613
Views
1
CrossRef citations to date
0
Altmetric
Research Article

Enhanced skin permeation of 6-methoxy-2-naphthylacetic acid by salt formation

, , &
Pages 359-366 | Received 14 Jan 2014, Accepted 11 Feb 2014, Published online: 27 Mar 2014

References

  • Altman RD. (2010). New guidelines for topical NSAIDs in the osteoarthritis treatment paradigm. Curr Med Res Opin 26:2871–6
  • Arsenijevic L, Arsenijevic V, Horeau A, Jacques J. (1988). Synthesis of 2-acetyl-6-methoxynaphthalene. Org Syn 6:34–6
  • Cheong HA, Choi HK. (2002). Enhanced percutaneous absoption of piroxicam via salt formation with ethanolamines. Pharm Res 19:1375–80
  • Davies NM. (1997). Clinical pharmacokinetics of nabumetone. The dawn of selective cyclo-oxygenase-2 inhibition? Clin Pharmacokinet 33:404–16
  • Evans JM, McMahon AD, McGilchrist MM, et al. (1995a). Topical non-steroidal anti-inflammatory drugs and admission to hospital for upper gastrointestinal bleeding and perforation: a record linkage case-control study. BMJ 311:22–6
  • Evans JM, McGregor E, McMahon AD, et al. (1995b). Non-steroidal anti-inflammatory drugs and hospitalization for acute renal failure. QJM 88:551–7
  • Fang L, Numajiri S, Kobayashi D, Morimoto Y. (2003). The use of complexation with alkanolamines to facilitate skin permeation of mefenamic acid. Int J Pharm 262:13–22
  • Friedel HA, Langtry HD, Buckley MM. (1993). Nabumetone: a reappraisal of its pharmacology and therapeutic use in rheumatic diseases. Drugs 45:131–56
  • Furniss BS, Hannaford JH, Smith PWG, Tachell AR. (1996). Vogel’s text book of practical organic chemistry, 5th edition. Singapore: Longman, 987–1054
  • Gerard C, Mazzenga B. (1991). The transdermal delivery of zwitterionic drugs I: the solubility of zwitterion salts. J Control Rel 16:77–88
  • Ki HM, Choi HK. (2007). The effect of meloxicam/ethanolamine salt formation on percutaneous absorption of meloxicam. Arch Pharm Res 30:215–21
  • Komatsu T, Sakurada T. (2012). Comparision of the efficacy and skin permeability of topical NSAID preparations used in Europe. Eur J Pharm Sci 18:890–5
  • Lee CM, Maibach HI. (2006). Deep percutaneous penetration into muscles and joints. J Pharm Sci 95:1405–13
  • Motsko SP, Rascati KL, Busti AJ, et al. (2006). Temporal relationship between use of NSAIDs, including selective COX-2 inhibitors, and cardiovascular risk. Drug Saf 29:621–32
  • Menassé R, Hedwall PR, Kraetz J, et al. (1978). Pharmacological properties of diclofenac sodium and its metabolites. Scand J Rheumatol 22:5–16
  • Rautio J, Nevalainen T, Taipale H, et al. (2000). Piperazinylalkyl prodrugs of naproxen improve in vitro skin permeation. Eur J Pharm Sci 11:157–63
  • Roberts MS, Cross SE. (1999). Percutaneous absorption of topically applied NSAIDs and other compounds: role of solute properties, skin physiology and delivery system. Inflammopharmacology 7:339–50
  • Singh S, Singh J. (1993). Transdermal drug delivery by passive diffusion and iontophoresis: a review. Med Res Rev 13:569–621
  • Singh P, Roberts MS. (1994). Skin permeability and local tissue concentrations of nonsteroidal anti-inflammatory drugs after topical application. J Pharmacol Exp Ther 268:144–51
  • Suh H, Jun HW, Dzimianski MT, Lu GW. (1997). Pharmacokinetic and local tissue disposition studies of naproxen following topical and systemic administration in dogs and rats. Biopharm Drug Disp 18:623–33
  • Yano T, Nakawaga A, Tsuji M, Noda K. (1986). Skin permeability of various non-steroidal anti-inflammatory drugs in man. Life Sci 39:1043–50

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.