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Research Article

Synthesis of some thiazolyl aminobenzothiazole derivatives as potential antibacterial, antifungal and anthelmintic agents

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Pages 22-28 | Received 23 Aug 2009, Accepted 13 Dec 2009, Published online: 21 Jan 2011

References

  • Marrero-Ponce Y, Castillo-Garit JA, Olazabal E, Serrano HS, Morales A, Castanedo N, Ibarra-Velarde F, Huesca-Guillen D, Sanchez Am, Torrens F, Castro EA. Atom, atom-type and total molecular linear indices as a promising approach for bioorganic and medicinal chemistry: theoretical and experimental assessment of a novel method for virtual screening and rational design of new lead anthelmintic. Bioorg Med Chem 2005;13:1005–1020.
  • Ducray P, Gauvry N, Pantrat F, Goebel T, Frechtel J, Desaules Y, Weber SS, Bouvier J, Wagner T, Froelich O, Kaminsky R. Discovery of amino-acetonitrile derivatives, a new class of synthetic anthelmintic compounds. Bioorg Med Chem Lett 2008;18:2935–2938.
  • Cruz MC, Bartlett MS, Edlind TD. In vitro susceptibility of the opportunistic fungus Cryptococcus neoformans to anthelmintic benzimidazoles. Antimicrob Agents Chemother 1994;38:378–380.
  • Davyt D, Entz W, Fernandez R, Mariezcurrena R, Mombru AW, Saldane J, Dominguez L, Coll J, Manta E. A new indole derivative from the red algae Chondria atropurpurea. Isolation, structure determination and anthelmintic activity. J Nat Prod 1998;61:1560–1563.
  • Ananda Kumar CS, Vinaya K, Chandra JN, Thimmegowda NR, Prasad SB, Sadashiva CT, Rangappa KS. Synthesis and antimicrobial studies of novel 1-benzhydryl-piperazine sulfonamide and carboxamide derivatives. J Enz Inhib Med Chem 2008;23:462–469.
  • Turan-Zitouni G, Demirayak S, Ozdemir A, Kaplancikh ZA, Yildiz MT. Synthesis of some 2-[(benzazole-2-yl)thioacetylamino]thiazole derivatives and their antimicrobial activity and toxicity. Eur J Med Chem 2003;39:267–272.
  • Gunawardana GP, Khomoto S, Gunasekara SP, McConnell OJ, Koehn FE. Dercitine, a new biologically active acridine alkaloid from a deep water marine sponge, Dercitus sp. J Am Chem Soc 1988;110:4856–4858.
  • Chavan AA, Pai NR. Synthesis and antimicrobial screening of 5-arylidene-2-imino-4-thiazolidinones. ARKIVOC 2007;16:148–155.
  • Bhusari KP, Amnerkar ND, Khedekar PB, Kale MK, Bhole RP. Synthesis and in vitro antimicrobial activity of some 4-amino-N-(1,3-benzothiazol-2-yl)benzene- sulphonamide derivatives. Asian J Res Chem 2008;1:53–57.
  • Vernon V, David R. Quinoxaline and adducts useful as anthelmintics. US Patent 1986; 4629790.
  • Bhusari KP, Khedekar PB, Umathe SN, Bahekar RH, Rao ARR. Synthesis of 8-bromo-9-substituted-1,3-benzothiazolo-[5,1-b]-1,3,4-triazoles and their anthelmintic activity. Indian J Heterocycl Chem 2000;9:275–278.
  • Mahran MA, William S, Ramzy F, Sembel AM. Synthesis and in vitro evaluation of new benzothiazole derivatives as schistosomicidal agents. Molecules 2007;12:622–633.
  • Russo F, Romeo G, Santagati NA, Caruso A, Cutuli V, Amore D. Synthesis of new thienopyrimidobenzothiazoles and thienopyrimidobenzoxazoles with analgesic and anti-inflammatory properties. Eur J Med Chem 1994;29:569–578 .
  • Caleta I, Grdisa M, Sermek D, Cetina M, Kulenovic V, Pavelic K, Zamola G. Synthesis, crystal structure and antiproliferative evaluation of some new substituted benzothiazoles and styrylbenzothiazoles. II Farmaco 2004;59:297–305.
  • Amnerkar ND, Bhusari KP. Synthesis, anticonvulsant activity and 3D-QSAR study of some prop-2-eneamido and 1-acetyl-pyrazolin derivatives of aminobenzothiazole. Eur J Med Chem 2010;45:149–159.
  • Siddiqui N, Rana A, Khan S, Bhat M, Haque S. Synthesis of benzothiazole semicarbazones as novel anticonvulsants-The role of hydrophobic domain. Bioorg Med Chem Lett 2007;17:4178–4182.
  • Walczynski K, Guryn R, Zuiderveld OP, Timmerma H. Non-imidazole histamine H3 ligands. Part I. Synthesis of 2-(1-piperazinyl) and 2-(hexahydro-1H-1,4-diazepin-1-yl)benzothiazole derivatives as H3 anatagonists with H1 blocking activities. II Farmaco 1999;54:684–694.
  • Khedekar PB, Bahekar RH, Chopade RS, Umathe SN, Rao ARR, Bhusari KP. Synthesis and anti-inflammatory activity of alkyl/arylidene-2-aminobenzothiazoles and 1-benzothiazol-2-yl-3-chloro-4-substituted-azetidine-2-ones. Arzneim-Forsch/ Drug Res 2003;9:640–647.
  • Mahler G, Serra G, Dematteis S, Saldana J, Dominguez L, Manta E. Synthesis and biological evaluation of simplified mycothiazole analogues. Bioorg Med Chem Lett 2006;16:1309–1311.
  • Pawar NS, Dalal DS, Shimpi SR, Mahulikar PP. Studies of antimicrobial activity of N-alkyl and N-acyl 2-(4-thiazolyl)-1H-benzimidazoles. Eur J Pharm Sci 2004;21:115–118.
  • Papadopoulou C, Geronikaki A, Hadjipavlou-Litina D. Synthesis and biological evaluation of new thiazolyl/benzothiazolyl-amides, derivative of 4-phenyl-piperazine. II Farmaco 2005;60:969–973.
  • Jones RN, Barry AL, Gavan TL, Washington JA. Susceptibility tests: Microdilution and macrodilution broth procedures. In: Lennette EH, Balows A, Hausler WJ, Shadomy HJ, eds. A Manual of clinical microbiology. Washington DC: ASM, 1991:1105–1112.
  • Khan ZK. In vitro and vivo screening techniques for bioactivity screening and evaluation. In: Proceeding Int. Workshop UNIDO-CDRI, 1997:210–211.
  • Poojary B, Belagali SL. Synthetic studies on cyclic octapeptides: Yunnanin F and Hymenistatin. Eur J Med Chem 2005;40:407–412.
  • Jimonet P, Audiau F, Barreau M, Blanchard J, Boireau A, Bour Y, Colno M, Doble A, Doerflinger G, Huu C, Donat M, DuchesneJ Ganil, P, Gurmy C, Honor E, Just B, KerphiriqueR Gontier, S, Hubert P, Laduron P, Blevec J, Meunier M, Miquet J, Nemecek C, Pasquet M, Piot O, Pratt J, Rataud J, Reibaud M, Stutzmann J, Migani S. Riluzole Series. Synthesis and in vitro “Antiglutamate” activity of 6-substituted-2-benzothiazolamines and 3-substituted-2-imino-benzothiazolines. J Med Chem 1999;42 2828–2843.
  • Mahran MA, William S, Ramzy F, Sembel AM. Synthesis and in vitro evaluation of new benzothiazole derivatives as schistosomicidal agents. Molecules 2007;12:622–633.

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