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Research Article

Optimization and evaluation of pluronic lecithin organogels as a transdermal delivery vehicle for sinomenine

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Pages 535-545 | Received 10 Jan 2015, Accepted 14 Feb 2015, Published online: 11 Mar 2015

References

  • Chen DP, Wong CK, Leung PC, et al. Anti-inflammatory activities of Chinese herbal medicine sinomenine and Liang Miao San on tumor necrosis factor-α-activated human fibroblast-like synoviocytes in rheumatoid arthritis. J Ethnopharmacol 2011;137:457–468
  • Li X, Li X, Zhou Y, et al. Development of patch and spray formulations for enhancing topical delivery of sinomenine hydrochloride. J Pharmacol Sci 2010;99:1790–1799
  • Wang Y, Ma D, Jie Y, et al. SIN can prolong high-risk corneal graft survival in a rat model. Immunotherapy 2012;4:581–586
  • Cheng Y, Zhang J, Hou W, et al. Immunoregulatory effects of sinomenine on the T-bet/GATA-3 ratio and Th1/Th2 cytokine balance in the treatment of mesangial proliferative nephritis. Int Immunopharmacol 2009;9:894–899
  • Zhang XZ, Zhu HD, Meng SF, Pan XG. Preparation of sinomenine microemulsion and its transdermal absorption. Zhongguo Zhong Yao Za Zhi 2007;32:2007–2010
  • Liu ZQ, Jiang ZH, Chan K, et al. Pharmacokinetic interaction of paeoniflorin and SIN: pharmacokinetic parameters and tissue distribution characteristics in rats and protein binding ability in vitro. J Pharm Sci 2005;99:381–391
  • Liu X, Chen T, Liu XS, et al. Penetration effect of ostrich oil as a promising vehicle on transdermal delivery of sinomenine. J Oleo Sci 2013;62:657–664
  • Wang J, Ruan J, Zhang C, et al. Development and evaluation of the sinomenine transdermal patch. Pak J Pharm Sci 2008;21:407–410
  • Song J, Bi HS, Xie XF, et al. Preparation and evaluation of sinomenine hydrochloride in situ gel for uveitis treatment. Int Immunopharmacol 2013;17:99–107
  • Jones M. The history of pluronic lecithin organogel: an interview with Marty Jones, BSPharm, FACA, FIACP. Int J Pharm Comp 2003;7:180–182
  • Franckum J, Ramsay D, Das NG, Das SK. Pluronic lecithin organogel for local delivery of anti-inflammatory drugs. Int J Pharm Comp 2004;8:101–105
  • Morales ME, Clarés B, López-Viota M, et al. Preparation, characterization, and in vitro release of new transdermal methimazole as alternative to oral delivery. Drug Deliv 2009;161:1–10
  • Willimann H, Walde P, Luisi PL, et al. Lecithin organogels as matrix for transdermal transport of drugs. J Pharm Sci 1992;81:871–874
  • Shchipunov YA. Lecithin organogel: a micellar system with unique properties, colloids and surfaces. Colloid Surf A 2001;183–185:541–554
  • Shchipunov YA, Shumilina EV. Lecithin bridging by hydrogen bonds in the organogel. Mater Sci Engg 1995;3:43–50
  • Veena SB, Mohit SP, Dhiraj SC, Sanjay JS. Pluronic lecithin organogel. Asian J Pharm 2008;2:134–138
  • Pandey M, Belgamwar V, Gattani S, et al. Pluronic lecithin organogel as a topical drug delivery system. Drug Deliv 2010;17:38–47
  • Glisson JK, Wood RL, Kyle PB, Cleary JD. Bioavailability of promethazine in a topical pluronic lecithin organogel: a pilot study. Int J Pharm Comp 2005;9:242–246
  • Balata G, Nahas HM, Radwan S. Propolis organogel as a novel topical delivery system for treating wounds. Drug Deliv 2014;21:55–61
  • Agrawal V, Gupta V, Ramteke S, Trivedi P. Preparation and evaluation of tubular micelles of pluronic lecithin organogel for transdermal delivery of sumatriptan. AAPSPharmSciTech 2010;11:1718–1725
  • Manda P, Hargett JK, Vaka SR, Repka MA. Delivery of cefotaxime to the brain via intranasal administration. Drug Dev Ind Pharm 2011;37:1306–1310
  • Holmgaard R, Nielsen JB, Benfeldt E. Microdialysis sampling for investigations of bioavailability and bioequivalence of topically administered drugs: current state and future perspectives. Skin Pharmacol Physiol 2010;23:225–243
  • Ebah L, Brenchley P, Coupes B, Mitra S. A modified in vivo flow variation technique of microdialysis for sampling uremic toxins in the subcutaneous interstitial compartment. Blood Purif 2011;32:96–103
  • Patel DR, Joshi A, Patel HH, Stagni G. Development and in-vivo evaluation of ondansetron gels for transdermal delivery. Drug Dev Ind Pharm 2015. [Epub ahead of print]. doi:10.3109/03639045.2014.925916
  • Zhou WH, He SY, Yang YJ, et al. Formulation, characterization and clinical evaluation of propranolol hydrochloride gel for transdermal treatment of superficial infantile hemangioma. Drug Dev Ind Pharm 2015. [Epub ahead of print]. doi:10.3109/03639045.2014.931968
  • Li SS, Li GF, Liu L, et al. Evaluation of paeonol skin-target delivery from its microsponge formulation: in vitro skin permeation and in vivo microdialysis. PLoS One 2013;8:e79881
  • Pinaki R, Desai PP, Shah RR, Patlolla MS. Dermal microdialysis technique to evaluate the trafficking of surface-modified lipid nanoparticles upon topical application. Pharm Res 2012;29:2587–2600
  • Pandey MS, Belgamwar VS, Surana SJ. Topical delivery of flurbiprofen from pluronic lecithin organogel. Ind J Pharm Sci 2009;71:87–90
  • Krishnaiah YS, Satyanarayana V, Bhasker P. Enhanced percutaneous permeability of nicardipine hydrochloride by carvone across the rat abdominal skin. Drug Dev Ind Pharm 2003;29:191–202
  • Nayak AK, Mohanty B, Sen KK. Comparative evaluation of in vitro diclofenac sodium permeability across excised mouse skin from different common pharmaceutical vehicles. Int J Pharm Tech Res 2010;2:920–930
  • Duangjit S, Opanasopit P, Rojanarata T, Ngawhirunpat T. Characterization and in vitro skin permeation of meloxicam-loaded liposomes versus transfersomes. J Drug Deliv 2011;2011:418–316
  • Yara PC, Vinícius P, Valéria PS, Maria B. In vitro characterization of chitosan gels for buccal delivery of celecoxib: influence of a penetration enhancer. AAPS PharmSciTech 2012;13:101–111
  • Anand B, Pisal SS, Paradkar AR. Applications of organogels in pharmaceuticals. J Sci Ind Res 2001;60:311–318
  • Shchipunov YA, Shumilina EV. Lecithin organogels: role of polar solvent and nature of intermolecular interactions. Colloid J 1996;58:117–125
  • Zhang YT, Shen LN, Zhao JH, Feng NP. Evaluation of psoralen ethosomes for topical delivery in rats by using in vivo microdialysis. Int J Nanomed 2014;9:669–678
  • Zhang YT, Xu YM, Zhang SJ, et al. In vivo microdialysis for the evaluation of transfersomes as a novel transdermal delivery vehicle for cinnamic acid. Drug Dev Ind Pharm 2014;40:301–307
  • Zhang Y, Huo MR, Zhou JP, Xie SF. PKSolver: an add-in program for pharmacokinetic and pharmacodynamic data analysis in Microsoft Excel. Comput Meth Programs Biomed 2010;99:306–314
  • Abdelbary G, Fahmy RH. Diazepam-loaded solid lipid nanoparticles: design and characterization. AAPS PharmSciTech 2009;10:211–219
  • Gonzalez-Mira E, Egea MA, Souto EB, et al. Optimizing flurbiprofen-loaded NLC by central conprosite factorial design for ocular delivery. Nanotechnology 2011;22:045101
  • Mills PC, Cross SE. Regional differences in the in vitro penetration of hydrocortisone through equine skin. J Vet Pharmacol Ther 2006;29:25–30
  • Mills PC, Magnusson BM, Cross SE. Investigation of in vitro transdermal absorption of fentanyl from patches placed on skin samples obtained from various anatomic regions of dogs. Am J Vet Res 2004;65:1697–1700
  • Rohit, Rao C, Krishna G. Effect of captopril and losartan on thermal and chemical induced pain in mice. Indian J Physiol Pharmacol 2006;50:169–174
  • Kulkarni SK, Jain NK. Pharmacological and pharmacokinetics studies on marketed gel formulations of nimesulide. Indian Drugs 2001;38:63–66
  • Ruiz MA, Clares B, Morales ME, et al. Preparation, rheological study, and characterization of an organogel as a system for transdermal release of active principles. Pharm Dev Technol 2007;12:637–644
  • Opdyke DL, Letizia C. Monographs on fragrance raw materials. Food Cosmet Toxicol 1982;20:633–852
  • Amrutiya N, Bajaj A, Madan M. Development of microsponges for topical delivery of mupirocin. AAPS PharmSciTech 2009;10:402–409
  • Benfeldt E. In vivo microdialysis for the investigation of drug levels in the dermis and the effect of barrier perturbation on cutaneous drug penetration. Studies in hairless rats and human subjects. Acta Derm Venereol Suppl (Stockh) 1999;206:1–59
  • Wei H, Wang S, Xu F, et al. Topical bioequivalence of acyclovir creams using dermal microdialysis in pigs: a new model to evaluate bioequivalence for topical formulations. Drug Dev Ind Pharm 2012;38:785–791
  • Shinkai N, Korenaga K, Okumura Y, et al. Microdialysis assessment of percutaneous penetration of ketoprofen after transdermal administration to hairless rats and domestic pigs. Eur J Pharm Biopharm 2011;78:415–421
  • Tettey-Amlalo RN, Kanfer I, Skinner MF, et al. Application of dermal microdialysis for the evaluation of bioequivalence of a ketoprofen topical gel. Eur J Pharm Sci 2009;36:219–225

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