619
Views
14
CrossRef citations to date
0
Altmetric
Research Article

Effect of microporation on passive and iontophoretic delivery of diclofenac sodium

, , &
Pages 1962-1967 | Received 16 Jul 2014, Accepted 26 Jan 2015, Published online: 11 Mar 2015

References

  • Arora A, Prausnitz MR, Mitragotri S. Micro-scale devices for transdermal drug delivery. Int J Pharm 2008;364:227–36
  • Shah UU, Roberts M, Orlu Gul M, et al. Needle-free and microneedle drug delivery in children: a case for disease-modifying antirheumatic drugs (DMARDs). Int J Pharm 2010;416:1–11
  • Xie Y, Xu B, Gao Y. Controlled transdermal delivery of model drug compounds by MEMS microneedle array. Nanomedicine 2005;1:184–90
  • Kochhar JS, Goh WJ, Chan SY, Kang L. A simple method of microneedle array fabrication for transdermal drug delivery. Drug Dev Ind Pharm 2012;39:299–309
  • Park JH, Choi SO, Seo S, et al. A microneedle roller for transdermal drug delivery. Eur J Pharm Biopharm 2010;76:282–9
  • Ito Y, Kashiwara S, Fukushima K, Takada K. Two-layered dissolving microneedles for percutaneous delivery of sumatriptan in rats. Drug Dev Ind Pharm 2011;37:1387–93
  • Wong CY, Guu YB, Wang MT, Wang DP. Percutaneous transport of diclofenac sodium from mixtures of fatty alcohol (or fatty acid) and propylene glycol through the rabbit abdominal skin. Drug Dev Ind Pharm 1999;25:1209–13
  • Gan TJ. Diclofenac: an update on its mechanism of action and safety profile. Curr Med Res Opin 2010;26:1715–31
  • Lehtola J, Sipponen P. A gastroscopic and histological double-blind study of the effects of diclofenac sodium and naproxen on the human gastric mucosa. Scand J Rheumatol 1977;6:97–102
  • Hsieh YL. Effects of ultrasound and diclofenac phonophoresis on inflammatory pain relief: suppression of inducible nitric oxide synthase in arthritic rats. Phys Ther 2006;86:39–49
  • Clijsen R, Taeymans J, Baeyens JP, et al. The effects of iontophoresis in the treatment of musculoskeletal disorders – a systematic review and meta-analysis. Drug Deliv Lett 2012;2:180–94
  • Pandey S, Patel B, Viral D, et al. Microneedle: various techniques of fabrications and evaluations. Int J ChemTech Res 2009;1:1058–62
  • Badran MM, Kuntsche J, Fahr A. Skin penetration enhancement by a microneedle device (Dermaroller) in vitro: dependency on needle size and applied formulation. Eur J Pharm Sci 2009;36:511–23
  • Kolli CS, Xiao J, Parsons DL, Babu RJ. Microneedle assisted iontophoretic transdermal delivery of prochlorperazine edisylate. Drug Dev Ind Pharm 2012;38:571–6
  • Kalluri H, Kolli CS, Banga AK. Characterization of microchannels created by metal microneedles: formation and closure. AAPS J 2011;13:473–81
  • Patel DR, Joshi A, Patel HH, Stagni G. Development and in-vivo evaluation of ondansetron gels for transdermal delivery. Drug Dev Ind Pharm 2015. [Epub ahead of print]. doi:10.3109/03639045.2014.925916
  • Stagni G. Cutaneous microdialysis. In: Murthy NS, ed. Dermatokinetics of theraputic agents. Boca Raton, London, New York: CRC Press, Taylor & Francis Group; 2011:131–47
  • Stagni G, O'Donnell D, Liu YJ, et al. Iontophoretic current and intradermal microdialysis recovery in humans. J Pharmacol Toxicol Methods 1999;41:49–54
  • Sintov AC, Botner S. Transdermal drug delivery using microemulsion and aqueous systems: influence of skin storage conditions on the in vitro permeability of diclofenac from aqueous vehicle systems. Int J Pharm 2006;311:55–62
  • Stagni G, Shukla C. Pharmacokinetics of methotrexate in rabbit skin and plasma after iv-bolus and iontophoretic administrations. J Control Release 2003;93:283–92
  • Mannem V, Nanjarapalle C, Stagni G. Iontophoresis of amoxicillin and cefuroxime: rapid therapeutic concentrations in skin. Drug Dev Ind Pharm 2014;40:325–9
  • Anigbogu A, Patil S, Singh P, et al. An in vivo investigation of the rabbit skin responses to transdermal iontophoresis. Int J Pharm 2000;200:195–206
  • Levin J, Maibach H. The correlation between transepidermal water loss and percutaneous absorption: an overview. J Control Release 2005;103:291–9
  • Velisetty S. Pharmacokinetics of diclofenac sodium in plasma and skin following IV-infusion in a rabbit model [master thesis]. Long Island University; 2013
  • Kasha PC, Anderson CR, Morris RL, et al. Subcutaneous concentrations following topical iontophoretic delivery of diclofenac. Drug Discov Ther 2012;6:256–62
  • Yan G, Warner KS, Zhang J, et al. Evaluation needle length and density of microneedle arrays in the pretreatment of skin for transdermal drug delivery. Int J Pharm 2010;391:7–12
  • Modepalli N, Jo S, Repka MA, Murthy SN. Microporation and ‘iron’tophoresis for treating iron deficiency anemia. Pharm Res 2013;30:889–98
  • Bal SM, Caussin J, Pavel S, Bouwstra JA. In vivo assessment of safety of microneedle arrays in human skin. Eur J Pharm Sci 2008;35:193–202
  • Zhou CP, Liu YL, Wang HL, et al. Transdermal delivery of insulin using microneedle rollers in vivo. Int J Pharm 2010;392:127–33
  • Riecke BF, Bartels EM, Torp-Pedersen S, et al. A microdialysis study of topically applied diclofenac to healthy humans: passive versus iontophoretic delivery. Results Pharma Sci 2011;1:76–9

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.