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Research Article

Matrix-type transdermal films to enhance simvastatin ex vivo skin permeability

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Pages 492-499 | Received 31 May 2015, Accepted 22 Sep 2015, Published online: 29 Oct 2015

References

  • World-Health-Organization. WHO model list of essential medicines: 18th list. 2013
  • Martindale W, Sweetman SC. Martindale: the complete drug reference. London: Pharmaceutical press; 1999
  • Jun SW, Kim MS, Kim J-S, et al. Preparation and characterization of simvastatin/hydroxypropyl-β-cyclodextrin inclusion complex using supercritical antisolvent (SAS) process. Eur J Pharmaceut Biopharmaceut 2007;66:413–421
  • Prausnitz MR, Mitragotri S, Langer R. Current status and future potential of transdermal drug delivery. Nat Rev Drug Discov 2004;3:115–124
  • Kim KS, Simon L. Modeling and design of transdermal drug delivery patches containing an external heating device. Comput Chem Eng 2011;35:1152–1163
  • Ammar H, Ghorab M, El-Nahhas S, Higazy I. Proniosomes as a carrier system for transdermal delivery of tenoxicam. Int J Pharm 2011;405:142–152
  • El-Say KM, Ahmed TA, Badr-Eldin SM, et al. Enhanced permeation parameters of optimized nanostructured simvastatin transdermal films: ex vivo and in vivo evaluation. Pharm Dev Technol 2015;20:919–926
  • Singh B, Kumar R, Ahuja N. Optimizing drug delivery systems using systematic “design of experiments.” Part I: fundamental aspects. Crit Rev Ther Drug Carrier Syst 2005;22:27–105
  • Plackett RL, Burman JP. The design of optimum multifactorial experiments. Biometrika 1946;33:305–325
  • Rowe RC, Sheskey PJ, Quinn ME, et al. Handbook of pharmaceutical excipients: London: Pharmaceutical press; 2009
  • Naseera K, Sajeeth C, Santhi K. Formulation, optimization and evaluation of matrix type of transdermal system of simvastatin using permeation enhancers. Int J Curr Pharm Res 2012;4:79–87
  • Shinde AJ, Garala KC, More HN. Development and characterization of transdermal therapeutics system of tramadol hydrochloride. Asian J Pharm 2008;2:265
  • Jayaprakash S, Halith SM, Firthouse PM, Nagarajan M. Preparation and evaluation of celecoxib transdermal patches. Pak J Pharm Sci 2010;23:279–283
  • Mukherjee B, Mahapatra S, Gupta R, et al. A comparison between povidone-ethylcellulose and povidone-eudragit transdermal dexamethasone matrix patches based on in vitro skin permeation. Eur J Pharm Biopharm 2005;59:475–483
  • Ahmed TA, Khalid M. Development of alginate-reinforced chitosan nanoparticles utilizing W/O nanoemulsification/internal crosslinking technique for transdermal delivery of rabeprazole. Life Sci 2014;110:35–43
  • Dixit RP, Barhate CR, Padhye SG, et al. Stability indicating RP-HPLC method for simultaneous determination of simvastatin and ezetimibe from tablet dosage form. Indian J Pharm Sci. 2010;72:204–210
  • Murtaza G. Solubility enhancement of simvastatin: a review. Acta Pol Pharm 2012;69:581–590
  • Siepmann J, Ainaoui A, Vergnaud J, Bodmeier R. Calculation of the dimensions of drug-polymer devices based on diffusion parameters. J Pharm Sci 1998;87:827–832
  • Langer R, Peppas N. Chemical and physical structure of polymers as carriers for controlled release of bioactive agents: a review. J Macromol Sci R M C 1983;23:61–126
  • Ouano A, Carothers J. Dissolution dynamics of some polymers: solvent‐polymer boundaries. Polym Eng Sci 1980;20:160–166
  • Lin SY, Lee CJ, Lin YY. Drug-polymer interaction affecting the mechanical properties, adhesion strength and release kinetics of piroxicam-loaded Eudragit E films plasticized with different plasticizers. J Control Release 1995;33:375–381
  • Mali S, Sakanaka L, Yamashita F, Grossmann M. Water sorption and mechanical properties of cassava starch films and their relation to plasticizing effect. Carbohydr Polym 2005;60:283–289
  • Elshafeey AH, Hamza YE, Amin SY, Zia H. In vitro transdermal permeation of fenoterol hydrobromide. J Adv Res 2012;3:125–132
  • Rujivipat S, Bodmeier R. Moisture plasticization for enteric Eudragit® L30D-55-coated pellets prior to compression into tablets. Eur J Pharm Biopharm 2012;81:223–229
  • Pichayakorn W, Suksaeree J, Boonme P, et al. Deproteinized natural rubber film forming polymeric solutions for nicotine transdermal delivery. Pharm Dev Technol 2013;18:1111–1121
  • Bodmeier R, Paeratakul O. Mechanical properties of dry and wet cellulosic and acrylic films prepared from aqueous colloidal polymer dispersions used in the coating of solid dosage forms. Pharmaceut Res 1994;11:882–888
  • Chen YC, Lee LW, Ho HO, et al. Evaluation of water uptake and mechanical properties of blended polymer films for preparing gas-generated multiple-unit floating drug delivery systems. J Pharm Sci 2012;101:3811–3822
  • Hung SF, Hsieh CM, Chen YC, et al. Characterizations of plasticized polymeric film coatings for preparing multiple-unit floating drug delivery systems (muFDDSs) with controlled-release characteristics. PLoS One 2014;9:e100321

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