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Research Article

Effect of cocrystallization techniques on compressional properties of caffeine/oxalic acid 2:1 cocrystal

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Pages 55-60 | Received 29 Jun 2011, Accepted 19 Aug 2011, Published online: 10 Oct 2011

References

  • Shan N, Toda F, Jones W. Mechanochemistry and co-crystal formation: Effect of solvent on reaction kinetics. Chem Commun (Camb) 2002;20:2372–2373.
  • Fleischman SG, Kuduva SS, McMahon JA, Moulton B, Walsh RDB, Rodriguez-Hornedo et al. Crystal engineering of the composition of pharmaceutical phases: Multiplecomponent crystalline solids involving carbamazepine. Cryst Growth Des 2003;3:909–919.
  • Childs SL, Mougin P, Stahly B. Screening for solid forms by ultrasound crystallization and cocrystallization using ultrasound. 2005; WO/2005/089375.
  • Trask AV, Motherwell WDS, Jones W. Pharmaceutical cocrystallization: Engineering a remedy for caffeine hydration. Cryst Growth Des 2005;5:1013–1021.
  • McNamara DP, Childs SL, Giordano J, Iarriccio A, Cassidy J, Shet MS et al. Use of a glutaric acid cocrystal to improve oral bioavailability of a low solubility API. Pharm Res 2006;23:1888–1897.
  • Bu Ccaron Ar DK, Macgillivray LR. Preparation and reactivity of nanocrystalline cocrystals formed via sonocrystallization. J Am Chem Soc 2007;129:32–33.
  • Friscic T, Jones W. Recent advances in understanding the mechanism of cocrystal formation via grinding. Cryst Growth Des 2009;9:1621–1637.
  • Friscic T, Childs SL, Rizvic SAA, Jones W. The role of solvent in mechanochemical and sonochemical cocrystal formation: A solubility-based approach for predicting cocrystallisation outcome. Cryst Eng Comm 2009;11:375–522.
  • Aher S, Dhumal R, Mahadik K, Paradkar A, York P. Ultrasound assisted cocrystallization from solution (USSC) containing a non-congruently soluble cocrystal component pair: Caffeine/maleic acid. Eur J Pharm Sci 2010;41:597–602.
  • Dhumal RS, Kelly AL, York P, Coates PD, Paradkar A. Cocrystalization and simultaneous agglomeration using hot melt extrusion. Pharm Res 2010;27:2725–2733.
  • Nokhodchi A, Bolourtchian N, Dinarvand R. Crystal modification of phenytoin using different solvents and crystallization conditions. Int J Pharm 2003;250:85–97.
  • Zhang GG, Henry RF, Borchardt TB, Lou X. Efficient co-crystal screening using solution-mediated phase transformation. J Pharm Sci 2007;96:990–995.
  • Sun CC, Hou H. Improving mechanical properties of caffeine and methyl gallate crystals by cocrystallization. Cryst Growth Des 2008;8:1575–1579.
  • Cassidy AM, Gardner CE, Jones W. Following the surface response of caffeine cocrystals to controlled humidity storage by atomic force microscopy. Int J Pharm 2009;379:59–66.
  • Ruecroft G, Hipkiss D, Ly T, Maxted N, Cains PW. Sonocrystallization: The use of ultrasound for improved industrial crystallization. Org Proc Res Dev 2005;9:923–932.
  • Li H, Li H, Guo Z, Liu Y. The application of power ultrasound to reaction crystallization. Ultrason Sonochem 2006;13:359–363.
  • Luque de Castro MD, Priego-Capote F. Ultrasound-assisted crystallization (sonocrystallization). Ultrason Sonochem 2007;14:717–724.
  • Zeng XM, Martin GP, Marriott C, Pritchard J. Crystallization of lactose from carbopol gels. Pharm Res 2000;17:879–886.
  • Miyasaka E, Kato Y, Hagisawa M, Hirasawa I. Effect of ultrasonic irradiation on the number of acetylsalicylic acid crystals produced under the supersaturated condition and the ability of controlling the final crystal size via primary nucleation. J Cryst Growth 2006;289:324–330.
  • Alderborn G, Nyström C. Studies on direct compression of tablets. IV. The effect of particle size on the mechanical strength of tablets. Acta Pharm Suec 1982;19:381–390.
  • Alderborn G, Nyström C. Studies on direct compression of tablets. III. The effect on tablet strength of changes in particle shape and texture obtained by milling. Acta Pharm Suec 1982;19:147–156.
  • Wong LW, Pilpel N. Effect of particle shape on the mechanical properties of powders. Int J Pharm 1990;59:145–154.
  • Amara N, Ratsimba B, Wilhelm AM, Delmas H. Crystallization of potash alum: Effect of power ultrasound. Ultrason Sonochem 2001;8:265–270.
  • Guo Z, Zhang M, Li H, Wang J, Kougoulos E. Effect of ultrasound on anti-solvent crystallization process. J Cryst Growth 2005;273:555–563.
  • Dhumal RS, Biradar SV, Yamamura S, Paradkar AR, York P. Preparation of amorphous cefuroxime axetil nanoparticles by sonoprecipitation for enhancement of bioavailability. Eur J Pharm Biopharm 2008;70:109–115.
  • Dhumal RS, Biradar SV, Paradkar AR, York P. Ultrasound assisted engineering of lactose crystals. Pharm Res 2008;25:2835–2844.
  • Dhumal RS, Biradar SV, Paradkar AR, York P. Particle engineering using sonocrystallization: Salbutamol sulphate for pulmonary delivery. Int J Pharm 2009;368:129–137.
  • Sun C, Grant DJ. Influence of crystal structure on the tableting properties of sulfamerazine polymorphs. Pharm Res 2001;18:274–280.

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