175
Views
4
CrossRef citations to date
0
Altmetric
Research Article

Application of hot-melt extrusion technology for designing an elementary osmotic pump system combined with solid dispersion for a novel poorly water-soluble antidepressant

, , , , , , , & show all
Pages 1006-1014 | Received 26 Mar 2015, Accepted 27 Aug 2015, Published online: 08 Oct 2015

References

  • Tian JW, Jiang WL, Zhong Y, et al.. Preclinical pharmacology of TP1, a novel potent triple reuptake inhibitor with antidepressant properties. Neuroscience 2011;196:124–130
  • Sauer D, Zheng W, Coots LB, McGinity JW. Influence of processing parameters and formulation factors on the drug release from tablets powder-coated with Eudragit L 100-55. Eur J Pharm Biopharm 2007;67:464–475
  • Verma RK, Mishra B, Garg S. Osmotically controlled oral drug delivery. Drug Dev Ind Pharm 2000;26:695–708
  • Rani M, Surana R, Sankar C, Mishra B. Development and biopharmaceutical evaluation of osmotic pump tablets for controlled delivery of diclofenac sodium. Acta Pharm 2003;53:263–273
  • Verma RK, Garg S. Development and evaluation of osmotically controlled oral drug delivery system of glipizide. Eur J Pharm Biopharm 2004;57:513–525
  • Theeuwes F. Elementary osmotic pump. J Pharm Sci 1975;64:1987–1991
  • Zentner GM, Rork GS, Himmelstein KJ. Osmotic flow through controlled porosity films: an approach to delivery of water soluble compounds. J Control Release 1985;2:217–229
  • Herrlich S, Spieth S, Messner S, Zengerle R. Osmotic micropumps for drug delivery. Adv Drug Deliv Rev 2012;64:1617–1627
  • Knezevic Z, Gosak D, Hraste M, et al. Application of hot-melt coating process for designing a lipid based controlled release drug delivery system for highly aqueous soluble drugs. Chem Pharm Bull (Tokyo) 2009;57:464–471
  • Piao H, Liu S, Piao H, et al. Development of an osmotically-driven pellet coated with acrylic copolymers (Eudragit® RS 30 D) for the sustained release of oxymatrine, a freely water soluble drug used to treat stress ulcers (I): in vitro and in vivo evaluation in rabbits. Drug Dev Ind Pharm 2013;39:1230–1237
  • Rao VM, Haslam JL, Stella VJ. Controlled and complete release of a model poorly water-soluble drug, prednisolone, from hydroxypropyl methylcellulose matrix tablets using (SBE)(7m)-beta-cyclodextrin as a solubilizing agent. J Pharm Sci 2001;90:807–816
  • Liu L, Khang G, Rhee JM, Lee HB. Monolithic osmotic tablet system for nifedipine delivery. J Control Release 2000;67:309–322
  • Ozeki T, Yuasa H, Okada H. Controlled release of drug via methylcellulose-carboxyvinylpolymer interpolymer complex solid dispersion. AAPS PharmSciTech 2005;6:E231–E236
  • Tran PH, Tran TT, Park JB, Lee BJ. Controlled release systems containing solid dispersions: strategies and mechanisms. Pharm Res 2011;28:2353–2378
  • Giri TK, Kumar K, Alexander A, et al. A novel and alternative approach to controlled release drug delivery system based on solid dispersion technique. Bull Fac Pharm Cairo U 2012;50:147–159
  • Vithani K, Maniruzzaman M, Slipper IJ, et al. Sustained release solid lipid matrices processed by hot-melt extrusion (HME). Colloids Surf B Biointerfaces 2013;110:403–410
  • Maniruzzaman M, Rana MM, Boateng JS, et al. Dissolution enhancement of poorly water-soluble APIs processed by hot-melt extrusion using hydrophilic polymers. Drug Dev Ind Pharm 2013;39:218–227
  • Deng W, Majumdar S, Singh A, et al. Stabilization of fenofibrate in low molecular weight hydroxypropylcellulose matrices produced by hot-melt extrusion. Drug Dev Ind Pharm 2013;39:290–298
  • Zhang SQ, Rahman Z, Thumma S, et al. Development and evaluation of a pH-dependent sustained release tablet for irritable bowel syndrome. Drug Dev Ind Pharm 2009;35:57–64
  • Keen JM, McGinity JW. Melt extruded controlled release dosage forms. In: Repka MA, Langley N, DiNunzio J, eds. Melt extrusion, materials, AAPS Advances in the pharmaceutical sciences series 9. New York: Springer; 2013:243–260
  • Zhu Y, Shah NH, Malick AW, et al. Controlled release of a poorly water-soluble drug from hot-melt extrudates containing acrylic polymers. Drug Dev Ind Pharm 2006;32:569–583
  • Kanagale P, Patel V, Venkatesan N, et al. Pharmaceutical development of solid dispersion based osmotic drug delivery system for nifedipine. Curr Drug Deliv 2008;5:306–311
  • Panda RR, Tiwary AK. Hot melt granulation: a facile approach for monolithic osmotic release tablets. Drug Dev Ind Pharm 2012;38:447–461
  • Sakurai A, Sakai T, Sako K, Maitani Y. Polymer combination increased both physical stability and oral absorption of solid dispersions containing a low glass transition temperature drug: physicochemical characterization and in vivo study. Chem Pharm Bull (Tokyo) 2012;60:459–464
  • Shah S, Maddineni S, Lu J, Repka MA. Melt extrusion with poorly soluble drugs. Int J Pharm 2013;453:233–252
  • Xie Y, Lu Y, Qi J, et al. Synchronized and controlled release of multiple components in silymarin achieved by the osmotic release strategy. Int J Pharm 2013;441:111–120

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.