
• Kalhapure RS, Akamanchi KG. Oleic acid based heterolipid synthesis, characterization and application in self-microemulsifying drug delivery system. Int J Pharm 2012;425:9–18
   PubMed Web of Science ®Google Scholar
• Shanmugam S, Baskaran R, Balakrishnan P, et al. Solid self-nanoemulsifying drug delivery system (S-SNEDDS) containing phosphatidylcholine for enhanced bioavailability of highly lipophilic bioactive carotenoid lutein. Eur J Pharm Biopharm 2011;79:250–7
   PubMed Web of Science ®Google Scholar
• Elnaggar YSR, El-Massik MA, Abdallah OY. Sildenafil citrate nanoemulsion vs self-nanoemulsifying delivery systems: rational development and transdermal permeation. Int J Nanotechnol 2011;8:749–63
   Web of Science ®Google Scholar
• Shen Q, Li X, Yuan D, et al. Enhanced oral bioavailability of daidzein by self-microemulsifying drug delivery system. Chem Pharm Bull 2010;58:639–43
   PubMed Web of Science ®Google Scholar
• Hu L, Yang J, Liu W, et al. Preparation and evaluation of ibuprofen-loaded microemulsion for improvement of oral bioavailability. Drug Deliv 2011;18:90–5
   PubMed Web of Science ®Google Scholar
• Yoo JH, Shanmugam S, Thapa P, et al. Novel self-nanoemulsifying drug delivery system for enhanced solubility and dissolution of lutein. Arch Pharm Res 2010;33:417–26
   PubMed Web of Science ®Google Scholar
• Franceschinis E, Bortoletto C, Perissutti B, et al. Self-emulsifying pellets in a lab-scale high shear mixer: formulation and production design. Powder Technol 2011;207:113–18
   Web of Science ®Google Scholar
• Li W, Yi S, Wang Z, et al. Self-nanoemulsifying drug delivery system of persimmon leaf extract: optimization and bioavailability studies. Int J Pharm 2011;420:161–71
   PubMed Web of Science ®Google Scholar
• Garg Y, Pathak K. Design and in vitro performance evaluation of purified microparticles of pravastatin sodium for intestinal delivery. AAPS PharmSciTech 2011;12:673–82
   PubMed Web of Science ®Google Scholar
• Ghai D, Sinha VR. Nanoemulsions as self-emulsified drug delivery carriers for enhanced permeability of the poorly water-soluble selective β1-adrenoreceptor blocker talinolol. Nanomedicine 2012;8:618–26
   PubMed Web of Science ®Google Scholar
• Matsaridou I, Barmpalexis P, Salis A, et al. The influence of surfactant HLB and oil/surfactant ratio on the formation and properties of self-emulsifying pellets and microemulsion reconstitution. AAPS PharmSciTech 2012;13:1319–30
   PubMed Web of Science ®Google Scholar
• Mahdi ES, Sakeena MH, Abdulkarim MF, et al. Effect of surfactant and surfactant blends on pseudoternary phase diagram behavior of newly synthesized palm kernel oil esters. Drug Des Devel Ther 2011;5:311–23
   PubMed Web of Science ®Google Scholar
• Bachhav YG, Date AA, Patravale VB. Exploring the potential of N-methyl pyrrolidone as a cosurfactant in the microemulsion systems. Int J Pharm 2006;326:186–9
   PubMed Web of Science ®Google Scholar
• Jouyban A, Fakhree MA, Shayanfar A. Review of pharmaceutical applications of N-Methyl-2-Pyrrolidone. J Pharm Pharmaceut Sci 2010;13:524–35
   PubMed Web of Science ®Google Scholar
• Liang L, Shojaei AH, Ibrahim SA, Burnside BA. Self-emulsifying formulations of fenofibrate and/or fenofibrate derivatives with improved oral bioavailability and/or reduced food effect. US Patent, No 7,022,337B2; 2006
   Google Scholar
• Sprunk A, Strachan CJ, Graf A. Rational formulation development and in vitro assessment of SMEDDS for oral delivery of poorly water soluble drugs. Eur J Pharm Sci 2012;46:508–15
   PubMed Web of Science ®Google Scholar
• Bali V, Ali M, Ali J. Nanocarrier for the enhanced bioavailability of a cardiovascular agent: in vitro, pharmacodynamic, pharmacokinetic and stability assessment. Int J Pharm 2011;403:46–56
   PubMed Web of Science ®Google Scholar
• Singh SK, Verma PR, Razdan B. Development and characterization of a carvedilolloaded self-microemulsifying delivery system. Clin Res Regul Aff 2009;26:50–64
   Google Scholar
• Basalious EB, Shawky N, Badr-Eldin SM. SNEDDS containing bioenhancers for improvement of dissolution and oral absorption of lacidipine I: development and optimization. Int J Pharm 2010;391:203–11
   PubMed Web of Science ®Google Scholar
• Xiao L, Yi T, Liu Y. A new self-microemulsifying mouth dissolving film to improve the oral bioavailability of poorly water soluble drugs. Drug Dev Ind Pharm 2012;39:1284–90
   PubMed Web of Science ®Google Scholar
• Zargar-Shoshtari S, Wen J, Alany RG. Formulation and physicochemical characterization of imwitor 308 based self microemulsifying drug delivery systems. Chem Pharm Bull 2010;58:1332–8
   PubMed Web of Science ®Google Scholar