Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 26, Issue 1 (2011)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 26, Issue 1 (2011)

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Research Article

Article
Pharmacological significance of triazole scaffold
Rajeev Kharb, Prabodh Chander Sharma & Mohammed Shahar Yar
Pages: 1-21
Published online: 28 Jun 2010
AbstractforPharmacological significance of triazole scaffold | Full Text | References | PDF (1.5 MB)
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Article
Synthesis of some thiazolyl aminobenzothiazole derivatives as potential antibacterial, antifungal and anthelmintic agents
Nikhil D. Amnerkar & Kishore P. Bhusari
Pages: 22-28
Published online: 21 Jan 2011
AbstractforSynthesis of some thiazolyl aminobenzothiazole derivatives as potential antibacterial, antifungal and anthelmintic agents | Full Text | References | PDF (620.7 KB)
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Article
Theoretical studies on the molecular basis of HIV-1RT/NNRTIs interactions
Panita Decha, Pathumwadee Intharathep, Thanyarat Udommaneethanakit, Pornthep Sompornpisut, Supot Hannongbua, Peter Wolschann & Vudhichai Parasuk
Pages: 29-36
Published online: 28 Jun 2010
AbstractforTheoretical studies on the molecular basis of HIV-1RT/NNRTIs interactions | Full Text | References | PDF (1,021.6 KB)
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Article
Synthesis and antiproliferative activities against Hep-G2 of salicylanide derivatives: potent inhibitors of the epidermal growth factor receptor (EGFR) tyrosine kinase
Zhen-Wei Zhu, Lei Shi, Xiao-Ming Ruan, Ying Yang, Huan-Qiu Li, Suo-Ping Xu & Hai-Liang Zhu
Pages: 37-45
Published online: 28 Jun 2010
AbstractforSynthesis and antiproliferative activities against Hep-G2 of salicylanide derivatives: potent inhibitors of the epidermal growth factor receptor (EGFR) tyrosine kinase | Full Text | References | PDF (767.1 KB)
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Article
Nantenine as an acetylcholinesterase inhibitor: SAR, enzyme kinetics and molecular modeling investigations
Stevan Pecic, Marie A. McAnuff & Wayne W. Harding
Pages: 46-55
Published online: 28 Jun 2010
AbstractforNantenine as an acetylcholinesterase inhibitor: SAR, enzyme kinetics and molecular modeling investigations | Full Text | References | PDF (1.1 MB)
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Article
Synthesis, spectral analysis and in vitro microbiological evaluation of novel ethyl 4-(naphthalen-2-yl)-2-oxo-6-arylcyclohex-3-enecarboxylates and 4,5-dihydro-6-(napthalen-2-yl)-4-aryl-2H-indazol-3-ols
V. Kanagarajan, J. Thanusu & M. Gopalakrishnan
Pages: 56-66
Published online: 08 Feb 2011
AbstractforSynthesis, spectral analysis and in vitro microbiological evaluation of novel ethyl 4-(naphthalen-2-yl)-2-oxo-6-arylcyclohex-3-enecarboxylates and 4,5-dihydro-6-(napthalen-2-yl)-4-aryl-2H-indazol-3-ols | Full Text | References | PDF (702.6 KB)
  • 473 Views
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Article
A facile microwave assisted green chemical synthesis of novel piperidino 2-thioxoimidazolidin-4-ones and their in vitro microbiological evaluation
V. Kanagarajan, J. Thanusu & M. Gopalakrishnan
Pages: 67-77
Published online: 28 Jun 2010
AbstractforA facile microwave assisted green chemical synthesis of novel piperidino 2-thioxoimidazolidin-4-ones and their in vitro microbiological evaluation | Full Text | References | PDF (731.1 KB)
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Article
Prediction of the relationship between the structural features of andrographolide derivatives and α-glucosidase inhibitory activity: A quantitative structure-activity relationship (QSAR) Study
NS Hari Narayana Moorthy, Maria J Ramos & Pedro A Fernandes
Pages: 78-87
Published online: 20 Dec 2010
AbstractforPrediction of the relationship between the structural features of andrographolide derivatives and α-glucosidase inhibitory activity: A quantitative structure-activity relationship (QSAR) Study | Full Text | References | PDF (1 MB) | Supplemental
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Article
Antioxidative iridoid glycosides from the sky flower (Duranta repens Linn)
Fozia Ijaz, Azhar Ul Haq, Ijaz Ahmad, Nisar Ahmad, Javid Hussain & Sibao Chen
Pages: 88-92
Published online: 08 Feb 2011
AbstractforAntioxidative iridoid glycosides from the sky flower (Duranta repens Linn) | Full Text | References | PDF (603.5 KB)
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Article
Changes of rat plasma total low molecular weight antioxidant level after tabun exposure and consequent treatment by acetylcholinesterase reactivators
Miroslav Pohanka, Jana Zdarova Karasova, Kamil Musilek, Kamil Kuca, Young-Sik Jung & Jiri Kassa
Pages: 93-97
Published online: 22 Jun 2010
AbstractforChanges of rat plasma total low molecular weight antioxidant level after tabun exposure and consequent treatment by acetylcholinesterase reactivators | Full Text | References | PDF (615.2 KB)
  • 399 Views
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Article
Substituted benzenediol Schiff bases as promising new anti-glycation agents
M. Iqbal Choudhary, Ghulam Abbas, Saqib Ali, Shaukat Shuja, Nasir Khalid, Khalid M. Khan, Atta-ur-Rahman & Fatima Z. Basha
Pages: 98-103
Published online: 28 Jun 2010
AbstractforSubstituted benzenediol Schiff bases as promising new anti-glycation agents | Full Text | References | PDF (708.1 KB)
  • 988 Views
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Article
Synthesis and characterisation of two novel proton transfer compounds and their inhibition studies on carbonic anhydrase isoenzymes
Cengiz Yenikaya, Musa Sarı, Metin Bülbül, Halil İlkimen, Burcu Çınar & Orhan Büyükgüngör
Pages: 104-114
Published online: 23 Sep 2010
AbstractforSynthesis and characterisation of two novel proton transfer compounds and their inhibition studies on carbonic anhydrase isoenzymes | Full Text | References | PDF (1.1 MB)
  • 904 Views
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Article
Analysis of highly potent amidine containing inhibitors of serine proteases and their N-hydroxylated prodrugs (amidoximes)
Joscha Kotthaus, Torsten Steinmetzer, Andreas van de Locht & Bernd Clement
Pages: 115-122
Published online: 28 Jun 2010
AbstractforAnalysis of highly potent amidine containing inhibitors of serine proteases and their N-hydroxylated prodrugs (amidoximes) | Full Text | References | PDF (1.2 MB)
  • 2030 Views
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Article
Synthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles
Eskandar Alipour, Saeed Emami, Azadeh Yahya-Meymandi, Maryam Nakhjiri, Farnaz Johari, Sussan K. Ardestani, Fatemeh Poorrajab, Maryam Hosseini, Abbas Shafiee & Alireza Foroumadi
Pages: 123-128
Published online: 28 Jun 2010
AbstractforSynthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles | Full Text | References | PDF (949.3 KB)
  • 704 Views
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Article
Development of a robust QSAR model to predict the affinity of pyrrolidine analogs for dipeptidyl peptidase IV (DPP- IV)
Sarvesh Paliwal, Deepika Seth, Divya Yadav, Rakesh Yadav & Shailendra Paliwal
Pages: 129-140
Published online: 08 Feb 2011
AbstractforDevelopment of a robust QSAR model to predict the affinity of pyrrolidine analogs for dipeptidyl peptidase IV (DPP- IV) | Full Text | References | PDF (1.1 MB)
  • 738 Views
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Article
Design, synthesis and pharmacological evaluation of novel azole derivatives of aryl acetic acid as anti-inflammatory and analgesic agents
Mohammad Amir, Khalid Saifullah & Wasim Akhter
Pages: 141-148
Published online: 28 Jun 2010
AbstractforDesign, synthesis and pharmacological evaluation of novel azole derivatives of aryl acetic acid as anti-inflammatory and analgesic agents | Full Text | References | PDF (628.5 KB)
  • 837 Views
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Article
Bis dihydropyrimidine: synthesis and antimycobacterial activity
Mohamed Ashraf Ali, Elumalai Manogaran, Jeyabalan Govindasamy, Velmurugan Sellappan & Suresh Pandian
Pages: 149-153
Published online: 28 Jun 2010
AbstractforBis dihydropyrimidine: synthesis and antimycobacterial activity | Full Text | References | PDF (606.5 KB)
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