136
Views
2
CrossRef citations to date
0
Altmetric
Non-themed Articles

Thermal, mechanical and drug release characteristics of an acrylic film using active pharmaceutical ingredient as non-traditional plasticizer

, , &
Pages 644-653 | Received 04 Feb 2015, Accepted 10 Jun 2015, Published online: 02 Jul 2015

References

  • Rosen SL. Fundamental principles of polymeric materials. New York: John Wiley & Sons; 1993
  • Snejdrova E, Dittrich M. Pharmaceutically used plasticizers. In: Luqman M, ed. Recent advances in plasticizers. Rijeka: InTech; 2012:45–68
  • Seniohev VY, Tereshatov VV. Influence of plasticizers on the glass transition temperature of polymers. In: Wypych G, ed. Handbook of plasticizers. New York: ChemTec Publishing; 2004:218–27
  • Bodmeier R, Paeratakul O. Determination of plasticizers commonly used in pharmaceutical dosage forms by high performance liquid chromatography. J Liq Chromatogr 1991;14:365–75
  • Bruce LD, Koleng JJ, McGinity JW. The influence of polymeric subcoats and pellet formulation on the release of chlorpheniramine maleate from enteric coated pellets. Drug Dev Ind Pharm 2003;29:909–24
  • Castle L, Gilbert J, Eklund T. Migration of plasticizer from poly(vinyl chloride) milk tubing. Food Addit Contam 1990;7:591–6
  • Sharman M, Read WA, Castle L, Gilbert J. Levels of di-(2-ethylhexyl)phthalate and total phthalate esters in milk, cream, butter and cheese. Food Addit Contam 1994;11:375–85
  • Castle L, Mercer AJ, Startin JR, Gilbert J. Migration from plasticized films into foods 3. Migration of phthalate, sebacate, citrate and phosphate esters from films used for retail food packaging. Food Addit Contam 1988;5:9–20
  • Castle L, Mayo A, Gilbert J. Migration of plasticizers from printing inks into foods. Food Addit Contam 1989;6:437–43
  • Nerín C, Cacho J, Gancedo P. Plasticizers from printing inks in a selection of food packagings and their migration to food. Food Addit Contam 1993;10:453–60
  • Page BD, Lacroix GM. The occurrence of phthalate ester and di-2-ethylhexyl adipate plasticizers in Canadian packaging and food sampled in 1985–1989: a survey. Food Addit Contam 1995;12:129–51
  • Murphy J. Additives for plastics handbook. New York: Elsevier; 2001
  • Baltacioğlu H, Balköse D. Effect of zinc stearate and/or epoxidized soybean oil on gelation and thermal stability of PVC-DOP plastigels. J Appl Polym Sci 1999;74:2488–98
  • Meier MM, Kanis LA, Soldi V. Characterization and drug-permeation profiles of microporous and dense cellulose acetate membranes: influence of plasticizer and pore forming agent. Int J Pharm 2004;278:99–110
  • Pongjanyakul T, Puttipipatkhachorn S. Alginate-magnesium aluminum silicate films: effect of plasticizers on film properties, drug permeation and drug release from coated tablets. Int J Pharm 2007;333:34–44
  • Aitken-nichol C, Zhang F, McGinity JW. Hot melt extrusion of acrylic films. Pharm Res 1996;13:804–8
  • Wu C, McGinity JW. Non-traditional plasticization of polymeric films. Int J Pharm 1999;177:15–27
  • Wu C, McGinity JW. Influence of ibuprofen as a solid-state plasticizer in Eudragit RS 30 D on the physicochemical properties of coated beads. AAPS PharmSciTech [electronic resource] 2001;2:24
  • Özgüney I, Shuwisitkul D, Bodmeier R. Development and characterization of extended release Kollidon® SR mini-matrices prepared by hot-melt extrusion. Eur J Pharm Biopharm 2009;73:140–5
  • Claeys B, Coen RD, De Geest BG, et al. Structural modifications of polymethacrylates: impact on thermal behavior and release characteristics of glassy solid solutions. Eur J Pharm Biopharm 2013;85:1206–14
  • Wiranidchapong C, Ruangpayungsak N, Suwattanasuk P, et al. Plasticizing effect of ibuprofen induced an alteration of drug released from Kollidon SR matrices produced by direct compression. Drug Dev Ind Pharm 2015;41:1037–46
  • Siepmann F, Le Brun V, Siepmann J. Drugs acting as plasticizers in polymeric systems: a quantitative treatment. J Control Release 2006;115:298–306
  • Jenquin MR, Liebowitz SM, Sarabia RE, McGinity JW. Physical and chemical factors influencing the release of drugs from acrylic resin films. J Pharm Sci 1990;79:811–16
  • Repka MA, Gerding TG, Repka SL, McGinity JW. Influence of plasticizers and drugs on the physical-mechanical properties of hydroxypropylcellulose films prepared by hot melt extrusion. Drug Dev Ind Pharm 1999;25:625–33
  • Zhu Y, Shah NH, Malick AW, et al. Solid-state plasticization of an acrylic polymer with chlorpheniramine maleate and triethyl citrate. Int J Pharm 2002;241:301–10
  • Selmin F, Franceschini I, Cupone IE, et al. Aminoacids as non-traditional plasticizers of maltodextrins fast-dissolving films. Carbohyd Poylm 2015;115:613–16
  • Kangarlou S, Haririan I, Gholipour Y. Physico-mechanical analysis of free ethyl cellulose films comprised with novel plasticizers of vitamin resources. Int J Pharm 2008;356:153–66
  • Schneider HA. The Gordon–Taylor equation: additivity and interaction in compatible polymer blends. Makromol Chem 1988;189:1941–55
  • Kuo SW, Chang FC. Miscibility and hydrogen bonding in blends of poly(vinylphenol-co-methyl methacrylate) with poly(ethylene oxide). Macromolecules 2001;34:4089–97
  • Kuo SW, Huang CF, Chang FC. Study of hydrogen-bonding strength in poly(ɛ-caprolactone) blends by DSC and FTIR. J Polym Sci Part B Polym Phys 2001;39:1348–59
  • Maldonado-Santoyo M, Ortíz-Estrada C, Luna-Bárcenas G, et al. Miscibility behavior and hydrogen bonding in blends of poly(vinyl phenyl ketone hydrogenated) and poly(2-ethyl-2-oxazoline). J Polym Sci Part B Polym Phys 2004;42:636–45
  • Wiranidchapong C, Tucker IG, Rades T, Kulvanich P. Miscibility and interactions between 17β-estradiol and Eudragit® RS in solid dispersion. J Pharm Sci 2008;97:4879–88
  • Wiranidchapong C, Rades T, Kulvanich P, Tucker IG. Method of preparation does not affect the miscibility between steroid hormone and polymethacrylate. Thermochim Acta 2009;485:57–64
  • Wiranidchapong C. Solid state and thermal behavior of 17β-estradiol in ammonioethyl methacrylate ester copolymer. In: Dubey R, ed. Sex hormones. Croatia: InTech; 2012:403--30
  • Barmpalexis P, Koutsidis I, Karavas E, et al. Development of PVP/PEG mixtures as appropriate carriers for the preparation of drug solid dispersions by melt mixing technique and optimization of dissolution using artificial neural networks. Eur J Pharm Biopharm 2013;85:1219–31
  • Buckland ST, Burnham KP, Augustin NH. Model selection: an integral part of inference. Biometrics 1997;53:603–18
  • Li Z, Chang P-H, Jean J-S, et al. Mechanism of chlorpheniramine adsorption on Ca-montmorillonite. Colloid Surf A 2011;385:213–18
  • Lv G, Liu L, Li Z, et al. Probing the interactions between chlorpheniramine and 2:1 phyllosilicates. J Colloid Interface Sci 2012;374:218–25
  • Nimkulrat S, Suchiva K, Phinyocheep P, Puttipipatkhachorn S. Influence of selected surfactants on the tackiness of acrylic polymer films. Int J Pharm 2004;287:27–37
  • Leuangsukrerk M, Phupoksakul T, Tananuwong K, et al. Properties of konjac glucomannan-whey protein isolate blend films. Food Sci Technol LEB 2014;59:94–100
  • Li X, Jiang F, Ni X, et al. Preparation and characterization of konjac glucomannan and ethyl cellulose blend films. Food Hydrocolloid 2015;44:229–36
  • Ghebremeskel AN, Vemavarapu C, Lodaya M. Use of surfactants as plasticizers in preparing solid dispersions of poorly soluble API: selection of polymer-surfactant combinations using solubility parameters and testing the processability. Int J Pharm 2007;328:119–29
  • Entwistle CA, Rowe RC. Plasticization of cellulose ethers used in the film coating of tablets. J Pharm Pharmacol 1979;31:269–72
  • Lin S-Y, Lee C-J, Lin Y-Y. Drug-polymer interaction affecting the mechanical properties, adhesion strength and release kinetics of piroxicam-loaded Eudragit E films plasticized with different plasticizers. J Control Release 1995;33:375–81
  • Rao PR, Diwan PV. Permeability studies of cellulose acetate free films for transdermal use: influence of plasticizers. Pharm Acta Helv 1997;72:47–51
  • Silverstein RM, Bassler GC, Morril TC. Infrared spectroscopy. In: Stiefel J, ed. Spectrometric identification of organic compounds. Singapore: John Wiley & Sons; 1991:91--164
  • Pignatello R, Ferro M, Puglisi G. Preparation of solid dispersions of nonsteroidal anti-inflammatory drugs with acrylic polymers and studies on mechanisms of drug-polymer interactions. AAPS PharmSciTech [electronic resource] 2002;3:1–11
  • Glaessl B, Siepmann F, Tucker I, et al. Characterisation of quaternary polymethacrylate films containing tartaric acid, metoprolol free base or metoprolol tartrate. Eur J Pharm Biopharm 2009;73:366–72
  • James MNG, Williams GJB. Structural studies of histamine H1 effector molecules: the crystal structure of the antihistamine drug (+)-chlorpheniramine maleate; [(+)-S-1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpropylamine maleate]. Can J Chem 1974;52:1872–9
  • Madheswaran T, Baskaran R, Yong CS, Yoo BK. Enhanced topical delivery of finasteride using glyceryl monooleate-based liquid crystalline nanoparticles stabilized by cremophor surfactants. AAPS PharmSciTech 2014;15:44–51
  • Papadimitriou SA, Barmpalexis P, Karavas E, Bikiaris DN. Optimizing the ability of PVP/PEG mixtures to be used as appropriate carriers for the preparation of drug solid dispersions by melt mixing technique using artificial neural networks: I. Eur J Pharm Biopharm 2012;82:175–86
  • Papageorgiou GZ, Bikiaris D, Karavas E, et al. Effect of physical state and particle size distribution on dissolution enhancement of nimodipine/PEG solid dispersions prepared by melt mixing and solvent evaporation. AAPS J 2006;8:E623–31
  • Docoslis A, Huszarik KL, Papageorgiou GZ, et al. Characterization of the distribution, polymorphism, and stability of nimodipine in its solid dispersions in polyethylene glycol by micro-Raman spectroscopy and powder X-ray diffraction. AAPS J 2007;9:E361–70
  • Moneghini M, Kikic I, Voinovich D, et al. Processing of carbamazepine-PEG 4000 solid dispersions with supercritical carbon dioxide: preparation, characterisation, and in vitro dissolution. Int J Pharm 2001;222:129–38
  • Zerrouk N, Chemtob C, Arnaud P, et al. In vitro and in vivo evaluation of carbamazepine-PEG 6000 solid dispersions. Int J Pharm 2001;225:49–62
  • Perissutti B, Newton JM, Podczeck F, Rubessa F. Preparation of extruded carbamazepine and PEG 4000 as a potential rapid release dosage form. Eur J Pharm Biopharm 2002;53:125–32
  • Thumma S, ElSohly MA, Zhang S-Q, et al. Influence of plasticizers on the stability and release of a prodrug of Δ9-tetrahydrocannabinol incorporated in poly (ethylene oxide) matrices. Eur J Pharm Biopharm 2008;70:605–14
  • Lecomte F, Siepmann J, Walther M, et al. Polymer blends used for the aqueous coating of solid dosage forms: importance of the type of plasticizer. J Control Release 2004;99:1–13
  • Muschert S, Siepmann F, Leclercq B, et al. Drug release mechanisms from ethylcellulose: PVA-PEG graft copolymer-coated pellets. Eur J Pharm Biopharm 2009;72:130–7

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.