Synthesis and analgesic activity of some acetamide derivatives

References

• Moore ND. In search of an ideal analgesic for common acute pain. Acute Pain 2009;11:129–137.
   Google Scholar
• Buschmann H, Christoph T, Friderichs E, Maul C, Sundermann B. Analgesics: From chemistry and pharmacology to clinical application. Weinheim: Wiley-VCH Germany, 2002: pp. 1–264.
   Google Scholar
• Turunen JH, Mäntyselkä PT, Kumpusalo EA, Ahonen RS. Frequent analgesic use at population level: Prevalence and patterns of use. Pain 2005;115:374–381.
   Google Scholar
• Simmons DL, Botting RM, Hla T. Cyclooxygenase isozymes: The biology of prostaglandin synthesis and inhibition. Pharmacol Rev 2004;56:387–437.
   PubMed Web of Science ®Google Scholar
• Dannhardt G, Laufer S. Structural approaches to explain the selectivity of COX-2 inhibitors: Is there a common pharmacophore? Curr Med Chem 2000;7:1101–1112.
   PubMed Web of Science ®Google Scholar
• Moore A, Collins S, Carroll D, McQuay H. Paracetamol with and without codeine in acute pain: A quantitative systematic review. Pain 1997;70:193–201.
   PubMed Web of Science ®Google Scholar
• Onkol T, Dogruer DS, Ito S, Sahin MF. Synthesis and antinociceptive activity of (5-chloro-2-benzothiazolinon-3-yl)acetamide derivatives. Arch Pharm (Weinheim) 2000;333:337–340.
   Google Scholar
• Pilli HG, Ozkanli F, Safak C, Erdogan H, Unlü S, Gümüsel B et al. 2-(6-Acyl-2-benzoxazolinone-3-yl)acetamide and acetonitrile derivatives with analgesic activities. Pharmazie 1994;49:63–64.
   Google Scholar
• Dogruer DS, Unlü S, Yesilada E, Fethi Sahin M. N-(2-pyridinyl)-2-[2(3H)-benzazolone-3-yl]acetamides: Synthesis, antinociceptive and anti-inflammatory activity. Farmaco 1997;52:745–750.
   Google Scholar
• Juby PF, Hudyma TW, Brown M. Preparation and antininflammatory properties of some 5-(2-anilinophenyl)tetrazoles. j Med Chem 1968;11:111–117.
   PubMedGoogle Scholar
• Bachar SC, Lahiri SC. Synthesis of chloro and bromo substituted 5-(indan-1′-yl)tetrazoles and 5-(indan-1′-yl)methyltetrazoles as possible analgesic agents. Pharmazie 2004;59:435–438.
   PubMed Web of Science ®Google Scholar
• Ciapetti P, Giethlen B. Molecular variations based on isosteric replacements. In: Wermuth CM (ed.). The Practice of Medicinal Chemistry, Burlington: Academic Press USA, 2008: pp. 290–342.
   Google Scholar
• Rajasekaran A, Thampi PP. Synthesis and analgesic evaluation of some 5-[β-(10-phenothiazinyl)ethyl]-1-(acyl)-1,2,3,4-tetrazoles. Eur j Med Chem 2004;39:273–279.
   PubMed Web of Science ®Google Scholar
• Vicini P, Amoretti L, Barocelli E, Chiavarini M, Impicciatore M. Synthesis and anti-inflammatory, antipyretic and analgesics properties of 5-(1,2-benzisothiazolyl)tetrazoles. Farmaco Sci 1986;41:111–118.
   PubMedGoogle Scholar
• Shanmugapandiyan P, Ramesh A. Synthesis and biological applications of certain 1-acetamido-(benzothiazol-2′-yl)-5-aryltetrazole and benzothiazol-2′-yl-1-ethylamine-5-aryltetrazoles. J Pharm Chem 2008;2:169–173.
   Google Scholar
• Paramashivappa R, Phani Kumar P, Subba Rao PV, Srinivasa Rao A. Design, synthesis and biological evaluation of benzimidazole/benzothiazole and benzoxazole derivatives as cyclooxygenase inhibitors. Bioorg Med Chem Lett 2003;13:657–660.
   PubMed Web of Science ®Google Scholar
• Yous S, Poupaert JH, Chavatte P, Espiard JG, Caignard DH, Lesieur D. Synthesis and pharmacological evaluation of analgesic 6-substituted 2(3H)-benzothiazolones. Drug Des Discov 2001;17:331–336.
   Google Scholar
• Gökce M, Cakir B, Erol K, Sahin MF. Synthesis and antinociceptive activity of [(2-oxobenzothiazolin-3-yl)methyl]-4-alkyl/aryl-1,2,4-triazoline-5-thiones. Arch Pharm (Weinheim) 2001;334:279–283.
   PubMed Web of Science ®Google Scholar
• Bahekar SS, Shinde DB. Synthesis and anti-inflammatory activity of [2-(benzothiazol-2-ylimino)-4-oxo-3-phenylthiazolidin-5-yl]-acetic acid derivatives. J Korean Chem Soc 2003;47:237–240.
   Google Scholar
• Bhargava PN, Ram P. Synthesis of local anesthetics. Bull Chem Soc Japan 1965;38:339–341.
   Google Scholar
• Connell RD, Lease TG, Ladouceur GH, Osterhout MH. α-Alkoxy- and α-thioalkoxyamide neuropeptide Y NPY5 receptor antagonists and therapeutic methods using them. US Patent 1999;5939462A 19990817.
   Google Scholar
• Kaplancikli ZA, Turan-Zitouni G, Ozdemir A, Can O, Chevallet P. Synthesis and antinociceptive activities of some pyrazoline derivatives. Eur J Med Chem 2009;44:2606–2610.
   PubMed Web of Science ®Google Scholar
• Can OD, Ozkay UD, Oztürk N, Oztürk Y. Effects of hawthorn seed and pulp extracts on the central nervous system. Pharm Biol 2010;48:924–931.
   PubMed Web of Science ®Google Scholar
• D’Amour FE, Smith DL. A method for determining loss of pain sensation. J Pharmacol Exp Ther 1941;72:74–79.
   Google Scholar
• Adeyemi OO, Okpo SO, Okpaka O. The analgesic effect of the methanolic extract of Acanthus montanus. J Ethnopharmacol 2004;90:45–48.
   PubMed Web of Science ®Google Scholar
• Oztürk N, Baser KH, Aydin S, Oztürk Y, Calis I. Effects of Gentiana lutea ssp. symphyandra on the central nervous system in mice. Phytother Res 2002;16:627–631.
   PubMed Web of Science ®Google Scholar
• Gabra BH, Sirois P. Beneficial effect of chronic treatment with the selective bradykinin B1 receptor antagonists, R-715 and R-954, in attenuating streptozotocin-diabetic thermal hyperalgesia in mice. Peptides 2003;24:1131–1139.
   PubMed Web of Science ®Google Scholar
• Wong CH, Dey P, Yarmush J, Wu WH, Zbuzek VK. Nifedipine-induced analgesia after epidural injection in rats. Anesth Analg 1994;79:303–306.
   PubMed Web of Science ®Google Scholar
• De Souza MM, Pereira MA, Ardenghi JV, Mora TC, Bresciani LF, Yunes RA et al. Filicene obtained from Adiantum cuneatum interacts with the cholinergic, dopaminergic, glutamatergic, GABAergic, and tachykinergic systems to exert antinociceptive effect in mice. Pharmacol Biochem Behav 2009;93:40–46.
   PubMed Web of Science ®Google Scholar
• Ikeda Y, Ueno A, Naraba H, Oh-ishi S. Involvement of vanilloid receptor VR1 and prostanoids in the acid-induced writhing responses of mice. Life Sci 2001;69:2911–2919.
   PubMed Web of Science ®Google Scholar